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Agonist Inhibitors

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  • Structure:939805-30-8
  • Chemical Name:ACTB-1003
  • CAS:939805-30-8
  • MF:C27H26F5N7O3

  • Structure:1345614-59-6
  • Chemical Name:AM-095
  • CAS:1345614-59-6
  • MF:C27H25N2NaO5

  • Structure:739366-20-2
  • Chemical Name:Anagliptin
  • CAS:739366-20-2
  • MF:C19H25N7O2

  • Structure:1226895-20-0
  • Chemical Name:ATB 346
  • CAS:1226895-20-0
  • MF:C21H19NO3S

  • Structure:853299-07-7
  • Chemical Name:AUZ 454
  • CAS:853299-07-7
  • MF:C24H26F3N7O2


  • Structure:442908-10-3
  • Chemical Name:Vipadenant
  • CAS:442908-10-3
  • MF:C16H15N7O

  • Structure:1379573-92-8
  • Chemical Name:CBB 1007
  • CAS:1379573-92-8
  • MF:C27H34N8O4

  • Structure:491833-29-5
  • Chemical Name:Eliglustat
  • CAS:491833-29-5
  • MF:C23H36N2O4

  • Structure:720690-73-3
  • Chemical Name:GSK 189254A
  • CAS:720690-73-3
  • MF:C21H25N3O2

  • Structure:376594-67-1
  • Chemical Name:LY 450108
  • CAS:376594-67-1
  • MF:C19H22F2N2O3S


  • Structure:464930-42-5
  • Chemical Name:SSR 240612
  • CAS:464930-42-5
  • MF:C42H53ClN4O7S

  • Structure:1166827-44-6
  • Chemical Name:AZD-7687
  • CAS:1166827-44-6
  • MF:C21H25N3O3



  • Structure:1146963-51-0
  • Chemical Name:J 147
  • CAS:1146963-51-0
  • MF:C18H17F3N2O2

  • Structure:871266-63-6
  • Chemical Name:PCI-27483
  • CAS:871266-63-6
  • MF:C26H24N6O9S

  • Structure:929901-49-5
  • Chemical Name:SGI-110
  • CAS:929901-49-5
  • MF:C18H24N9O10P



  • Structure:863513-91-1
  • Chemical Name:GRT6005
  • CAS:863513-91-1
  • MF:C24H27FN2O



  • Structure:304853-42-7
  • Chemical Name:NSP989
  • CAS:304853-42-7
  • MF:C16H15N3OS

  • Structure:1005780-62-0
  • Chemical Name:TAK-593
  • CAS:1005780-62-0
  • MF:C23H23N7O3

  • Structure:1320288-17-2
  • Chemical Name:UNC0646
  • CAS:1320288-17-2
  • MF:C36H59N7O2


  • Structure:733030-01-8
  • Chemical Name:TAS-102
  • CAS:733030-01-8
  • MF:C19H23Cl2F3N6O7


  • Structure:769856-81-7
  • Chemical Name:TPT-260
  • CAS:769856-81-7
  • MF:C8H12N4S3

  • Structure:344897-95-6
  • Chemical Name:Leukadherin 1
  • CAS:344897-95-6
  • MF:C22H15NO4S2


  • Structure:1619994-68-1
  • Chemical Name:GSK 2801
  • CAS:1619994-68-1
  • MF:C20H21NO4S

  • Structure:897732-93-3
  • Chemical Name:JNJ-38431055
  • CAS:897732-93-3
  • MF:C21H29N5O6S



  • Structure:1398044-45-5
  • Chemical Name:Piribedil-d8
  • CAS:1398044-45-5
  • MF:C16H18N4O2



  • Structure:1421438-81-4
  • Chemical Name:LY3039478
  • CAS:1421438-81-4
  • MF:C22H23F3N4O4

  • Structure:913611-97-9
  • Chemical Name:Brexpiprazole
  • CAS:913611-97-9
  • MF:C25H27N3O2S

  • Structure:866460-33-5
  • Chemical Name:Setipiprant
  • CAS:866460-33-5
  • MF:C24H19FN2O3

  • Structure:1216665-49-4
  • Chemical Name:APY29
  • CAS:1216665-49-4
  • MF:C17H16N8


  • Structure:220551-92-8
  • Chemical Name:DAA-1106
  • CAS:220551-92-8
  • MF:C23H22FNO4


  • Structure:878385-84-3
  • Chemical Name:AZD-5069
  • CAS:878385-84-3
  • MF:C18H22F2N4O5S2

  • Structure:1254036-77-5
  • Chemical Name:GSK-2269557
  • CAS:1254036-77-5
  • MF:C26H29ClN6O

  • Structure:932730-51-3
  • Chemical Name:CDDO-EA
  • CAS:932730-51-3
  • MF:C33H46N2O3


