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Agonist Inhibitors
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- Structure:

- Chemical Name:Sarecycline Hydrochloride
- CAS:1035979-44-2
- MF:C24H30ClN3O8
- Structure:

- Chemical Name:KML-29
- CAS:1380424-42-9
- MF:C24H21F6NO7
- Structure:

- Chemical Name:4H-1,2,4-Triazole-4-carboxaMide, 1-(2,4-dichlorophenyl) -N-(2,4-difluorophenyl)-1,5-dihydro-N-(1-Methylethyl)- 5-oxo-
- CAS:212201-70-2
- MF:C18H14Cl2F2N4O2
- Structure:

- Chemical Name:Relugolix
- CAS:737789-87-6
- MF:C29H27F2N7O5S
- Structure:

- Chemical Name:VTX-2337
- CAS:926927-61-9
- MF:C28H34N4O2
- Structure:

- Chemical Name:TUG-770
- CAS:1402601-82-4
- MF:C19H14FNO2
- Structure:

- Chemical Name:AMD 070 hydrochloride
- CAS:880549-30-4
- MF:C21H28ClN5
- Structure:

- Chemical Name:Azaphenonxazine dihydrochloride Monohydrate
- CAS:63302-99-8
- MF:C16H23Cl2N5O2
- Structure:

- Chemical Name:CCT 241533 hydrochloride
- CAS:1431697-96-9
- MF:C23H28ClFN4O4
- Structure:

- Chemical Name:CX 6258 hydrochloride hydrate
- CAS:1353858-99-7
- MF:C26H27Cl2N3O4
- Structure:

- Chemical Name:LDE-225 Diphosphate
- CAS:1218778-77-8
- MF:C26H32F3N3O11P2
- Structure:

- Chemical Name:LY-2795050
- CAS:1346133-08-1
- MF:C23H22ClN3O2
- Structure:

- Chemical Name:SodiuM Channel inhibitor 1
- CAS:1198117-23-5
- MF:C24H19F4N3O3
- Structure:

- Chemical Name:Tipiracil hydrochloride
- CAS:183204-72-0
- MF:C9H12Cl2N4O2
- Structure:

- Chemical Name:CEP-28122
- CAS:1022958-60-6
- MF:C28H35ClN6O3
- Structure:

- Chemical Name:HMN 176
- CAS:173529-10-7
- MF:C20H18N2O4S
- Structure:

- Chemical Name:HM 30181A
- CAS:849675-66-7
- MF:C38H36N6O7
- Structure:

- Chemical Name:CTEP Derivative
- CAS:802906-73-6
- MF:C18H13ClFN3
- Structure:

- Chemical Name:1H-Isoindole-1,3(2H)-dione, 5-[5-[[3-(4-broMophenyl)-2-iMino-4-oxo-5-thiazolidinylidene]Methyl]-2-furanyl]-
- CAS:1420071-30-2
- MF:C22H12BrN3O4S
- Structure:

- Chemical Name:PF 04995274
- CAS:1331782-27-4
- MF:C23H32N2O6
- Structure:

- Chemical Name:AC710
- CAS:1351522-04-7
- MF:C31H42N6O4
- Structure:

- Chemical Name:AgoMelatine (hydrochloride)
- CAS:1176316-99-6
- MF:C15H18ClNO2
- Structure:

- Chemical Name:Ledipasvir (acetone)
- CAS:1441674-54-9
- MF:C52H60F2N8O7
- Structure:

- Chemical Name:SP-420
- CAS:911714-45-9
- MF:C16H21NO6S
- Structure:

- Chemical Name:Mps1-IN-2
- CAS:1228817-38-6
- MF:C26H36N6O3
- Structure:

- Chemical Name:QL47
- CAS:1469988-75-7
- MF:C27H21N5O2
- Structure:

- Chemical Name:PF-01247324
- CAS:875051-72-2
- MF:C13H10Cl3N3O
- Structure:

- Chemical Name:AP-III-a4
- CAS:1177827-73-4
- MF:C31H43FN8O3
- Structure:

- Chemical Name:PSI-7976
- CAS:1190308-01-0
- MF:C22H29FN3O9P
- Structure:

- Chemical Name:GSK2141795
- CAS:1047634-65-0
- MF:C18H16Cl2F2N4O2
- Structure:

- Chemical Name:NVP-TNKS656
- CAS:1419949-20-4
- MF:C27H34N4O5
- Structure:

- Chemical Name:N1-(2,2,6,6-tetraMethylpiperidin-4-yl)-N2-p-tolyloxalaMide
- CAS:144217-65-2
- MF:C18H27N3O2
- Structure:

- Chemical Name:Optovin
- CAS:348575-88-2
- MF:C15H13N3OS2
- Structure:

- Chemical Name:Resmetirom
- CAS:920509-32-6
- MF:C17H12Cl2N6O4
- Structure:

- Chemical Name:Dafadine-A
- CAS:1065506-69-5
- MF:C23H25N3O3
- Structure:

- Chemical Name:GK921
- CAS:1025015-40-0
- MF:C21H20N4O
- Structure:

- Chemical Name:LDN-27219
- CAS:312946-37-5
- MF:C20H16N4O2S2
- Structure:

- Chemical Name:Skp2 Inhibitor C1
- CAS:432001-69-9
- MF:C18H13BrN2O4S2
- Structure:

- Chemical Name:Decernotinib
- CAS:944842-54-0
- MF:C18H19F3N6O
- Structure:

- Chemical Name:JIB-04 (NSC 693627) -Z
- CAS:199596-24-2
- MF:C17H13ClN4
- Structure:

- Chemical Name:Eluxadoline Dihydrochloride
- CAS:864825-13-8
- MF:C32H39Cl2N5O5
- Structure:

- Chemical Name:ERDAFITINIB
- CAS:1346242-81-6
- MF:C25H30N6O2
- Structure:

- Chemical Name:N,N'-(2,2'-(1,4-phenylene)bis(ethane-2,1-diyl))dipropane-2-sulfonaMide
- CAS:380607-77-2
- MF:C16H28N2O4S2
- Structure:

- Chemical Name:(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride
- CAS:135383-60-7
- MF:C11H13ClN2S
- Structure:

- Chemical Name:CPI 360
- CAS:1802175-06-9
- MF:C25H31N3O4
- Structure:

- Chemical Name:IKK epsilon-IN-1
- CAS:1292310-49-6
- MF:C26H27N5O3
- Structure:

- Chemical Name:GV-58
- CAS:1402821-41-3
- MF:C18H26N6OS
- Structure:

- Chemical Name:Z-360
- CAS:209219-38-5
- MF:C29H36N4O5
- Structure:

- Chemical Name:CX-4945 (sodiuM salt)
- CAS:1309357-15-0
- MF:C19H13ClN3NaO2
- Structure:

- Chemical Name:Exherin (trifluoroacetate)
- CAS:1135237-88-5
- MF:C24H35F3N8O8S2
- Structure:

- Chemical Name:Pyridoclax
- CAS:1651890-44-6
- MF:C29H22N4
- Structure:

- Chemical Name:GSK2879552
- CAS:1401966-69-5
- MF:C23H28N2O2
- Structure:

- Chemical Name:CAS:932749-62-7
- CAS:932749-62-7
- MF:C20H16Br2O3
- Structure:

- Chemical Name:(S)-1-((5-chloropyridin-3-yl)methyl)-8-((R)-3-methylmorpholino)-2-(trifluoromethyl)-3,4-dihydro-1H-pyrimido[1,2-a]pyrimidin-6(2H)-one
- CAS:1523406-39-4
- MF:C19H21ClF3N5O2
- Structure:

- Chemical Name:ML-228
- CAS:1357171-62-0
- MF:C27H21N5
- Structure:

- Chemical Name:4-((3,5-Dichloro-2-hydroxybenzyl)amino)-2-hydroxybenzoic acid
- CAS:1181226-02-7
- MF:C14H11Cl2NO4
- Structure:

- Chemical Name:Wnt Agonist
- CAS:853220-52-7
- MF:C19H18N4O3
- Structure:

- Chemical Name:N-(2-Aminophenyl)pyrazine-2-carboxamide
- CAS:926259-99-6
- MF:C11H10N4O
- Structure:

- Chemical Name:Theophylline-7-acetic acid
- CAS:652-37-9
- MF:C9H10N4O4
- Structure:

- Chemical Name:PFK-158
- CAS:1462249-75-7
- MF:C18H11F3N2O
- Structure:

- Chemical Name:CYM 50260
- CAS:1355026-60-6
- MF:C14H11Cl3FNO2
- Structure:

- Chemical Name:N-(4-ethylphenyl)-3-(hydroxymethyl)-N-isobutyl-4-((tetrahydro-2H-pyran-4-yl)methoxy)benzenesulfonamide
- CAS:1474110-21-8
- MF:C25H35NO5S
- Structure:

- Chemical Name:Epacadostat (INCB024360)
- CAS:1204669-58-8
- MF:C11H13BrFN7O4S
- Structure:

