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Agonist Inhibitors
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- Structure:

- Chemical Name:Regorafenib (Hydrochloride)
- CAS:835621-07-3
- MF:C21H16Cl2F4N4O3
- Structure:

- Chemical Name:VTP-27999 (Hydrochloride)
- CAS:1264191-73-2
- MF:C26H42Cl2N4O5
- Structure:

- Chemical Name:Phenol, 4-chloro-3-[5-Methyl-3-[[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]aMino]-1,2,4-benzotriazin-7-yl]-
- CAS:867334-05-2
- MF:C26H26ClN5O2
- Structure:

- Chemical Name:1alpha-Hydroxy VD4
- CAS:143032-85-3
- MF:C28H46O2
- Structure:

- Chemical Name:2,4-IMidazolidinedione, 5-[(7-chloro-1H-indol-3-yl)Methyl]-3-Methyl-, (5R)-
- CAS:852391-19-6
- MF:C13H12ClN3O2
- Structure:

- Chemical Name:ACTB-1003
- CAS:939805-30-8
- MF:C27H26F5N7O3
- Structure:

- Chemical Name:AM-095
- CAS:1345614-59-6
- MF:C27H25N2NaO5
- Structure:

- Chemical Name:Anagliptin
- CAS:739366-20-2
- MF:C19H25N7O2
- Structure:

- Chemical Name:ATB 346
- CAS:1226895-20-0
- MF:C21H19NO3S
- Structure:

- Chemical Name:AUZ 454
- CAS:853299-07-7
- MF:C24H26F3N7O2
- Structure:

- Chemical Name:BenzaMide, 3-[[4-[(5-hydroxy-2-Methylphenyl)aMino]-2-pyriMidinyl]aMino]-
- CAS:944795-06-6
- MF:C18H17N5O2
- Structure:

- Chemical Name:Vipadenant
- CAS:442908-10-3
- MF:C16H15N7O
- Structure:

- Chemical Name:CBB 1007
- CAS:1379573-92-8
- MF:C27H34N8O4
- Structure:

- Chemical Name:Eliglustat
- CAS:491833-29-5
- MF:C23H36N2O4
- Structure:

- Chemical Name:GSK 189254A
- CAS:720690-73-3
- MF:C21H25N3O2
- Structure:

- Chemical Name:LY 450108
- CAS:376594-67-1
- MF:C19H22F2N2O3S
- Structure:

- Chemical Name:MethanesulfonaMide, N-[5-[4-[5-[[(2R,6S)-2,6-diMethyl-4-Morpholinyl]Methyl]-2-oxazolyl]-1H-indazol-6-yl]-2-Methoxy-3-pyridinyl]-, rel-
- CAS:1254036-66-2
- MF:C24H28N6O5S
- Structure:

- Chemical Name:SSR 240612
- CAS:464930-42-5
- MF:C42H53ClN4O7S
- Structure:

- Chemical Name:AZD-7687
- CAS:1166827-44-6
- MF:C21H25N3O3
- Structure:

- Chemical Name:AG 7352 Hydrochloride
- CAS:175519-16-1
- MF:C18H20ClN5O4S
- Structure:

- Chemical Name:11-Piperazinyldibenzo[b,e][1,4]diazepine
- CAS:56296-18-5
- MF:C17H18N4
- Structure:

- Chemical Name:J 147
- CAS:1146963-51-0
- MF:C18H17F3N2O2
- Structure:

- Chemical Name:PCI-27483
- CAS:871266-63-6
- MF:C26H24N6O9S
- Structure:

- Chemical Name:SGI-110
- CAS:929901-49-5
- MF:C18H24N9O10P
- Structure:

- Chemical Name:(S)-3-(3-fluoro-4-(6-(2-Methyl-2H-tetrazol-5-yl)pyridin-3-yl)phenyl)-5-(hydroxyMethyl)oxazolidin-2-one
- CAS:1431699-67-0
- MF:C17H15FN6O3
- Structure:

- Chemical Name:BMN 673 (8R,9S)
- CAS:1207456-00-5
- MF:C19H14F2N6O
- Structure:

- Chemical Name:GRT6005
- CAS:863513-91-1
- MF:C24H27FN2O
- Structure:

- Chemical Name:NVP BGJ398 phosphate
- CAS:1310746-10-1
- MF:C26H34Cl2N7O7P
- Structure:

- Chemical Name:SDZ 220-581 (AMMoniuM salt)
- CAS:179411-94-0
- MF:C16H20ClN2O5P
- Structure:

- Chemical Name:NSP989
- CAS:304853-42-7
- MF:C16H15N3OS
- Structure:

