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Agonist Inhibitors

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  • Structure:1380424-42-9
  • Chemical Name:KML-29
  • CAS:1380424-42-9
  • MF:C24H21F6NO7


  • Structure:737789-87-6
  • Chemical Name:Relugolix
  • CAS:737789-87-6
  • MF:C29H27F2N7O5S

  • Structure:926927-61-9
  • Chemical Name:VTX-2337
  • CAS:926927-61-9
  • MF:C28H34N4O2

  • Structure:1402601-82-4
  • Chemical Name:TUG-770
  • CAS:1402601-82-4
  • MF:C19H14FNO2






  • Structure:1346133-08-1
  • Chemical Name:LY-2795050
  • CAS:1346133-08-1
  • MF:C23H22ClN3O2



  • Structure:1022958-60-6
  • Chemical Name:CEP-28122
  • CAS:1022958-60-6
  • MF:C28H35ClN6O3

  • Structure:173529-10-7
  • Chemical Name:HMN 176
  • CAS:173529-10-7
  • MF:C20H18N2O4S

  • Structure:849675-66-7
  • Chemical Name:HM 30181A
  • CAS:849675-66-7
  • MF:C38H36N6O7



  • Structure:1331782-27-4
  • Chemical Name:PF 04995274
  • CAS:1331782-27-4
  • MF:C23H32N2O6

  • Structure:1351522-04-7
  • Chemical Name:AC710
  • CAS:1351522-04-7
  • MF:C31H42N6O4



  • Structure:911714-45-9
  • Chemical Name:SP-420
  • CAS:911714-45-9
  • MF:C16H21NO6S

  • Structure:1228817-38-6
  • Chemical Name:Mps1-IN-2
  • CAS:1228817-38-6
  • MF:C26H36N6O3

  • Structure:1469988-75-7
  • Chemical Name:QL47
  • CAS:1469988-75-7
  • MF:C27H21N5O2

  • Structure:875051-72-2
  • Chemical Name:PF-01247324
  • CAS:875051-72-2
  • MF:C13H10Cl3N3O

  • Structure:1177827-73-4
  • Chemical Name:AP-III-a4
  • CAS:1177827-73-4
  • MF:C31H43FN8O3

  • Structure:1190308-01-0
  • Chemical Name:PSI-7976
  • CAS:1190308-01-0
  • MF:C22H29FN3O9P

  • Structure:1047634-65-0
  • Chemical Name:GSK2141795
  • CAS:1047634-65-0
  • MF:C18H16Cl2F2N4O2

  • Structure:1419949-20-4
  • Chemical Name:NVP-TNKS656
  • CAS:1419949-20-4
  • MF:C27H34N4O5


  • Structure:348575-88-2
  • Chemical Name:Optovin
  • CAS:348575-88-2
  • MF:C15H13N3OS2

  • Structure:920509-32-6
  • Chemical Name:Resmetirom
  • CAS:920509-32-6
  • MF:C17H12Cl2N6O4

  • Structure:1065506-69-5
  • Chemical Name:Dafadine-A
  • CAS:1065506-69-5
  • MF:C23H25N3O3

  • Structure:1025015-40-0
  • Chemical Name:GK921
  • CAS:1025015-40-0
  • MF:C21H20N4O

  • Structure:312946-37-5
  • Chemical Name:LDN-27219
  • CAS:312946-37-5
  • MF:C20H16N4O2S2


  • Structure:944842-54-0
  • Chemical Name:Decernotinib
  • CAS:944842-54-0
  • MF:C18H19F3N6O



  • Structure:1346242-81-6
  • Chemical Name:ERDAFITINIB
  • CAS:1346242-81-6
  • MF:C25H30N6O2



  • Structure:1802175-06-9
  • Chemical Name:CPI 360
  • CAS:1802175-06-9
  • MF:C25H31N3O4


  • Structure:1402821-41-3
  • Chemical Name:GV-58
  • CAS:1402821-41-3
  • MF:C18H26N6OS

  • Structure:209219-38-5
  • Chemical Name:Z-360
  • CAS:209219-38-5
  • MF:C29H36N4O5



  • Structure:1651890-44-6
  • Chemical Name:Pyridoclax
  • CAS:1651890-44-6
  • MF:C29H22N4

  • Structure:1401966-69-5
  • Chemical Name:GSK2879552
  • CAS:1401966-69-5
  • MF:C23H28N2O2



  • Structure:1357171-62-0
  • Chemical Name:ML-228
  • CAS:1357171-62-0
  • MF:C27H21N5


