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Agonist Inhibitors

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  • Structure:1401708-83-5
  • Chemical Name:Dihexa
  • CAS:1401708-83-5
  • MF:C27H44N4O5

  • Structure:269730-03-2
  • Chemical Name:RPI-1
  • CAS:269730-03-2
  • MF:C17H15NO4


  • Structure:1449685-96-4
  • Chemical Name:DDR1-IN-1
  • CAS:1449685-96-4
  • MF:C30H31F3N4O3

  • Structure:957135-43-2
  • Chemical Name:SM-164
  • CAS:957135-43-2
  • MF:C62H84N14O6

  • Structure:736992-21-5
  • Chemical Name:Elamipretide
  • CAS:736992-21-5
  • MF:C32H49N9O5

  • Structure:425399-05-9
  • Chemical Name:CASIN
  • CAS:425399-05-9
  • MF:C20H22N2O

  • Structure:1207283-85-9
  • Chemical Name:Eravacycline
  • CAS:1207283-85-9
  • MF:C27H31FN4O8

  • Structure:159857-79-1
  • Chemical Name:Val-cit-PAB-OH
  • CAS:159857-79-1
  • MF:C18H29N5O4


  • Structure:353519-63-8
  • Chemical Name:HLM006474
  • CAS:353519-63-8
  • MF:C25H25N3O2

  • Structure:947914-18-3
  • Chemical Name:ML365
  • CAS:947914-18-3
  • MF:C22H20N2O3

  • Structure:6310-41-4
  • Chemical Name:NSC-41589
  • CAS:6310-41-4
  • MF:C9H11NOS


  • Structure:1234480-46-6
  • Chemical Name:ACK1-B19
  • CAS:1234480-46-6
  • MF:C24H27N7O2

  • Structure:1338806-73-7
  • Chemical Name:CFI-400945
  • CAS:1338806-73-7
  • MF:C33H34N4O3

  • Structure:1239875-86-5
  • Chemical Name:SGI 7079
  • CAS:1239875-86-5
  • MF:C26H26FN7

  • Structure:1439399-58-2
  • Chemical Name:CB-839
  • CAS:1439399-58-2
  • MF:C26H24F3N7O3S

  • Structure:870281-34-8
  • Chemical Name:GS-9820
  • CAS:870281-34-8
  • MF:C21H16FN7O

  • Structure:309739-67-1
  • Chemical Name:PP2 analog
  • CAS:309739-67-1
  • MF:C16H17ClN4

  • Structure:1588521-78-1
  • Chemical Name:BET-BAY-002
  • CAS:1588521-78-1
  • MF:C22H18ClN5O

  • Structure:949912-58-7
  • Chemical Name:ReModelin
  • CAS:949912-58-7
  • MF:C15H14N4S


  • Structure:1126084-37-4
  • Chemical Name:ASP-9521
  • CAS:1126084-37-4
  • MF:C19H26N2O3

  • Structure:429653-73-6
  • Chemical Name:Y16
  • CAS:429653-73-6
  • MF:C24H20N2O3

  • Structure:1025967-78-5
  • Chemical Name:lifitegrast
  • CAS:1025967-78-5
  • MF:C29H24Cl2N2O7S

  • Structure:1345847-93-9
  • Chemical Name:Altiratinib
  • CAS:1345847-93-9
  • MF:C26H21F3N4O4

  • Structure:1352226-88-0
  • Chemical Name:AZD6738
  • CAS:1352226-88-0
  • MF:C20H24N6O2S


  • Structure:1346527-98-7
  • Chemical Name:CID-49830258
  • CAS:1346527-98-7
  • MF:C23H20N6O

  • Structure:1351635-67-0
  • Chemical Name:ONO-4059
  • CAS:1351635-67-0
  • MF:C25H24N6O3



  • Structure:1234423-95-0
  • Chemical Name:Tenapanor
  • CAS:1234423-95-0
  • MF:C50H66Cl4N8O10S2


  • Structure:1254205-52-1
  • Chemical Name:RQ-00203078
  • CAS:1254205-52-1
  • MF:C21H13ClF6N2O5S

  • Structure:1354825-58-3
  • Chemical Name:WEHI-345
  • CAS:1354825-58-3
  • MF:C22H23N7O

  • Structure:1361951-15-6
  • Chemical Name:TP-3654
  • CAS:1361951-15-6
  • MF:C22H25F3N4O

  • Structure:1562338-42-4
  • Chemical Name:LMI070
  • CAS:1562338-42-4
  • MF:C22H27N5O2