- Chemical Name:5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine
- CAS:1527503-11-2
- MF:C19H27N3O2
- Structure:

- Chemical Name:ML346
- CAS:100872-83-1
- MF:C14H12N2O4
- Structure:

- Chemical Name:IN00076730
- CAS:1454700-89-0
- MF:C17H21BrO2
- Structure:

- Chemical Name:JH-II-127
- CAS:1700693-08-8
- MF:C19H21ClN6O3
- Structure:

- Chemical Name:A-196
- CAS:1982372-88-2
- MF:C18H16Cl2N4
- Structure:

- Chemical Name:ODM-201
- CAS:1297538-32-9
- MF:C19H19ClN6O2
- Structure:

- Chemical Name:GSK-2881078
- CAS:1539314-06-1
- MF:C14H13F3N2O2S
- Structure:

- Chemical Name:Acamprosate calcium
- CAS:77337-73-6
- MF:C10H20CaN2O8S2
- Structure:

- Chemical Name:JNJ 63533054
- CAS:1802326-66-4
- MF:C17H17ClN2O2
- Structure:

- Chemical Name:mk-1064
- CAS:1207253-08-4
- MF:C24H20ClN5O3
- Chemical Name:EPZ031686
- CAS:1808011-22-4
- MF:C26H34ClF3N4O4S
- Structure:

- Chemical Name:RSL3
- CAS:1219810-16-8
- MF:C23H21ClN2O5
- Structure:

- Chemical Name:MS049
- CAS:1502816-23-0
- MF:C15H24N2O
- Structure:

- Chemical Name:PIK-III
- CAS:1383716-40-2
- MF:C17H17N7
- Structure:

- Chemical Name:ALS-8176
- CAS:1445385-02-3
- MF:C18H25ClFN3O6
- Chemical Name:SBI-0640756
- CAS:1821280-29-8
- MF:C23H14ClFN2O2
- Structure:

- Chemical Name:SirReal2
- CAS:709002-46-0
- MF:C22H20N4OS2
- Structure:

- Chemical Name:9-Propenyladenine
- CAS:1446486-33-4
- MF:C8H9N5
- Structure:

- Chemical Name:SRT3025
- CAS:1231952-55-8
- MF:C31H31N5O2S2
- Structure:

- Chemical Name:BI-9564
- CAS:1883429-22-8
- MF:C20H23N3O3
- Structure:

- Chemical Name:CFMTI
- CAS:864864-17-5
- MF:C19H16FN5O
- Structure:

- Chemical Name:N-(4-((1R,3S,5S)-3-amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide
- CAS:1210608-43-7
- MF:C24H23F3N4O
- Structure:

- Chemical Name:APS-2-79
- CAS:2002381-31-7
- MF:C23H22ClN3O3
- Structure:

- Chemical Name:ml390
- CAS:2029049-79-2
- MF:C21H21F3N2O3
- Structure:

- Chemical Name:Amiselimod(MT-1303) free base
- CAS:942399-20-4
- MF:C19H30F3NO3
- Structure:

- Chemical Name:NMS-P118
- CAS:1262417-51-5
- MF:C20H24F3N3O2
- Structure:

- Chemical Name:HDAC-IN-4
- CAS:934828-12-3
- MF:C24H29N5O
- Structure:

- Chemical Name:MX-69
- CAS:1005264-47-0
- MF:C27H26N2O4S
- Structure:

- Chemical Name:ASK1-IN-1
- CAS:1262041-49-5
- MF:C23H21N7O
- Structure:

- Chemical Name:BAY41-4109 Racemic
- CAS:298708-79-9
- MF:C18H13ClF3N3O2
- Structure:

- Chemical Name:MELK-8a
- CAS:1922153-17-0
- MF:C25H32N6O
- Structure:

- Chemical Name:1-(3,6-DIBROMO-9H-CARBAZOL-9-YL)-3-(DIMETHYLAMINO)PROPAN-2-OL
- CAS:253449-04-6
- MF:C17H18Br2N2O
- Structure:

- Chemical Name:RO 31-8220 METHANESULFONATE
- CAS:125314-64-9
- MF:C25H23N5O2S
- Structure:

- Chemical Name:Deoxythymidine triphosphate
- CAS:18423-43-3
- MF:C10H18N2NaO14P3
- Structure:

- Chemical Name:Testolactone
- CAS:968-93-4
- MF:C19H24O3
- Structure:

- Chemical Name:O-304
- CAS:1261289-04-6
- MF:C16H11Cl2N3O2S
- Structure:

- Chemical Name:Flunisolide
- CAS:3385-03-3
- MF:C24H31FO6