- Chemical Name:TAK-593
- CAS:1005780-62-0
- MF:C23H23N7O3
- Structure:

- Chemical Name:UNC0646
- CAS:1320288-17-2
- MF:C36H59N7O2
- Structure:

- Chemical Name:Ripasudil hydrochloride dihydrate
- CAS:887375-67-9
- MF:C15H21ClFN3O3S
- Structure:

- Chemical Name:TAS-102
- CAS:733030-01-8
- MF:C19H23Cl2F3N6O7
- Structure:

- Chemical Name:2-Acetylfuro-1,4-naphthoquinone
- CAS:83280-65-3
- MF:C14H8O4
- Structure:

- Chemical Name:TPT-260
- CAS:769856-81-7
- MF:C8H12N4S3
- Structure:

- Chemical Name:Leukadherin 1
- CAS:344897-95-6
- MF:C22H15NO4S2
- Structure:

- Chemical Name:BenzaMide, N-[3-[3-[4-[(diMethylaMino)Methyl]phenyl]pyrazolo[1,5-a]pyriMidin-7-yl]phenyl]-3-(trifluoroMethyl)-
- CAS:950736-05-7
- MF:C29H24F3N5O
- Structure:

- Chemical Name:GSK 2801
- CAS:1619994-68-1
- MF:C20H21NO4S
- Structure:

- Chemical Name:JNJ-38431055
- CAS:897732-93-3
- MF:C21H29N5O6S
- Structure:

- Chemical Name:2-Methyl-3-furoic acid iMidazolide
- CAS:1415238-77-5
- MF:C9H8N2O2
- Structure:

- Chemical Name:RGB-286638 (free base)
- CAS:784210-88-4
- MF:C29H35N7O4
- Structure:

- Chemical Name:Piribedil-d8
- CAS:1398044-45-5
- MF:C16H18N4O2
- Structure:

- Chemical Name:MK-8033 (hydrochloride)
- CAS:1283000-43-0
- MF:C25H22ClN5O3S
- Structure:

- Chemical Name:Arginase inhibitor 1
- CAS:1345808-25-4
- MF:C13H27BN2O4
- Structure:

- Chemical Name:LY3039478
- CAS:1421438-81-4
- MF:C22H23F3N4O4
- Structure:

- Chemical Name:Brexpiprazole
- CAS:913611-97-9
- MF:C25H27N3O2S
- Structure:

- Chemical Name:Setipiprant
- CAS:866460-33-5
- MF:C24H19FN2O3
- Structure:

- Chemical Name:APY29
- CAS:1216665-49-4
- MF:C17H16N8
- Structure:

- Chemical Name:4-Methyl-2-(1-piperidinyl)-quinoline
- CAS:5465-86-1
- MF:C15H18N2
- Structure:

- Chemical Name:DAA-1106
- CAS:220551-92-8
- MF:C23H22FNO4
- Structure:

- Chemical Name:N,N'-(Dithiodi-2,1-ethanediyl)bis[2,5-dichloro-benzenesulfonaMide
- CAS:927822-86-4
- MF:C16H16Cl4N2O4S4
- Structure:

- Chemical Name:AZD-5069
- CAS:878385-84-3
- MF:C18H22F2N4O5S2
- Structure:

- Chemical Name:GSK-2269557
- CAS:1254036-77-5
- MF:C26H29ClN6O
- Structure:

- Chemical Name:CDDO-EA
- CAS:932730-51-3
- MF:C33H46N2O3
- Structure:

- Chemical Name:GDC-0834 (RaceMate)
- CAS:1133432-46-8
- MF:C33H36N6O3S
- Structure:

- Chemical Name:ITD-1
- CAS:1099644-42-4
- MF:C27H29NO3
- Structure:

- Chemical Name:Afobazole (hydrochloride)
- CAS:173352-39-1
- MF:C15H22ClN3O2S
- Structure:

- Chemical Name:CDK7-IN-1
- CAS:1604810-84-5
- MF:C31H28ClN7O2
- Structure:

- Chemical Name:JW 642
- CAS:1416133-89-5
- MF:C21H20F6N2O3
- Structure:

- Chemical Name:CUDC-427
- CAS:1446182-94-0
- MF:C29H36N6O4S
- Structure:

- Chemical Name:OTSSP167HCL
- CAS:1431698-10-0
- MF:C25H29Cl3N4O2
- Structure:

- Chemical Name:BMS-983970
- CAS:1584713-87-0
- MF:C26H26F4N4O3
- Structure:

- Chemical Name:AZD-5582
- CAS:1258392-53-8
- MF:C58H78N8O8
- Structure:

- Chemical Name:SUN11602
- CAS:704869-38-5
- MF:C26H37N5O2
- Structure:

- Chemical Name:Bucladesine (calciuM salt)
- CAS:938448-87-4
- MF:C18H26CaN5O8P
- Structure:

- Chemical Name:PF-06447475
- CAS:1527473-33-1
- MF:C17H15N5O
- Structure:

- Chemical Name:EPZ011969
- CAS:1598383-40-4
- MF:C35H51N5O4
- Structure:

- Chemical Name:MCC950
- CAS:210826-40-7
- MF:C20H24N2O5S
- Structure:

- Chemical Name:6-amino-4-(2,5-dimethoxyphenyl)-1,4-dihydro-3-(2-naphthalenyl)-pyrano[2,3-c]pyrazole-5-carbonitrile
- CAS:361185-42-4
- MF:C25H20N4O3
- Structure:

- Chemical Name:WZB117
- CAS:1223397-11-2
- MF:C20H13FO6
- Structure:

- Chemical Name:Csn-B
- CAS:321661-62-5
- MF:C18H26O5
- Structure:

- Chemical Name:2-[1-PIPERAZINYL]QUINOLINE MALEATE SALT
- CAS:5786-68-5
- MF:C17H19N3O4
- Structure:

- Chemical Name:Bis(4-cyanophenyl)methanol
- CAS:134521-16-7
- MF:C15H10N2O
- Structure:

- Chemical Name:CDKI-73
- CAS:1421693-22-2
- MF:C15H15FN6O2S2
- Structure:

- Chemical Name:3,6-Dichlorotrimellitic anhydride
- CAS:81742-10-1
- MF:C9H2Cl2O5
- Structure:

- Chemical Name:E6446 (dihydrochloride)
- CAS:1345675-25-3
- MF:C27H36ClN3O3
- Structure:

- Chemical Name:PDE1-IN-1 (phosphate)
- CAS:1642303-38-5
- MF:C29H29FN7O5P
- Structure:

- Chemical Name:RSV604
- CAS:676128-63-5
- MF:C22H17FN4O2
- Structure:

- Chemical Name:AZD 3759
- CAS:1626387-80-1
- MF:C22H23ClFN5O3
- Structure:

- Chemical Name:Nampt-IN-1
- CAS:1698878-14-6
- MF:C20H25N3O5S
- Structure:

- Chemical Name:DASA-58
- CAS:1203494-49-8
- MF:C19H23N3O6S2
- Structure:

- Chemical Name:GR148672X
- CAS:263890-70-6
- MF:C15H11F3N2O2S
- Structure:

- Chemical Name:PLX7904
- CAS:1393465-84-3
- MF:C24H22F2N6O3S
- Structure:

- Chemical Name:XEN907
- CAS:912656-34-9
- MF:C21H21NO4
- Structure:

- Chemical Name:Naquotinib
- CAS:1448232-80-1
- MF:C30H42N8O3
- Structure:

- Chemical Name:TASP0415914
- CAS:1292300-75-4
- MF:C13H17N5O3S
- Structure:

- Chemical Name:GPRP (acetate)
- CAS:157009-81-9
- MF:C20H35N7O7
- Structure:

- Chemical Name:NSC5844
- CAS:140926-75-6
- MF:C20H16Cl2N4
- Structure:

- Chemical Name:Upadacitinib
- CAS:1310726-60-3
- MF:C17H19F3N6O
- Structure:

- Chemical Name:jnj39758979
- CAS:1046447-90-8
- MF:C11H19N5
- Structure:

- Chemical Name:DG172 (dihydrochloride)
- CAS:1361504-77-9
- MF:C20H21BrClN3
- Structure:

- Chemical Name:HLCL-61 (hydrochloride)
- CAS:1158279-20-9
- MF:C23H25ClN2O
- Structure:

- Chemical Name:TA-01
- CAS:1784751-18-3
- MF:C20H12F3N3
- Structure:

- Chemical Name:BI-7273
- CAS:1883429-21-7
- MF:C20H23N3O3
- Structure:

- Chemical Name:SHP099
- CAS:1801747-42-1
- MF:C16H19Cl2N5
- Structure:

- Chemical Name:Lu AF21934
- CAS:1445605-23-1
- MF:C14H16Cl2N2O2
- Structure:

- Chemical Name:BLU-554
- CAS:1707289-21-1
- MF:C24H24Cl2N4O4
- Structure:

- Chemical Name:Elacestrant dihydrochloride
- CAS:1349723-93-8
- MF:C30H40Cl2N2O2
- Structure:

- Chemical Name:SHP-627
- CAS:1001288-58-9
- MF:C20H17NO5