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Agonist Inhibitors
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- Structure:

- Chemical Name:7-(Chlorodifluoromethyl)-5-(2-furanyl)-N-(2-thienylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
- CAS:442666-98-0
- MF:C17H11ClF2N4O2S
- Structure:

- Chemical Name:CAY10650
- CAS:1233706-88-1
- MF:C28H25NO6
- Structure:

- Chemical Name:Cl-Amidine
- CAS:913723-61-2
- MF:C14H19ClN4O2
- Structure:

- Chemical Name:Genz-123346
- CAS:491833-30-8
- MF:C24H38N2O4
- Structure:

- Chemical Name:6-[(3-aMinophenyl)Methyl]-4,6-dihydro-4-Methyl-2-(Methylsulfinyl)-5H-Thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one
- CAS:1221186-53-3
- MF:C17H16N4O2S2
- Structure:

- Chemical Name:N-Ethyl-7,10-dihydro-8-nitro-7-oxo-N-propyl-1,10-phenanthroline-3-carboxamide
- CAS:223666-07-7
- MF:C18H18N4O4
- Structure:

- Chemical Name:9-(6-Amino-3-pyridinyl)-1-[4-fluoro-3-(trifluoromethyl)phenyl]benzo[h]-1,6-naphthyridin-2(1H)-one
- CAS:1223002-54-7
- MF:C24H14F4N4O
- Structure:

- Chemical Name:GNE 477
- CAS:1032754-81-6
- MF:C21H28N8O3S2
- Structure:

- Chemical Name:JNJ-28312141
- CAS:885692-52-4
- MF:C26H32N6O2
- Structure:

- Chemical Name:CTS-1027
- CAS:193022-04-7
- MF:C19H20ClNO6S
- Structure:

- Chemical Name:CYT387 2H2SO4 salt
- CAS:1056636-06-6
- MF:C23H26N6O10S2
- Structure:

- Chemical Name:sodiuM 4-pentynoate
- CAS:101917-30-0
- MF:C5H5O2.Na
- Structure:

- Chemical Name:CHF 5074
- CAS:749269-83-8
- MF:C16H11Cl2FO2
- Structure:

- Chemical Name:Rigosertib sodium
- CAS:592542-60-4
- MF:C21H24NNaO8S
- Structure:

- Chemical Name:SB-681323
- CAS:444606-18-2
- MF:C23H19F3N4O3
- Structure:

- Chemical Name:INCB8761(PF-4136309)
- CAS:1341224-83-6
- MF:C29H31F3N6O3
- Structure:

- Chemical Name:LCQ-908
- CAS:956136-95-1
- MF:C25H24F3N3O2
- Structure:

- Chemical Name:MB-05032
- CAS:261365-11-1
- MF:C11H15N2O4PS
- Structure:

- Chemical Name:MK-6892
- CAS:917910-45-3
- MF:C19H22N4O5
- Structure:

- Chemical Name:NKP-1339
- CAS:197723-00-5
- MF:C14H12Cl4N4NaRu
- Structure:

- Chemical Name:RO 9187
- CAS:876708-03-1
- MF:C9H12N6O5
- Structure:

- Chemical Name:SB-649868
- CAS:380899-24-1
- MF:C26H24FN3O3S
- Structure:

- Chemical Name:TAK-960
- CAS:1137868-52-0
- MF:C27H34F3N7O3
- Structure:

- Chemical Name:ST101
- CAS:887603-94-3
- MF:C15H12N2O
- Structure:

- Chemical Name:ML 161
- CAS:423735-93-7
- MF:C17H17BrN2O2
- Structure:

- Chemical Name:N-(1-phenylethyl)-2-(pyrrolidin-1-yl)quinazolin-4-aMine
- CAS:662163-81-7
- MF:C20H22N4
- Structure:

- Chemical Name:CHIR-090
- CAS:728865-23-4
- MF:C24H27N3O5
- Structure:

- Chemical Name:NSC 42834
- CAS:195371-52-9
- MF:C23H24N2O
- Structure:

- Chemical Name:L778123
- CAS:253863-00-2
- MF:C22H21Cl2N5O
- Structure:

- Chemical Name:GDC-0032
- CAS:1282512-48-4
- MF:C24H28N8O2
- Structure:

- Chemical Name:360 A
- CAS:794458-56-3
- MF:C27H23N5O2+2
- Structure:

- Chemical Name:Exjade Fe3+ chelate
- CAS:554435-83-5
- MF:C21H12FeN3O4
- Structure:

- Chemical Name:ZP 1609 Hydrochloride
- CAS:943133-81-1
- MF:C14H18ClN3O4
- Structure:

- Chemical Name:IDO inhibitor 1
- CAS:1204669-37-3
- MF:C11H13BrFN7O4S
- Structure:

- Chemical Name:Kalydeco benzenesulfonate
- CAS:1134822-09-5
- MF:C30H34N2O6S
- Structure:

- Chemical Name:R-1530
- CAS:882531-87-5
- MF:C18H14ClFN4O
- Structure:

- Chemical Name:RGFP-966
- CAS:1357389-11-7
- MF:C21H19FN4O
- Structure:

- Chemical Name:ZD 6474 trifluoroacetate
- CAS:338992-53-3
- MF:C24H25BrF4N4O4
- Structure:

- Chemical Name:XMD17 109
- CAS:1435488-37-1
- MF:C36H46N8O3
- Structure:

- Chemical Name:FG 2216
- CAS:223387-75-5
- MF:C12H9ClN2O4
- Structure:

- Chemical Name:SKLB 610
- CAS:1125780-41-7
- MF:C21H16F3N3O3
- Structure:

- Chemical Name:APD668
- CAS:832714-46-2
- MF:C21H24FN5O5S
- Structure:

- Chemical Name:BRD-9539
- CAS:1374601-41-8
- MF:C24H21N3O3
- Structure:

- Chemical Name:2-ThiophenecarboxaMide, 4-cyano-5-[(3,5-dichloro-4-pyridinyl)thio]-N-[4-(Methylsulfonyl)phenyl]-
- CAS:1247825-37-1
- MF:C18H11Cl2N3O3S3
- Structure:

- Chemical Name:MonoMethylauristatin F
- CAS:745017-94-1
- MF:C39H65N5O8
- Structure:

- Chemical Name:TAS 103
- CAS:174634-09-4
- MF:C20H21Cl2N3O2
- Structure:

- Chemical Name:Necrosulfonamide
- CAS:1360614-48-7
- MF:C18H15N5O6S2
- Structure:

- Chemical Name:2-(2-Chlorophenyl)-4-(3-(diMethylaMino)phenyl)-5-Methyl-1H-pyrazolo[4,3-c]pyridine-3,6(2H,5H)-dione
- CAS:1218942-37-0
- MF:C21H19ClN4O2
- Structure:

- Chemical Name:AVE 0991 (sodiuM salt)
- CAS:306288-04-0
- MF:C29H33N4NaO5S2
- Structure:

- Chemical Name:Inauhzin
- CAS:309271-94-1
- MF:C25H19N5OS2
- Structure:

- Chemical Name:ABT-333
- CAS:1132935-63-7
- MF:C26H27N3O5S
- Structure:

- Chemical Name:Y320
- CAS:288250-47-5
- MF:C27H29ClN6O2
- Structure:

- Chemical Name:CEP-37440
- CAS:1391712-60-9
- MF:C30H38ClN7O3
- Structure:

- Chemical Name:3-[(3-Methoxybenzoyl)aMino]-4-(4-Methyl-1-piperazinyl)benzoic Acid Methyl Ester
- CAS:890190-22-4
- MF:C21H25N3O4
- Structure:

- Chemical Name:Dapagliflozin propanediol monohydrate
- CAS:960404-48-2
- MF:C24H33ClO8
- Structure:

- Chemical Name:Saroglitazar
- CAS:495399-09-2
- MF:C25H29NO4S
- Structure:

- Chemical Name:N-DesMethyl Netupitant
- CAS:290296-72-9
- MF:C29H30F6N4O
- Structure:

- Chemical Name:GSK2194069
- CAS:1332331-08-4
- MF:C25H24N4O3
- Structure:

- Chemical Name:ML355
- CAS:1532593-30-8
- MF:C21H19N3O4S2
- Structure:

- Chemical Name:SAR245409
- CAS:934493-76-2
- MF:C13H14N6O
- Structure:

- Chemical Name:6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)-
- CAS:202592-23-2
- MF:C19H17ClN4O2S
- Structure:

- Chemical Name:Elbasvir
- CAS:1370468-36-2
- MF:C49H55N9O7
- Structure:

- Chemical Name:GDC-0994
- CAS:1453848-26-4
- MF:C21H18ClFN6O2
- Structure:

- Chemical Name:Umbralisib
- CAS:1532533-67-7
- MF:C31H24F3N5O3
- Structure:

- Chemical Name:CVT-10216
- CAS:1005334-57-5
- MF:C24H19NO7S
- Structure:

- Chemical Name:URMC-099
- CAS:1229582-33-5
- MF:C27H27N5
- Structure:

- Chemical Name:LSN2814617
- CAS:1313498-08-6
- MF:C18H20FN5O
- Structure:

- Chemical Name:K-Ras G12C-IN-3
- CAS:1629268-19-4
- MF:C21H19Cl3N2O3
- Structure:

- Chemical Name:TRV-130
- CAS:1401031-39-7
- MF:C22H31ClN2O2S
- Structure:

- Chemical Name:DM1-SMCC
- CAS:1228105-51-8
- MF:C51H66ClN5O16S
- Structure:

- Chemical Name:BAL27862
- CAS:798577-91-0
- MF:C20H17N7O2
- Structure:

- Chemical Name:EX-527 (R-enantioMer)
- CAS:848193-69-1
- MF:C13H13ClN2O
- Structure:

- Chemical Name:TAK-063
- CAS:1238697-26-1
- MF:C23H17FN6O2
- Structure:

- Chemical Name:AI-10-49
- CAS:1256094-72-0
- MF:C30H22F6N6O5
- Structure:

- Chemical Name:ethyl 4-(((2R,3R,4S,5R,6S)-4,5-bis(benzo[d][1,3]dioxol-5-ylcarbamoyloxy)-2-(hydroxymethyl)-6-methoxy-tetrahydro-2H-pyran-3-yloxy)carbonyl)benzoate
- CAS:1137359-47-7
- MF:C33H33N3O15
- Structure:

- Chemical Name:TP0903
- CAS:1341200-45-0
- MF:C24H30ClN7O2S
- Structure:

- Chemical Name:3-([1,4′-Bipiperidin]-1′-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2-[3-(trifluoromethyl)phenyl]-4-quinolinecarboxamide
- CAS:1336960-13-4
- MF:C37H38BrF3N4O
- Structure:

- Chemical Name:H-ASP-PHE-OH
- CAS:13433-09-5
- MF:C13H16N2O5
- Structure:

- Chemical Name:Lumateperone
- CAS:313368-91-1
- MF:C24H28FN3O
- Structure:

- Chemical Name:2-butylsulfinyl-4-phenyl-6-thiophen-2-ylthieno[5,4-b]pyridin-3-amine
- CAS:459147-39-8
- MF:C21H20N2OS3
- Structure:

- Chemical Name:cyclopentyl 2-cyclohexyl-2-((6-(3-(hydroxyamino)-3-oxopropyl)pyridin-3-yl)methylamino)acetate
- CAS:1018673-42-1
- MF:C22H33N3O4
- Structure:

- Chemical Name:sbc-115076
- CAS:489415-96-5
- MF:C31H33N3O5
- Structure:

- Chemical Name:4-(2-(3-amino-1H-pyrazol-4-yl)-4-chlorophenoxy)-5-chloro-2-fluoro-N-(thiazol-4-yl)benzenesulfonamide Molecular Weight: 500.35
- CAS:1235403-62-9
- MF:C18H12Cl2FN5O3S2
- Structure:

- Chemical Name:Endoxifen HCl
- CAS:1032008-74-4
- MF:C25H28ClNO2
- Structure:

- Chemical Name:Centrinone
- CAS:1798871-30-3
- MF:C26H25F2N7O6S2
- Structure:

- Chemical Name:K-Ras-IN-1
- CAS:84783-01-7
- MF:C11H13NOS
- Structure:

- Chemical Name:Verinurad
- CAS:1352792-74-5
- MF:C20H16N2O2S
- Structure:

- Chemical Name:1-(4-(5-(5-amino-6-(5-(tert-butyl)-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one
- CAS:1620576-64-8
- MF:C22H31N9O3
- Structure:

- Chemical Name:CPI-268456
- CAS:1380087-86-4
- MF:C20H15Cl2N3O2
- Structure:

- Chemical Name:AZ-33
- CAS:1370290-34-8
- MF:C25H27N3O6S
- Structure:

- Chemical Name:AMG-337
- CAS:1173699-31-4
- MF:C23H22FN7O3
- Structure:

- Chemical Name:JAK3-IN-1
- CAS:1805787-93-2
- MF:C26H30ClN7O2
- Structure:

- Chemical Name:4-[4-(1-methyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]-benzonitrile
- CAS:1665195-94-7
- MF:C20H19N7
- Structure:

- Chemical Name:Revefenacin
- CAS:864750-70-9
- MF:C35H43N5O4
- Structure:

- Chemical Name:CP-456773 sodium
- CAS:256373-96-3
- MF:C20H23N2NaO5S
- Structure:

- Chemical Name:MS023
- CAS:1831110-54-3
- MF:C17H25N3O
- Structure:

- Chemical Name:XMU-MP-1
- CAS:2061980-01-4
- MF:C17H16N6O3S2
- Structure:

- Chemical Name:AKT inhibitor 2
- CAS:1313881-70-7
- MF:C27H24N6
- Structure:

- Chemical Name:MK-4101
- CAS:935273-79-3
- MF:C24H24F5N5O
- Structure:

- Chemical Name:GSK583
- CAS:1346547-00-9
- MF:C20H19FN4O2S