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Agonist Inhibitors
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- Structure:

- Chemical Name:Beclabuvir
- CAS:958002-33-0
- MF:C36H45N5O5S
- Structure:

- Chemical Name:Eluxadoline
- CAS:864821-90-9
- MF:C32H35N5O5
- Structure:

- Chemical Name:LB-100
- CAS:1026680-07-8
- MF:C13H20N2O4
- Structure:

- Chemical Name:RGW 611
- CAS:6497-78-5
- MF:C9H14N4O3
- Structure:

- Chemical Name:GLPG-0778
- CAS:1206163-45-2
- MF:C22H23N5O2
- Structure:

- Chemical Name:ESI 09
- CAS:263707-16-0
- MF:C16H15ClN4O2
- Structure:

- Chemical Name:TZ-9
- CAS:1002789-86-7
- MF:C17H14N6O4
- Structure:

- Chemical Name:3-Methyl-2-((1S,2S)-2-(quinolin-2-yl)cyclopropyl)-3H-iMidazo[4,5-f]quinoline
- CAS:1516896-09-5
- MF:C21H19N7
- Structure:

- Chemical Name:PRT-060318
- CAS:1194961-19-7
- MF:C18H24N6O
- Structure:

- Chemical Name:Pyr6
- CAS:245747-08-4
- MF:C17H9F7N4O
- Structure:

- Chemical Name:AG-120
- CAS:1448346-63-1
- MF:C28H22ClF3N6O3
- Structure:

- Chemical Name:AZ-5104
- CAS:1421373-98-9
- MF:C27H31N7O2
- Structure:

- Chemical Name:"6,7-diphenyl-2-sulfanylidene-1H-pteridin-4-one
- CAS:14892-97-8
- MF:C18H12N4OS
- Structure:

- Chemical Name:BI-847325
- CAS:1207293-36-4
- MF:C29H28N4O2
- Structure:

- Chemical Name:STK321130
- CAS:923562-23-6
- MF:C21H16ClF3N4
- Structure:

- Chemical Name:HEXADECYL[2-([P-METHOXYBENZYL]-2-PYRIMIDINYLAMINO)ETHYL]DIMETHYL-AMMONIUM BROMIDE
- CAS:553-08-2
- MF:C32H55BrN4O
- Structure:

- Chemical Name:Theophylline monohydrate
- CAS:5967-84-0
- MF:C7H10N4O3
- Structure:

- Chemical Name:YHO-13351
- CAS:1346753-00-1
- MF:C27H37N3O7S2
- Structure:

- Chemical Name:Philanthotoxin 74
- CAS:1227301-51-0
- MF:C24H43ClN4O3
- Structure:

- Chemical Name:ARV-825
- CAS:1818885-28-7
- MF:C46H47ClN8O9S
- Structure:

- Chemical Name:MK2-IN-1 (hydrochloride)
- CAS:1314118-94-9
- MF:C27H26Cl2N4O2
- Structure:

- Chemical Name:PFI-4
- CAS:900305-37-5
- MF:C21H24N4O3
- Structure:

- Chemical Name:PD-L1 inhibitor 1
- CAS:1675203-84-5
- MF:C25H29N3O3
- Structure:

- Chemical Name:EPZ020411
- CAS:1700663-41-7
- MF:C25H38N4O3
- Structure:

- Chemical Name:ROR gamma-t-IN-1
- CAS:1426802-50-7
- MF:C23H18Cl2F3NO4S
- Structure:

- Chemical Name:VR23
- CAS:1624602-30-7
- MF:C19H16ClN5O6S
- Structure:

- Chemical Name:FIIN-2
- CAS:1633044-56-0
- MF:C35H38N8O4
- Structure:

- Chemical Name:Naloxegol Oxalate
- CAS:1354744-91-4
- MF:C36H55NO15
- Structure:

- Chemical Name:Fevipiprant
- CAS:872365-14-5
- MF:C19H17F3N2O4S
- Structure:

- Chemical Name:A-1155463
- CAS:1235034-55-5
- MF:C35H32FN5O4S2
- Structure:

- Chemical Name:DCEBIO
- CAS:60563-36-2
- MF:C9H8Cl2N2O
- Structure:

- Chemical Name:ACT-678689
- CAS:1783256-96-1
- MF:C23H22ClFN6O4S2
- Structure:

- Chemical Name:BAY-1217389
- CAS:1554458-53-5
- MF:C27H24F5N5O3
- Structure:

- Chemical Name:GPR39-C3
- CAS:1621175-65-2
- MF:C18H19ClN6O2S
- Structure:

- Chemical Name:Lusutrombopag
- CAS:1110766-97-6
- MF:C29H32Cl2N2O5S
- Structure:

- Chemical Name:CCF-642
- CAS:346640-08-2
- MF:C15H10N2O4S3
- Structure:

- Chemical Name:FIIN-3
- CAS:1637735-84-2
- MF:C34H36Cl2N8O4
- Structure:

- Chemical Name:5-(((1R,1aS,6bR)-1-(6-(trifluoromethyl)-1H-benzo[d]imidazol-2-yl)-1a,6b-dihydro-1H-cyclopropa[b]benzofuran-5-yl)oxy)-3,4-dihydro-1,8-naphthyridin-2(1H)-one
- CAS:1446090-77-2
- MF:C25H17F3N4O3
- Structure:

- Chemical Name:N-((3R,4R)-4-fluoro-1-(6-((3-methoxy-1-methyl-1H-pyrazol-4-yl)amino)-9-methyl-9H-purin-2-yl)pyrrolidin-3-yl)acrylamide
- CAS:1776112-90-3
- MF:C18H22FN9O2
- Structure:

- Chemical Name:CHZ868
- CAS:1895895-38-1
- MF:C22H19F2N5O2
- Structure:

- Chemical Name:CCT245737
- CAS:1489389-18-5
- MF:C16H16F3N7O
- Structure:

- Chemical Name:AM2394
- CAS:1442684-77-6
- MF:C22H25N5O4
- Structure:

- Chemical Name:Batefenterol
- CAS:743461-65-6
- MF:C40H42ClN5O7
- Structure:

- Chemical Name:MK-0812 (Succinate)
- CAS:851916-42-2
- MF:C28H40F3N3O7
- Structure:

- Chemical Name:RK-33
- CAS:1070773-09-9
- MF:C23H20N6O3
- Structure:

- Chemical Name:Rbin-1
- CAS:328023-11-6
- MF:C13H12N4S
- Structure:

- Chemical Name:IPI-549
- CAS:1693758-51-8
- MF:C30H24N8O2
- Structure:

- Chemical Name:UK-371804
- CAS:256477-09-5
- MF:C14H16ClN5O4S
- Structure:

- Chemical Name:NIH-12848
- CAS:959551-10-1
- MF:C20H14F3N3S
- Structure:

- Chemical Name:NCB-0846
- CAS:1792999-26-8
- MF:C21H21N5O2
- Structure:

- Chemical Name:Belizatinib
- CAS:1357920-84-3
- MF:C33H44FN5O3
- Structure:

- Chemical Name:Propionyl-L-carnitine hydrochloride
- CAS:119793-66-7
- MF:C10H20ClNO4
- Structure:

- Chemical Name:2-Hydroxybenzimidazole
- CAS:615-16-7
- MF:C7H6N2O
- Structure:

- Chemical Name:(+/-)-4-(4-AMINOPHENYL)-1,2-DIHYDRO-1-METHYL-2-PROPYLCARBAMOYL-6,7-METHYLENEDIOXYPHTHALAZINE
- CAS:173952-44-8
- MF:C20H22N4O3
- Structure:

- Chemical Name:NI-(S)-BPB-GLY
- CAS:96293-19-5
- MF:C27H25N3NiO3
- Structure:

- Chemical Name:1,3-DICHLORO-5-[(1E)-2(4-TRIFLUOROMETHYLPHENYL)ETHENYL]-BENZENE
- CAS:688348-33-6
- MF:C15H9Cl2F3
- Structure:

- Chemical Name:DL-Carnitine
- CAS:406-76-8
- MF:C7H15NO3
- Structure:

- Chemical Name:ACETAZOLAMIDE-D3
- CAS:1189904-01-5
- MF:C4H6N4O3S2
- Structure:

- Chemical Name:ICILIN
- CAS:36945-98-9
- MF:C16H13N3O4
- Structure:

- Chemical Name:CLORGYLINE HYDROCHLORIDE
- CAS:17780-75-5
- MF:C13H16Cl3NO
- Structure:

- Chemical Name:KENPAULLONE
- CAS:142273-20-9
- MF:C16H11BrN2O
- Structure:

- Chemical Name:N-(2-METHYL-6-BENZOXAZOLYL)-N'-1,5-NAPHTHYRIDIN-4-YL UREA
- CAS:249889-64-3
- MF:C17H13N5O2
- Structure:

- Chemical Name:(E)-3-[[[3-[2-(7-CHLORO-2-QUINOLINYL)ETHENYL]PHENYL]-[[(3-DIMETHYLAMINO)-3-OXOPROPYL]THIO]METHYL]THIO]-PROPANOIC ACID, SODIUM SALT
- CAS:115104-28-4
- MF:C26H27ClN2O3S2
- Structure:

- Chemical Name:IRBESARTAN-D4
- CAS:1216883-23-6
- MF:C25H28N6O
- Structure:

- Chemical Name:PX-866
- CAS:502632-66-8
- MF:C29H35NO8
- Structure:

- Chemical Name:AKTI-1/2
- CAS:612847-09-3
- MF:C34H29N7O
- Structure:

- Chemical Name:Gadodiamide
- CAS:131410-48-5
- MF:C16H26GdN5O8
- Structure:

- Chemical Name:DNQX
- CAS:2379-57-9
- MF:C8H4N4O6
- Structure:

- Chemical Name:(Z)-CAPSAICIN
- CAS:25775-90-0
- MF:C18H27NO3
- Structure:

- Chemical Name:H-SER-LEU-ILE-GLY-ARG-LEU-NH2
- CAS:171436-38-7
- MF:C29H56N10O7
- Structure:

- Chemical Name:(+/-)-SKF-38393 HYDROCHLORIDE
- CAS:81633-77-4
- MF:C16H18ClNO2
- Structure:

- Chemical Name:L-701,324
- CAS:142326-59-8
- MF:C21H14ClNO3
- Structure:

- Chemical Name:4-(4-(2,3-DIHYDROBENZO[1,4]DIOXIN-6-YL)-5-PYRIDIN-2-YL-1H-IMIDAZOL-2-YL)BENZAMIDE
- CAS:301836-43-1
- MF:C23H18N4O3
- Chemical Name:N-PHTHALYL-1-TRYPTOPHAN
- CAS:
- MF:
- Structure:

- Chemical Name:N-(2-[P-BROMOCINNAMYLAMINO]ETHYL)-5-ISOQUINOLINESULFONAMIDE HYDROCHLORIDE
- CAS:127243-85-0
- MF:C20H20BrN3O2S
- Structure:

- Chemical Name:9-[(R)-2-(Phosphonomethoxy)propyl]adenine monohydrate
- CAS:206184-49-8
- MF:C9H16N5O5P
- Structure:

- Chemical Name:Naratriptan
- CAS:121679-13-8
- MF:C17H25N3O2S
- Structure:

- Chemical Name:Beclamide
- CAS:501-68-8
- MF:C10H12ClNO
- Structure:

- Chemical Name:treosulfan
- CAS:299-75-2
- MF:C6H14O8S2
- Structure:

- Chemical Name:AM555S,TAC-101
- CAS:125973-56-0
- MF:C20H27NO3Si2
- Structure:

- Chemical Name:PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO-
- CAS:152811-62-6
- MF:C22H31N3O2
- Structure:

- Chemical Name:RUBOXISTAURIN MESYLATE
- CAS:169939-94-0
- MF:C28H28N4O3
- Structure:

- Chemical Name:Pipobroman
- CAS:54-91-1
- MF:C10H16Br2N2O2
- Structure:

- Chemical Name:dido
- CAS:69839-83-4
- MF:C7H7NO4
- Structure:

- Chemical Name:DAF-FM DA
- CAS:254109-22-3
- MF:C25H18F2N2O7
- Structure:

- Chemical Name:Co102862
- CAS:181144-66-1
- MF:C14H12FN3O2
- Structure:

- Chemical Name:1-(2-Diphenylmethoxyethyl)-4-(3-phenylpropyl)piperazinedihydrochloride
- CAS:76778-22-8
- MF:C28H34N2O
- Structure:

- Chemical Name:Centhaquine citrate
- CAS:1480809-77-5
- MF:C28H33N3O7
- Structure:

- Chemical Name:3-CARBOXY-4-OCTYL-2-METHYLENEBUTYROLACTONE
- CAS:218137-86-1
- MF:C14H22O4
- Structure:

- Chemical Name:Deracoxib
- CAS:169590-41-4
- MF:C17H14F3N3O3S
- Structure:

- Chemical Name:(3S,5R,8R,9S,10S,13R,14S,17R)-17-(3-furyl)-10,13-dimethyl-2,3,4,5,6,7, 8,9,11,12,15,16-dodecahydro-1H-cyclopenta[a]phenanthrene-3,14,17-triol
- CAS:156722-18-8
- MF:C23H34O4
- Structure:

- Chemical Name:Eflornithine hydrochloride hydrate
- CAS:96020-91-6
- MF:C6H15ClF2N2O3
- Structure:

- Chemical Name:2-[[(2S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperi dyl]propanoyl]amino]acetic acid dihydrate
- CAS:170098-38-1
- MF:C25H36N2O6
- Structure:

- Chemical Name:TAS 103
- CAS:174634-08-3
- MF:C20H19N3O2
- Structure:

- Chemical Name:KS 176
- CAS:1253452-78-6
- MF:C22H19N3O5
- Chemical Name:Uridine 5′-(tetrahydrogen triphosphate), 4-thio-, tetralithium salt
- CAS:20188-72-1
- MF:C9H15N2O14P3S.4Li
- Structure:

- Chemical Name:2-HYDROXYOLEICACID
- CAS:56472-29-8
- MF:C18H34O3
- Structure:

- Chemical Name:Uridine-5'-diphosphate disodium salt
- CAS:27821-45-0
- MF:C9H15N2NaO12P2
- Structure:

- Chemical Name:4,4'-DIACETAMIDODIPHENYLMETHANE
- CAS:2719-05-3
- MF:C17H18N2O2
- Structure:

- Chemical Name:Anamorelin
- CAS:249921-19-5
- MF:C31H42N6O3