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Agonist Inhibitors

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  • Structure:1352066-68-2
  • Chemical Name:AMG 232
  • CAS:1352066-68-2
  • MF:C28H35Cl2NO5S

  • Structure:919351-41-0
  • Chemical Name:AZD1283
  • CAS:919351-41-0
  • MF:C23H26N4O5S

  • Structure:1252594-99-2
  • Chemical Name:ETP-46321
  • CAS:1252594-99-2
  • MF:C20H27N9O3S


  • Structure:1619903-54-6
  • Chemical Name:LY2857785
  • CAS:1619903-54-6
  • MF:C26H36N6O

  • Structure:1430213-30-1
  • Chemical Name:ML216
  • CAS:1430213-30-1
  • MF:C15H9F4N5OS

  • Structure:1604810-83-4
  • Chemical Name:THZ1
  • CAS:1604810-83-4
  • MF:C31H28ClN7O2

  • Structure:1258226-87-7
  • Chemical Name:ABT-267
  • CAS:1258226-87-7
  • MF:C50H67N7O8

  • Structure:1268454-23-4
  • Chemical Name:INK1117
  • CAS:1268454-23-4
  • MF:C19H17N5O3

  • Structure:548470-11-7
  • Chemical Name:ISRIB
  • CAS:548470-11-7
  • MF:C22H24Cl2N2O4


  • Structure:1629265-17-3
  • Chemical Name:K-Ras G12C-IN-1
  • CAS:1629265-17-3
  • MF:C22H23Cl2N3O3

  • Structure:119391-56-9
  • Chemical Name:MAChR-IN-1
  • CAS:119391-56-9
  • MF:C23H25IN2O2



  • Structure:1186426-66-3
  • Chemical Name:DBPR108
  • CAS:1186426-66-3
  • MF:C16H25FN4O2

  • Structure:1338545-07-5
  • Chemical Name:OTS964
  • CAS:1338545-07-5
  • MF:C23H24N2O2S


  • Structure:1609960-31-7
  • Chemical Name:TH588
  • CAS:1609960-31-7
  • MF:C13H12Cl2N4

  • Structure:1516895-53-6
  • Chemical Name:SEP-0372814
  • CAS:1516895-53-6
  • MF:C21H19N7

  • Structure:1417162-36-7
  • Chemical Name:RI-2
  • CAS:1417162-36-7
  • MF:C21H18Cl2N2O4



  • Structure:894002-50-7
  • Chemical Name:LDN-212320
  • CAS:894002-50-7
  • MF:C17H15N3S



  • Structure:1228013-15-7
  • Chemical Name:CC-115
  • CAS:1228013-15-7
  • MF:C16H16N8O


  • Structure:1353625-73-6
  • Chemical Name:Presatovir
  • CAS:1353625-73-6
  • MF:C24H30ClN7O3S

  • Structure:1672665-49-4
  • Chemical Name:PT-2385
  • CAS:1672665-49-4
  • MF:C17H12F3NO4S

  • Structure:448947-81-7
  • Chemical Name:GlyT2-IN-1
  • CAS:448947-81-7
  • MF:C13H8Cl2N4S2

  • Structure:1162656-22-5
  • Chemical Name:MCB-613
  • CAS:1162656-22-5
  • MF:C20H20N2O

  • Structure:1793053-37-8
  • Chemical Name:LLY-507
  • CAS:1793053-37-8
  • MF:C36H42N6O

  • Structure:1638250-96-0
  • Chemical Name:ETC-159
  • CAS:1638250-96-0
  • MF:C19H17N7O3

  • Structure:2070015-09-5
  • Chemical Name:NU6300
  • CAS:2070015-09-5
  • MF:C20H23N5O3S

  • Structure:415903-37-6
  • Chemical Name:Grapiprant
  • CAS:415903-37-6
  • MF:C26H29N5O3S

  • Structure:1627710-50-2
  • Chemical Name:1627710-50-2
  • CAS:1627710-50-2
  • MF:C22H21F2N3O


  • Structure:178946-89-9
  • Chemical Name:C-DIM12
  • CAS:178946-89-9
  • MF:C23H17ClN2

  • Structure:1616392-22-3
  • Chemical Name:GSK-3326595
  • CAS:1616392-22-3
  • MF:C24H32N6O3

  • Structure:1448428-04-3
  • Chemical Name:Selonsertib
  • CAS:1448428-04-3
  • MF:C24H24FN7O


  • Structure:1550008-55-3
  • Chemical Name:ML264
  • CAS:1550008-55-3
  • MF:C17H21ClN2O4S

  • Structure:1622849-58-4
  • Chemical Name:GSK481
  • CAS:1622849-58-4
  • MF:C21H19N3O4

  • Structure:1415823-73-2
  • Chemical Name:evobrutinib
  • CAS:1415823-73-2
  • MF:C25H27N5O2

  • Structure:1123837-84-2
  • Chemical Name:Sitravatinib
  • CAS:1123837-84-2
  • MF:C33H29F2N5O4S

  • Structure:932737-65-0
  • Chemical Name:FITM
  • CAS:932737-65-0
  • MF:C18H18FN5OS


  • Structure:1414943-88-6
  • Chemical Name:BAY-1143572.
  • CAS:1414943-88-6
  • MF:C18H18FN5O2S


  • Structure:1190932-38-7
  • Chemical Name:COH-29
  • CAS:1190932-38-7
  • MF:C22H16N2O5S

  • Structure:222716-34-9
  • Chemical Name:SZL P1-41
  • CAS:222716-34-9
  • MF:C24H24N2O3S

  • Structure:890128-81-1
  • Chemical Name:BFH772
  • CAS:890128-81-1
  • MF:C23H16F3N3O3

  • Structure:1420367-28-7
  • Chemical Name:Lp-PLA2 -IN-1
  • CAS:1420367-28-7
  • MF:C21H17F5N4O3

  • Structure:1796596-46-7
  • Chemical Name:NSC23005 Sodium
  • CAS:1796596-46-7
  • MF:C13H18NNaO4S

  • Structure:1448169-71-8
  • Chemical Name:Futibatinib
  • CAS:1448169-71-8
  • MF:C22H22N6O3

  • Structure:1093119-54-0
  • Chemical Name:MKC3946
  • CAS:1093119-54-0
  • MF:C21H20N2O3S


  • Structure:1629869-44-8
  • Chemical Name:Pimodivir
  • CAS:1629869-44-8
  • MF:C20H19F2N5O2

  • Structure:107097-80-3
  • Chemical Name:LOXIGLUMIDE
  • CAS:107097-80-3
  • MF:C21H30Cl2N2O5



  • Structure:293754-55-9
  • Chemical Name:T0901317
  • CAS:293754-55-9
  • MF:C17H12F9NO3S


  • Structure:808-26-4
  • Chemical Name:Sancycline
  • CAS:808-26-4
  • MF:C21H22N2O7


  • Structure:82-98-4
  • Chemical Name:PIPERIDOLATE
  • CAS:82-98-4
  • MF:C21H25NO2

  • Structure:313348-27-5
  • Chemical Name:REGADENOSON
  • CAS:313348-27-5
  • MF:C15H18N8O5

  • Structure:127373-66-4
  • Chemical Name:Sivelestat
  • CAS:127373-66-4
  • MF:C20H22N2O7S

  • Structure:1320-66-7
  • Chemical Name:Chlorobutanol
  • CAS:1320-66-7
  • MF:C4H7Cl3O

  • Chemical Name:SN 2
  • CAS:
  • MF:


  • Structure:146986-50-7
  • Chemical Name:Y-27632
  • CAS:146986-50-7
  • MF:C14H21N3O


  • Structure:115066-14-3
  • Chemical Name:CNQX
  • CAS:115066-14-3
  • MF:C9H4N4O4



  • Structure:439083-90-6
  • Chemical Name:BAY 60-7550
  • CAS:439083-90-6
  • MF:C27H32N4O4



  • Structure:165668-41-7
  • Chemical Name:Indisulam
  • CAS:165668-41-7
  • MF:C14H12ClN3O4S2

  • Structure:116122-36-2
  • Chemical Name:BREVISCAPIN
  • CAS:116122-36-2
  • MF:C21H18O11.C21H18O12



  • Structure:85175-67-3
  • Chemical Name:Zatebradine
  • CAS:85175-67-3
  • MF:C26H36N2O5

  • Structure:211867-47-9
  • Chemical Name:Flumorph
  • CAS:211867-47-9
  • MF:C21H22FNO4

  • Structure:5581-42-0
  • Chemical Name:Glyparamide
  • CAS:5581-42-0
  • MF:C15H16ClN3O3S

  • Structure:88058-88-2
  • Chemical Name:Naxagolide
  • CAS:88058-88-2
  • MF:C15H21NO2

  • Structure:85604-00-8
  • Chemical Name:Zaltidine
  • CAS:85604-00-8
  • MF:C8H10N6S






  • Structure:133085-33-3
  • Chemical Name:BIBS 39
  • CAS:133085-33-3
  • MF:C32H36N4O3



  • Structure:89590-98-7
  • Chemical Name:mogroside VI
  • CAS:89590-98-7
  • MF:C66H112O34