  • Structure:1099644-42-4
  • Chemical Name:ITD-1
  • CAS:1099644-42-4
  • MF:C27H29NO3


  • Structure:1604810-84-5
  • Chemical Name:CDK7-IN-1
  • CAS:1604810-84-5
  • MF:C31H28ClN7O2

  • Structure:1416133-89-5
  • Chemical Name:JW 642
  • CAS:1416133-89-5
  • MF:C21H20F6N2O3

  • Structure:1446182-94-0
  • Chemical Name:CUDC-427
  • CAS:1446182-94-0
  • MF:C29H36N6O4S

  • Structure:1431698-10-0
  • Chemical Name:OTSSP167HCL
  • CAS:1431698-10-0
  • MF:C25H29Cl3N4O2

  • Structure:1584713-87-0
  • Chemical Name:BMS-983970
  • CAS:1584713-87-0
  • MF:C26H26F4N4O3

  • Structure:1258392-53-8
  • Chemical Name:AZD-5582
  • CAS:1258392-53-8
  • MF:C58H78N8O8

  • Structure:704869-38-5
  • Chemical Name:SUN11602
  • CAS:704869-38-5
  • MF:C26H37N5O2


  • Structure:1527473-33-1
  • Chemical Name:PF-06447475
  • CAS:1527473-33-1
  • MF:C17H15N5O

  • Structure:1598383-40-4
  • Chemical Name:EPZ011969
  • CAS:1598383-40-4
  • MF:C35H51N5O4

  • Structure:210826-40-7
  • Chemical Name:MCC950
  • CAS:210826-40-7
  • MF:C20H24N2O5S


  • Structure:1223397-11-2
  • Chemical Name:WZB117
  • CAS:1223397-11-2
  • MF:C20H13FO6

  • Structure:321661-62-5
  • Chemical Name:Csn-B
  • CAS:321661-62-5
  • MF:C18H26O5



  • Structure:1421693-22-2
  • Chemical Name:CDKI-73
  • CAS:1421693-22-2
  • MF:C15H15FN6O2S2




  • Structure:676128-63-5
  • Chemical Name:RSV604
  • CAS:676128-63-5
  • MF:C22H17FN4O2

  • Structure:1626387-80-1
  • Chemical Name:AZD 3759
  • CAS:1626387-80-1
  • MF:C22H23ClFN5O3

  • Structure:1698878-14-6
  • Chemical Name:Nampt-IN-1
  • CAS:1698878-14-6
  • MF:C20H25N3O5S

  • Structure:1203494-49-8
  • Chemical Name:DASA-58
  • CAS:1203494-49-8
  • MF:C19H23N3O6S2

  • Structure:263890-70-6
  • Chemical Name:GR148672X
  • CAS:263890-70-6
  • MF:C15H11F3N2O2S

  • Structure:1393465-84-3
  • Chemical Name:PLX7904
  • CAS:1393465-84-3
  • MF:C24H22F2N6O3S

  • Structure:912656-34-9
  • Chemical Name:XEN907
  • CAS:912656-34-9
  • MF:C21H21NO4

  • Structure:1448232-80-1
  • Chemical Name:Naquotinib
  • CAS:1448232-80-1
  • MF:C30H42N8O3

  • Structure:1292300-75-4
  • Chemical Name:TASP0415914
  • CAS:1292300-75-4
  • MF:C13H17N5O3S

  • Structure:157009-81-9
  • Chemical Name:GPRP (acetate)
  • CAS:157009-81-9
  • MF:C20H35N7O7

  • Structure:140926-75-6
  • Chemical Name:NSC5844
  • CAS:140926-75-6
  • MF:C20H16Cl2N4

  • Structure:1310726-60-3
  • Chemical Name:Upadacitinib
  • CAS:1310726-60-3
  • MF:C17H19F3N6O

  • Structure:1046447-90-8
  • Chemical Name:jnj39758979
  • CAS:1046447-90-8
  • MF:C11H19N5



  • Structure:1784751-18-3
  • Chemical Name:TA-01
  • CAS:1784751-18-3
  • MF:C20H12F3N3

  • Structure:1883429-21-7
  • Chemical Name:BI-7273
  • CAS:1883429-21-7
  • MF:C20H23N3O3

  • Structure:1801747-42-1
  • Chemical Name:SHP099
  • CAS:1801747-42-1
  • MF:C16H19Cl2N5

  • Structure:1445605-23-1
  • Chemical Name:Lu AF21934
  • CAS:1445605-23-1
  • MF:C14H16Cl2N2O2

  • Structure:1707289-21-1
  • Chemical Name:BLU-554
  • CAS:1707289-21-1
  • MF:C24H24Cl2N4O4


  • Structure:1001288-58-9
  • Chemical Name:SHP-627
  • CAS:1001288-58-9
  • MF:C20H17NO5