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Agonist Inhibitors

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  • Structure:1233706-88-1
  • Chemical Name:CAY10650
  • CAS:1233706-88-1
  • MF:C28H25NO6

  • Structure:913723-61-2
  • Chemical Name:Cl-Amidine
  • CAS:913723-61-2
  • MF:C14H19ClN4O2

  • Structure:491833-30-8
  • Chemical Name:Genz-123346
  • CAS:491833-30-8
  • MF:C24H38N2O4




  • Structure:1032754-81-6
  • Chemical Name:GNE 477
  • CAS:1032754-81-6
  • MF:C21H28N8O3S2

  • Structure:885692-52-4
  • Chemical Name:JNJ-28312141
  • CAS:885692-52-4
  • MF:C26H32N6O2

  • Structure:193022-04-7
  • Chemical Name:CTS-1027
  • CAS:193022-04-7
  • MF:C19H20ClNO6S



  • Structure:749269-83-8
  • Chemical Name:CHF 5074
  • CAS:749269-83-8
  • MF:C16H11Cl2FO2


  • Structure:444606-18-2
  • Chemical Name:SB-681323
  • CAS:444606-18-2
  • MF:C23H19F3N4O3


  • Structure:956136-95-1
  • Chemical Name:LCQ-908
  • CAS:956136-95-1
  • MF:C25H24F3N3O2

  • Structure:261365-11-1
  • Chemical Name:MB-05032
  • CAS:261365-11-1
  • MF:C11H15N2O4PS

  • Structure:917910-45-3
  • Chemical Name:MK-6892
  • CAS:917910-45-3
  • MF:C19H22N4O5

  • Structure:197723-00-5
  • Chemical Name:NKP-1339
  • CAS:197723-00-5
  • MF:C14H12Cl4N4NaRu

  • Structure:876708-03-1
  • Chemical Name:RO 9187
  • CAS:876708-03-1
  • MF:C9H12N6O5

  • Structure:380899-24-1
  • Chemical Name:SB-649868
  • CAS:380899-24-1
  • MF:C26H24FN3O3S

  • Structure:1137868-52-0
  • Chemical Name:TAK-960
  • CAS:1137868-52-0
  • MF:C27H34F3N7O3

  • Structure:887603-94-3
  • Chemical Name:ST101
  • CAS:887603-94-3
  • MF:C15H12N2O

  • Structure:423735-93-7
  • Chemical Name:ML 161
  • CAS:423735-93-7
  • MF:C17H17BrN2O2


  • Structure:728865-23-4
  • Chemical Name:CHIR-090
  • CAS:728865-23-4
  • MF:C24H27N3O5

  • Structure:195371-52-9
  • Chemical Name:NSC 42834
  • CAS:195371-52-9
  • MF:C23H24N2O

  • Structure:253863-00-2
  • Chemical Name:L778123
  • CAS:253863-00-2
  • MF:C22H21Cl2N5O

  • Structure:1282512-48-4
  • Chemical Name:GDC-0032
  • CAS:1282512-48-4
  • MF:C24H28N8O2

  • Structure:794458-56-3
  • Chemical Name:360 A
  • CAS:794458-56-3
  • MF:C27H23N5O2+2



  • Structure:1204669-37-3
  • Chemical Name:IDO inhibitor 1
  • CAS:1204669-37-3
  • MF:C11H13BrFN7O4S


  • Structure:882531-87-5
  • Chemical Name:R-1530
  • CAS:882531-87-5
  • MF:C18H14ClFN4O

  • Structure:1357389-11-7
  • Chemical Name:RGFP-966
  • CAS:1357389-11-7
  • MF:C21H19FN4O


  • Structure:1435488-37-1
  • Chemical Name:XMD17 109
  • CAS:1435488-37-1
  • MF:C36H46N8O3

  • Structure:223387-75-5
  • Chemical Name:FG 2216
  • CAS:223387-75-5
  • MF:C12H9ClN2O4

  • Structure:1125780-41-7
  • Chemical Name:SKLB 610
  • CAS:1125780-41-7
  • MF:C21H16F3N3O3

  • Structure:832714-46-2
  • Chemical Name:APD668
  • CAS:832714-46-2
  • MF:C21H24FN5O5S

  • Structure:1374601-41-8
  • Chemical Name:BRD-9539
  • CAS:1374601-41-8
  • MF:C24H21N3O3



  • Structure:174634-09-4
  • Chemical Name:TAS 103
  • CAS:174634-09-4
  • MF:C20H21Cl2N3O2




  • Structure:309271-94-1
  • Chemical Name:Inauhzin
  • CAS:309271-94-1
  • MF:C25H19N5OS2

  • Structure:1132935-63-7
  • Chemical Name:ABT-333
  • CAS:1132935-63-7
  • MF:C26H27N3O5S

  • Structure:288250-47-5
  • Chemical Name:Y320
  • CAS:288250-47-5
  • MF:C27H29ClN6O2

