1498300-31-4

TNKS1/2-IN-1 is a potent tankyrase TNKS1/2 inhibitor with pIC50s ranging from 7.1-8.2. TNKS1/2-IN-1 can be used for research of cancer, fibrosis, and other hyperproliferative diseases[1].

[1] Keenan Richard M, et al. Preparation of quinazolinediones as tankyrase inhibitors for the treatment of cancer: World Intellectual Property Organization, WO2013177349 A2 2013-11-28.