  • Structure:853220-52-7
  • Chemical Name:Wnt Agonist
  • CAS:853220-52-7
  • MF:C19H18N4O3



  • Structure:1462249-75-7
  • Chemical Name:PFK-158
  • CAS:1462249-75-7
  • MF:C18H11F3N2O

  • Structure:1355026-60-6
  • Chemical Name:CYM 50260
  • CAS:1355026-60-6
  • MF:C14H11Cl3FNO2




  • Structure:100872-83-1
  • Chemical Name:ML346
  • CAS:100872-83-1
  • MF:C14H12N2O4

  • Structure:1454700-89-0
  • Chemical Name:IN00076730
  • CAS:1454700-89-0
  • MF:C17H21BrO2

  • Structure:1700693-08-8
  • Chemical Name:JH-II-127
  • CAS:1700693-08-8
  • MF:C19H21ClN6O3

  • Structure:1982372-88-2
  • Chemical Name:A-196
  • CAS:1982372-88-2
  • MF:C18H16Cl2N4

  • Structure:1297538-32-9
  • Chemical Name:ODM-201
  • CAS:1297538-32-9
  • MF:C19H19ClN6O2

  • Structure:1539314-06-1
  • Chemical Name:GSK-2881078
  • CAS:1539314-06-1
  • MF:C14H13F3N2O2S


  • Structure:1802326-66-4
  • Chemical Name:JNJ 63533054
  • CAS:1802326-66-4
  • MF:C17H17ClN2O2

  • Structure:1207253-08-4
  • Chemical Name:mk-1064
  • CAS:1207253-08-4
  • MF:C24H20ClN5O3

  • Chemical Name:EPZ031686
  • CAS:1808011-22-4
  • MF:C26H34ClF3N4O4S

  • Structure:1219810-16-8
  • Chemical Name:RSL3
  • CAS:1219810-16-8
  • MF:C23H21ClN2O5

  • Structure:1502816-23-0
  • Chemical Name:MS049
  • CAS:1502816-23-0
  • MF:C15H24N2O

  • Structure:1383716-40-2
  • Chemical Name:PIK-III
  • CAS:1383716-40-2
  • MF:C17H17N7

  • Structure:1445385-02-3
  • Chemical Name:ALS-8176
  • CAS:1445385-02-3
  • MF:C18H25ClFN3O6

  • Chemical Name:SBI-0640756
  • CAS:1821280-29-8
  • MF:C23H14ClFN2O2

  • Structure:709002-46-0
  • Chemical Name:SirReal2
  • CAS:709002-46-0
  • MF:C22H20N4OS2


  • Structure:1231952-55-8
  • Chemical Name:SRT3025
  • CAS:1231952-55-8
  • MF:C31H31N5O2S2

  • Structure:1883429-22-8
  • Chemical Name:BI-9564
  • CAS:1883429-22-8
  • MF:C20H23N3O3

  • Structure:864864-17-5
  • Chemical Name:CFMTI
  • CAS:864864-17-5
  • MF:C19H16FN5O


  • Structure:2002381-31-7
  • Chemical Name:APS-2-79
  • CAS:2002381-31-7
  • MF:C23H22ClN3O3

  • Structure:2029049-79-2
  • Chemical Name:ml390
  • CAS:2029049-79-2
  • MF:C21H21F3N2O3


  • Structure:1262417-51-5
  • Chemical Name:NMS-P118
  • CAS:1262417-51-5
  • MF:C20H24F3N3O2

  • Structure:934828-12-3
  • Chemical Name:HDAC-IN-4
  • CAS:934828-12-3
  • MF:C24H29N5O

  • Structure:1005264-47-0
  • Chemical Name:MX-69
  • CAS:1005264-47-0
  • MF:C27H26N2O4S

  • Structure:1262041-49-5
  • Chemical Name:ASK1-IN-1
  • CAS:1262041-49-5
  • MF:C23H21N7O


  • Structure:1922153-17-0
  • Chemical Name:MELK-8a
  • CAS:1922153-17-0
  • MF:C25H32N6O




  • Structure:968-93-4
  • Chemical Name:Testolactone
  • CAS:968-93-4
  • MF:C19H24O3

  • Structure:1261289-04-6
  • Chemical Name:O-304
  • CAS:1261289-04-6
  • MF:C16H11Cl2N3O2S

  • Structure:3385-03-3
  • Chemical Name:Flunisolide
  • CAS:3385-03-3
  • MF:C24H31FO6