  • Structure:1391712-60-9
  • Chemical Name:CEP-37440
  • CAS:1391712-60-9
  • MF:C30H38ClN7O3



  • Structure:495399-09-2
  • Chemical Name:Saroglitazar
  • CAS:495399-09-2
  • MF:C25H29NO4S


  • Structure:1332331-08-4
  • Chemical Name:GSK2194069
  • CAS:1332331-08-4
  • MF:C25H24N4O3

  • Structure:1532593-30-8
  • Chemical Name:ML355
  • CAS:1532593-30-8
  • MF:C21H19N3O4S2

  • Structure:934493-76-2
  • Chemical Name:SAR245409
  • CAS:934493-76-2
  • MF:C13H14N6O


  • Structure:1370468-36-2
  • Chemical Name:Elbasvir
  • CAS:1370468-36-2
  • MF:C49H55N9O7

  • Structure:1453848-26-4
  • Chemical Name:GDC-0994
  • CAS:1453848-26-4
  • MF:C21H18ClFN6O2

  • Structure:1532533-67-7
  • Chemical Name:Umbralisib
  • CAS:1532533-67-7
  • MF:C31H24F3N5O3

  • Structure:1005334-57-5
  • Chemical Name:CVT-10216
  • CAS:1005334-57-5
  • MF:C24H19NO7S

  • Structure:1229582-33-5
  • Chemical Name:URMC-099
  • CAS:1229582-33-5
  • MF:C27H27N5

  • Structure:1313498-08-6
  • Chemical Name:LSN2814617
  • CAS:1313498-08-6
  • MF:C18H20FN5O

  • Structure:1629268-19-4
  • Chemical Name:K-Ras G12C-IN-3
  • CAS:1629268-19-4
  • MF:C21H19Cl3N2O3

  • Structure:1401031-39-7
  • Chemical Name:TRV-130
  • CAS:1401031-39-7
  • MF:C22H31ClN2O2S

  • Structure:1228105-51-8
  • Chemical Name:DM1-SMCC
  • CAS:1228105-51-8
  • MF:C51H66ClN5O16S

  • Structure:798577-91-0
  • Chemical Name:BAL27862
  • CAS:798577-91-0
  • MF:C20H17N7O2


  • Structure:1238697-26-1
  • Chemical Name:TAK-063
  • CAS:1238697-26-1
  • MF:C23H17FN6O2

  • Structure:1256094-72-0
  • Chemical Name:AI-10-49
  • CAS:1256094-72-0
  • MF:C30H22F6N6O5


  • Structure:1341200-45-0
  • Chemical Name:TP0903
  • CAS:1341200-45-0
  • MF:C24H30ClN7O2S


  • Structure:13433-09-5
  • Chemical Name:H-ASP-PHE-OH
  • CAS:13433-09-5
  • MF:C13H16N2O5

  • Structure:313368-91-1
  • Chemical Name:Lumateperone
  • CAS:313368-91-1
  • MF:C24H28FN3O



  • Structure:489415-96-5
  • Chemical Name:sbc-115076
  • CAS:489415-96-5
  • MF:C31H33N3O5


  • Structure:1032008-74-4
  • Chemical Name:Endoxifen HCl
  • CAS:1032008-74-4
  • MF:C25H28ClNO2

  • Structure:1798871-30-3
  • Chemical Name:Centrinone
  • CAS:1798871-30-3
  • MF:C26H25F2N7O6S2

  • Structure:84783-01-7
  • Chemical Name:K-Ras-IN-1
  • CAS:84783-01-7
  • MF:C11H13NOS

  • Structure:1352792-74-5
  • Chemical Name:Verinurad
  • CAS:1352792-74-5
  • MF:C20H16N2O2S


  • Structure:1380087-86-4
  • Chemical Name:CPI-268456
  • CAS:1380087-86-4
  • MF:C20H15Cl2N3O2

  • Structure:1370290-34-8
  • Chemical Name:AZ-33
  • CAS:1370290-34-8
  • MF:C25H27N3O6S

  • Structure:1173699-31-4
  • Chemical Name:AMG-337
  • CAS:1173699-31-4
  • MF:C23H22FN7O3

  • Structure:1805787-93-2
  • Chemical Name:JAK3-IN-1
  • CAS:1805787-93-2
  • MF:C26H30ClN7O2


  • Structure:864750-70-9
  • Chemical Name:Revefenacin
  • CAS:864750-70-9
  • MF:C35H43N5O4


  • Structure:1831110-54-3
  • Chemical Name:MS023
  • CAS:1831110-54-3
  • MF:C17H25N3O

  • Structure:2061980-01-4
  • Chemical Name:XMU-MP-1
  • CAS:2061980-01-4
  • MF:C17H16N6O3S2


  • Structure:935273-79-3
  • Chemical Name:MK-4101
  • CAS:935273-79-3
  • MF:C24H24F5N5O

  • Structure:1346547-00-9
  • Chemical Name:GSK583
  • CAS:1346547-00-9
  • MF:C20H19FN4O2S