  • Structure:1383716-33-3
  • Chemical Name:Vps34-IN-1
  • CAS:1383716-33-3
  • MF:C21H24ClN7O

  • Structure:1494675-86-3
  • Chemical Name:ZA7371
  • CAS:1494675-86-3
  • MF:C18H21N5O3

  • Structure:803647-40-7
  • Chemical Name:NSC59984
  • CAS:803647-40-7
  • MF:C12H15N3O4


  • Structure:882405-89-2
  • Chemical Name:BBT594
  • CAS:882405-89-2
  • MF:C28H30F3N7O3

  • Structure:1334493-07-0
  • Chemical Name:BP-1-102
  • CAS:1334493-07-0
  • MF:C29H27F5N2O6S

  • Structure:1257213-50-5
  • Chemical Name:BMS-986020
  • CAS:1257213-50-5
  • MF:C29H26N2O5

  • Structure:1235560-28-7
  • Chemical Name:ABT-639
  • CAS:1235560-28-7
  • MF:C20H20ClF2N3O3S


  • Structure:836620-48-5
  • Chemical Name:AS1842856
  • CAS:836620-48-5
  • MF:C18H22FN3O3


  • Structure:1382979-44-3
  • Chemical Name:GDC-0084
  • CAS:1382979-44-3
  • MF:C18H22N8O2

  • Structure:1645286-75-4
  • Chemical Name:AZ6102
  • CAS:1645286-75-4
  • MF:C25H28N6O


  • Structure:176161-24-3
  • Chemical Name:BENZIMIDAVIR
  • CAS:176161-24-3
  • MF:C15H19Cl2N3O4



  • Structure:719277-26-6
  • Chemical Name:TG003
  • CAS:719277-26-6
  • MF:C13H15NO2S


  • Structure:681159-27-3
  • Chemical Name:CBR-5884
  • CAS:681159-27-3
  • MF:C14H12N2O4S2

  • Structure:1629268-00-3
  • Chemical Name:ARS-853
  • CAS:1629268-00-3
  • MF:C22H29ClN4O3

  • Structure:331862-41-0
  • Chemical Name:IMR-1A
  • CAS:331862-41-0
  • MF:C13H11NO5S2

  • Structure:861875-60-7
  • Chemical Name:NVP-BAW2881
  • CAS:861875-60-7
  • MF:C22H15F3N4O2

  • Structure:1163719-56-9
  • Chemical Name:CCT196969
  • CAS:1163719-56-9
  • MF:C27H24FN7O3

  • Structure:1627696-51-8
  • Chemical Name:LY-3177833
  • CAS:1627696-51-8
  • MF:C16H12FN5O

  • Structure:1609402-14-3
  • Chemical Name:HA-15
  • CAS:1609402-14-3
  • MF:C23H22N4O3S2

  • Structure:1435467-37-0
  • Chemical Name:PF-06282999
  • CAS:1435467-37-0
  • MF:C13H12ClN3O3S

  • Structure:1351758-37-6
  • Chemical Name:RR6
  • CAS:1351758-37-6
  • MF:C16H23NO4

  • Structure:1872382-47-2
  • Chemical Name:UNC3866
  • CAS:1872382-47-2
  • MF:C43H66N6O8

  • Structure:174262-13-6
  • Chemical Name:SDZ285-428
  • CAS:174262-13-6
  • MF:C24H20ClN3O

  • Structure:1345098-78-3
  • Chemical Name:XMD16-5
  • CAS:1345098-78-3
  • MF:C23H24N6O2


  • Structure:133550-35-3
  • Chemical Name:TYRPHOSTIN B48
  • CAS:133550-35-3
  • MF:C16H12N2O3






  • Structure:538-09-0
  • Chemical Name:Nortropine
  • CAS:538-09-0
  • MF:C7H13NO


  • Structure:1400989-25-4
  • Chemical Name:SC-43
  • CAS:1400989-25-4
  • MF:C21H13ClF3N3O2

  • Structure:597578-70-6
  • Chemical Name:PEN (human)
  • CAS:597578-70-6
  • MF:C97H159N27O32



  • Structure:173903-47-4
  • Chemical Name:TIZOXANIDE
  • CAS:173903-47-4
  • MF:C10H7N3O4S


  • Structure:
  • Chemical Name:TDZD-8
  • CAS:
  • MF:C10H10N2O2S










  • Structure:113558-14-8
  • Chemical Name:IKARISOSIDE F
  • CAS:113558-14-8
  • MF:C31H36O14


  • Chemical Name:VX-745
  • CAS:
  • MF: