IDO1-IN-12 is a potent and orally available IDO1 inhibitor.
References
[1] Pu Q, et al. Discovery of Potent and Orally Available Bicyclo[1.1.1]pentane-Derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors. ACS Med Chem Lett. 2020 Jul 15;11(8):1548-1554. DOI:10.1021/acsmedchemlett.0c00195