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Agonist Inhibitors
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- Structure:

- Chemical Name:VidofludiMus
- CAS:717824-30-1
- MF:C20H18FNO4
- Structure:

- Chemical Name:UNC569
- CAS:1350547-65-7
- MF:C22H29FN6
- Structure:

- Chemical Name:XL-518 raceMate
- CAS:934662-91-6
- MF:C21H21F3IN3O2
- Structure:

- Chemical Name:TAK-441
- CAS:1186231-83-3
- MF:C28H31F3N4O6
- Structure:

- Chemical Name:UNC-926 Hydochloride
- CAS:1184136-10-4
- MF:C16H21BrN2O
- Structure:

- Chemical Name:GDC-0623
- CAS:1168091-68-6
- MF:C16H14FIN4O3
- Structure:

- Chemical Name:BVT-14225
- CAS:376638-65-2
- MF:C16H20ClN3O3S2
- Structure:

- Chemical Name:5-(9-isopropyl-2-Morpholino-9H-purin-6-yl)pyriMidin-2-aMine
- CAS:1246535-95-4
- MF:C16H20N8O
- Structure:

- Chemical Name:ONO 7643 FuMarate
- CAS:339539-92-3
- MF:C35H46N6O7
- Structure:

- Chemical Name:N2'-((1r,4r)-4-aMinocyclohexyl)-5'-chloro-N6-(3-fluorobenzyl)-[2,4'-bipyridine]-2',6-diaMine-rel-
- CAS:1263369-28-3
- MF:C23H25ClFN5
- Structure:

- Chemical Name:LDK-378 dihydrochloride
- CAS:1380575-43-8
- MF:C28H37Cl2N5O3S
- Structure:

- Chemical Name:LY 2801653 dihydrochloride
- CAS:1206801-37-7
- MF:C30H23ClF2N6O3
- Structure:

- Chemical Name:pilaralisib
- CAS:934526-89-3
- MF:C25H25ClN6O4S
- Structure:

- Chemical Name:DL-threo-2-Methylisocitrate
- CAS:71183-66-9
- MF:C7H10O7
- Structure:

- Chemical Name:SC 144
- CAS:895158-95-9
- MF:C16H11FN6O
- Structure:

- Chemical Name:PLX647
- CAS:873786-09-5
- MF:C21H17F3N4
- Structure:

- Chemical Name:BVT 2733
- CAS:376640-41-4
- MF:C17H21ClN4O3S2
- Structure:

- Chemical Name:kobe-2602
- CAS:454453-49-7
- MF:C14H9F4N5O4S
- Structure:

- Chemical Name:X-376
- CAS:1365267-27-1
- MF:C25H25Cl2FN6O3
- Structure:

- Chemical Name:Benzonitrile, 4-[[(1R,2R)-2-[(3R)-3-aMino-1-piperidinyl]-2,3-dihydro-1H-inden-1-yl]oxy]-3-chloro-
- CAS:1333210-07-3
- MF:C21H22ClN3O
- Structure:

- Chemical Name:TC-G 1001
- CAS:494191-73-0
- MF:C17H11FN2O3S
- Structure:

- Chemical Name:HJC-0350
- CAS:885434-70-8
- MF:C15H19NO2S
- Structure:

- Chemical Name:Walrycin B
- CAS:878419-78-4
- MF:C14H10F3N5O2
- Structure:

- Chemical Name:GSK J1
- CAS:1373422-53-7
- MF:C22H23N5O2
- Structure:

- Chemical Name:(S)-2-nitro-6-((6-(4-(trifluoroMethoxy)phenyl)pyridin-3-yl)Methoxy)-6,7-dihydro-5H-iMidazo[2,1-b][1,3]oxazine
- CAS:1257426-19-9
- MF:C19H15F3N4O5
- Structure:

- Chemical Name:K145 (hydrochloride)
- CAS:1449240-68-9
- MF:C18H25ClN2O3S
- Structure:

- Chemical Name:S1RA (hydrochloride)
- CAS:1265917-14-3
- MF:C20H24ClN3O2
- Structure:

- Chemical Name:AcotiaMide
- CAS:185106-16-5
- MF:C21H30N4O5S
- Structure:

- Chemical Name:ApiliMod (Mesylate)
- CAS:870087-36-8
- MF:C24H30N6O5S
- Structure:

- Chemical Name:N-(2-(2-(2-Methoxy-4-MorpholinophenylaMino)-5-fluoropyriMidin-4-ylaMino)phenyl)MethanesulfonaMide
- CAS:1191911-26-8
- MF:C22H25FN6O4S
- Structure:

- Chemical Name:GSK2141795 (hydrochloride)
- CAS:1047635-80-2
- MF:C18H17Cl3F2N4O2
- Structure:

- Chemical Name:MSX-122
- CAS:897657-95-3
- MF:C16H16N6
- Structure:

- Chemical Name:Mcl1-IN-1
- CAS:713492-66-1
- MF:C23H18ClN3O4
- Structure:

- Chemical Name:afoxolaner
- CAS:1093861-60-9
- MF:C26H17ClF9N3O3
- Structure:

- Chemical Name:2-(4-Isopropylpheny)-4H-chroMen-4-one
- CAS:92831-11-3
- MF:C18H16O2
- Structure:

- Chemical Name:LY-3009120
- CAS:1454682-72-4
- MF:C23H29FN6O
- Structure:

- Chemical Name:PF 04554878 hydrochloride
- CAS:1073160-26-5
- MF:C20H22ClF3N8O3S
- Structure:

- Chemical Name:Z-Ile-Glu-Pro-Phe-OMe
- CAS:252557-97-4
- MF:C34H44N4O9
- Structure:

- Chemical Name:Molidustat(BAY 85-3934)
- CAS:1154028-82-6
- MF:C13H14N8O2
- Structure:

- Chemical Name:1H-1,2,3-Triazole-1-acetic acid, 4-[[bis[[1-(1,1-diMethylethyl)-1H-1,2,3-triazol-4-yl]Methyl]aMino]Methyl]-
- CAS:1334179-85-9
- MF:C19H30N10O2
- Structure:

- Chemical Name:HUHS015
- CAS:1453097-13-6
- MF:C19H18N4O
- Structure:

- Chemical Name:NPS-1034
- CAS:1221713-92-3
- MF:C31H23F2N5O3
- Structure:

- Chemical Name:SAR-020106
- CAS:1184843-57-9
- MF:C19H19ClN6O
- Structure:

- Chemical Name:GS967
- CAS:1262618-39-2
- MF:C14H7F6N3O
- Structure:

- Chemical Name:Tipifarnib (S enantioMer)
- CAS:192185-71-0
- MF:C27H22Cl2N4O
- Structure:

- Chemical Name:Mitapivat
- CAS:1260075-17-9
- MF:C24H26N4O3S
- Structure:

- Chemical Name:N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-isopropyl-3-methyl-6-(6-(4-methylpiperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide
- CAS:1346572-63-1
- MF:C31H38N6O2
- Structure:

- Chemical Name:BIO-32546
- CAS:1548743-66-3
- MF:C28H31F6NO3
- Structure:

- Chemical Name:(E)-3-(3-bromo-4,5-dihydroxyphenyl)-N-(3,4,5-trihydroxybenzyl)prop-2-enethioamide
- CAS:1384426-12-3
- MF:C16H14BrNO5S
- Structure:

- Chemical Name:CB5083
- CAS:1542705-92-9
- MF:C24H23N5O2
- Structure:

- Chemical Name:2-(7-Fluoropyrrolo[1,2-a]quinoxalin-4-yl)hydrazide-2-pyrazinecarboxylic acid hydrochloride
- CAS:917497-70-2
- MF:C17H12ClFN6O3
- Structure:

- Chemical Name:BMS817378
- CAS:1174161-69-3
- MF:C24H18ClF2N4O7P
- Structure:

- Chemical Name:Bempedoic acid
- CAS:738606-46-7
- MF:C19H36O5
- Structure:

- Chemical Name:5-(4,6-dimorpholino-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine
- CAS:1225037-39-7
- MF:C17H20F3N7O2
- Structure:

- Chemical Name:Pyr10
- CAS:1315323-00-2
- MF:C18H13F6N3O2S
- Structure:

- Chemical Name:A-1210477
- CAS:1668553-26-1
- MF:C46H55N7O7S
- Structure:

- Chemical Name:AZD9496
- CAS:1639042-08-2
- MF:C25H25F3N2O2
- Structure:

- Chemical Name:IDO-IN-1
- CAS:914638-30-5
- MF:C9H7BrFN5O2
- Structure:

- Chemical Name:PSI-6206 13CD3
- CAS:1256490-42-2
- MF:C10H10D3FN2O5
- Structure:

- Chemical Name:NCT-501
- CAS:1802088-50-1
- MF:C21H32N6O3
- Structure:

- Chemical Name:Urolithin C
- CAS:165393-06-6
- MF:C13H8O5
- Structure:

- Chemical Name:AZD3264
- CAS:1609281-86-8
- MF:C21H23N5O4S
- Structure:

- Chemical Name:Voxelotor
- CAS:1446321-46-5
- MF:C19H19N3O3
- Structure:

- Chemical Name:AR-13324 (hydrochloride)
- CAS:1253952-02-1
- MF:C28H29Cl2N3O3
- Structure:

- Chemical Name:SGC707
- CAS:1687736-54-4
- MF:C16H18N4O2
- Structure:

- Chemical Name:ON123300
- CAS:1357470-29-1
- MF:C24H27N7O
- Structure:

- Chemical Name:Valbenazine
- CAS:1025504-45-3
- MF:C24H38N2O4
- Structure:

- Chemical Name:Danirixin
- CAS:954126-98-8
- MF:C19H21ClFN3O4S
- Structure:

- Chemical Name:PI3Kα inhibitor 1
- CAS:1235449-52-1
- MF:C23H25N9O3S
- Structure:

- Chemical Name:TY-52156
- CAS:934369-14-9
- MF:C18H19Cl2N3O
- Structure:

- Chemical Name:MK-0941
- CAS:1137916-97-2
- MF:C22H28N4O9S2
- Structure:

- Chemical Name:Ezutromid
- CAS:945531-77-1
- MF:C19H15NO3S
- Structure:

- Chemical Name:SHP099 (hydrochloride)
- CAS:1801747-11-4
- MF:C16H20Cl3N5
- Structure:

- Chemical Name:BAY-1125976.
- CAS:1402608-02-9
- MF:C23H21N5O
- Structure:

- Chemical Name:BAY-876
- CAS:1799753-84-6
- MF:C24H16F4N6O2
- Structure:

- Chemical Name:SKQ1 Bromide
- CAS:934826-68-3
- MF:C36H42BrO2P
- Structure:

- Chemical Name:CC-122
- CAS:1015474-32-4
- MF:C14H14N4O3
- Structure:

- Chemical Name:2-(4-fluoro-2-methylphenoxy)-N-(2-oxo-1l4,2l5-pyridin-4-yl)-4-(trifluoromethyl)benzamide
- CAS:1620846-16-3
- MF:C20H14F4N2O3
- Structure:

- Chemical Name:N-(4-((1R,3S,5S)-3-amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide
- CAS:1820565-69-2
- MF:C24H23F3N4O
- Structure:

- Chemical Name:GNE-495
- CAS:1449277-10-4
- MF:C22H20FN5O2
- Structure:

- Chemical Name:GSK6853
- CAS:1910124-24-1
- MF:C22H27N5O3
- Structure:

- Chemical Name:SH5-07
- CAS:1456632-41-9
- MF:C29H28F5N3O5S
- Structure:

- Chemical Name:BAY-1082439
- CAS:1375469-38-7
- MF:C25H30N6O5
- Structure:

- Chemical Name:TB5
- CAS:948841-07-4
- MF:C15H14BrNOS
- Structure:

- Chemical Name:GJ-103 sodium salt
- CAS:1459687-96-7
- MF:C16H15N4NaO3S
- Structure:

- Chemical Name:AMG-3969
- CAS:1361224-53-4
- MF:C21H20F6N4O3S
- Structure:

- Chemical Name:TD 139
- CAS:1450824-22-2
- MF:C28H30F2N6O8S
- Structure:

- Chemical Name:N-BUTYLDEOXYNOJIRIMYCIN, HYDROCHLORIDE
- CAS:210110-90-0
- MF:C10H22ClNO4
- Structure:

- Chemical Name:YU238259
- CAS:1943733-16-1
- MF:C22H22ClN3O4S
- Structure:

- Chemical Name:SM 324405
- CAS:677773-91-0
- MF:C19H23N5O4
- Structure:

- Chemical Name:BQR695
- CAS:1513879-21-4
- MF:C19H20N4O3
- Structure:

- Chemical Name:3,5-Dimethyl-1-adamantanol
- CAS:707-37-9
- MF:C12H20O
- Structure:

- Chemical Name:2-CARBOXYPHENYL PHOSPHATE
- CAS:6064-83-1
- MF:C7H7O6P
- Structure:

- Chemical Name:6-Ethyl-3-oxa-6-azaoctanol
- CAS:140-82-9
- MF:C8H19NO2
- Structure:

- Chemical Name:Flavopiridol
- CAS:146426-40-6
- MF:C21H20ClNO5
- Structure:

- Chemical Name:(4-BROMOPHENYL)[3-FLUORO-4-[[6-(METHYL-2-PROPENYLAMINO)HEXYL]OXY]PHENYL]-METHANONE
- CAS:161582-11-2
- MF:C23H27BrFNO2
- Structure:

- Chemical Name:MILNACIPRAN HYDROCHLORIDE
- CAS:92623-85-3
- MF:C15H22N2O
- Structure:

- Chemical Name:R-(-)-2-(4-ISOBUTYLPHENYL)PROPIONYL METHANSULPHONAMIDE, LYSINE SALT
- CAS:266359-93-7
- MF:C20H35N3O5S
- Structure:

- Chemical Name:Zoxazolamine
- CAS:61-80-3
- MF:C7H5ClN2O
- Structure:

- Chemical Name:COMPOUND 52
- CAS:212779-48-1
- MF:C16H19ClN6O