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Agonist Inhibitors
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- Structure:

- Chemical Name:7-Amino-3-methyl-3-cephem-4-carboxylic acid
- CAS:22252-43-3
- MF:C8H10N2O3S
- Structure:

- Chemical Name:RO 41-1049 HCL MAO-A INHIBITOR
- CAS:127500-84-9
- MF:C12H12FN3OS
- Structure:

- Chemical Name:VALROCEMIDE
- CAS:92262-58-3
- MF:C10H20N2O2
- Structure:

- Chemical Name:Dimesna
- CAS:16208-51-8
- MF:C4H8Na2O6S4
- Chemical Name:ODN 2007
- CAS:
- MF:
- Structure:

- Chemical Name:ENALAPRILAT-D5, SODIUM SALT
- CAS:1356922-29-6
- MF:C18H18D5N2NaO5
- Structure:

- Chemical Name:ERLOTINIB MESYLATE
- CAS:248594-19-6
- MF:C23H27N3O7S
- Structure:

- Chemical Name:Almotriptan
- CAS:154323-57-6
- MF:C17H25N3O2S
- Structure:

- Chemical Name:ATHIDATHION
- CAS:19691-80-6
- MF:C8H15N2O4PS3
- Structure:

- Chemical Name:SKF 96365 HYDROCHLORIDE
- CAS:130495-35-1
- MF:C22H27ClN2O3
- Structure:

- Chemical Name:Moguisteine
- CAS:119637-67-1
- MF:C16H21NO5S
- Structure:

- Chemical Name:5-Pyrimidinecarboxamide, N-hydroxy-2-[4-(2-naphthalenylsulfonyl)-1-piperazinyl]- (9CI)
- CAS:604769-01-9
- MF:C19H19N5O4S
- Structure:

- Chemical Name:4-(3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl)-phenylamine
- CAS:123066-64-8
- MF:C11H7F6N3
- Structure:

- Chemical Name:(R)-(+)-Etomoxir sodium salt
- CAS:828934-41-4
- MF:C15H20ClNaO4
- Structure:

- Chemical Name:IRAK-1/4 INHIBITOR I
- CAS:509093-47-4
- MF:C20H21N5O4
- Structure:

- Chemical Name:1,2,4-Oxadiazol-5(2H)-one, 3-[(1S,2S)-1-[2-[[(4S)-2-(4-fluoro-3,5-dimethylphenyl)-3-[3-(4-fluoro-1-methyl-1H-indazol-5-yl)-2,3-dihydro-2-oxo-1H-imidazol-1-yl]-2,4,6,7-tetrahydro-4-methyl-5H-pyrazolo[4,3-c]pyridin-5-yl]carbonyl]-5-[(4S)-tetrahydro-2,2-dimethyl-2H-pyran-4-yl]-1H-indol-1-yl]-2-methylcyclopropyl]-, calcium salt (2:1)
- CAS:2415797-61-2
- MF:C48H50CaF2N10O5
- Structure:

- Chemical Name:Ampalex
- CAS:154235-83-3
- MF:C14H15N3O
- Structure:

- Chemical Name:Indiplon
- CAS:325715-02-4
- MF:C20H16N4O2S
- Structure:

- Chemical Name:H-LYS-THR-GLU-GLU-ILE-SER-GLU-VAL-ASN-STA-VAL-ALA-GLU-PHE-OH
- CAS:350228-37-4
- MF:C73H118N16O27
- Structure:

- Chemical Name:Lexacalcitol
- CAS:131875-08-6
- MF:C29H48O4
- Structure:

- Chemical Name:3,4-Pyrrolidinediol, 2-(4-amino-5H-pyrrolo3,2-dpyrimidin-7-yl)-5-(hydroxymethyl)-, (2S,3S,4R,5R)-
- CAS:249503-25-1
- MF:C11H15N5O3
- Structure:

- Chemical Name:(R,R)-Formoterol
- CAS:67346-49-0
- MF:C19H24N2O4
- Structure:

- Chemical Name:Atipamezole
- CAS:104054-27-5
- MF:C14H16N2
- Structure:

- Chemical Name:NQ301
- CAS:130089-98-4
- MF:C18H12ClNO3
- Structure:

- Chemical Name:Bupropion
- CAS:34911-55-2
- MF:C13H18ClNO
- Structure:

- Chemical Name:6-THIO-2'-DEOXYGUANOSINE
- CAS:789-61-7
- MF:C10H13N5O3S
- Structure:

- Chemical Name:Linaprazan
- CAS:248919-64-4
- MF:C21H26N4O2
- Structure:

- Chemical Name:CHLORPHENOXAMINE
- CAS:77-38-3
- MF:C18H22ClNO
- Structure:

- Chemical Name:CYCLO(-ARG-GLY-ASP-D-TYR-LYS)
- CAS:217099-14-4
- MF:C27H41N9O8
- Structure:

- Chemical Name:2,3,4-TRIMETHOXYBENZYL ALCOHOL
- CAS:71989-96-3
- MF:C10H14O4
- Structure:

- Chemical Name:GW843682, 5-(5,6-Dimethoxy-1H-benzimidazol-1-yl)-3-{[2-(trifluoromethyl)-benzyl]oxy}thiophene-2-carboxamide
- CAS:660868-91-7
- MF:C22H18F3N3O4S
- Structure:

- Chemical Name:Atrasentan hydrochloride
- CAS:195733-43-8
- MF:C29H38N2O6.ClH
- Structure:

- Chemical Name:Talaporfin sodium
- CAS:220201-34-3
- MF:C38H42N5NaO9
- Structure:

- Chemical Name:4-Methylpyrazole
- CAS:7554-65-6
- MF:C4H6N2
- Structure:

- Chemical Name:Zacopride hydrochloride
- CAS:101303-98-4
- MF:C15H21Cl2N3O2
- Structure:

- Chemical Name:CP-547632
- CAS:252003-65-9
- MF:C20H24BrF2N5O3S
- Structure:

- Chemical Name:1-(4-Fluorophenyl)-N-[3-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-1,2-dihydro-2-oxo-3-pyridinecarboxamide
- CAS:888719-03-7
- MF:C25H16F2N4O3
- Structure:

- Chemical Name:3-[3-[2-(1-Piperidinyl)ethoxy]phenyl]-5-(1H-1,2,4-triazol-5-yl)-1H-indazole
- CAS:395104-30-0
- MF:C22H24N6O
- Structure:

- Chemical Name:N-[2,4-Difluoro-3-[[5-(3-pyridinyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]carbonyl]phenyl]-2-propanesulfonamide
- CAS:918505-61-0
- MF:C22H18F2N4O3S
- Structure:

- Chemical Name:Nsc66811
- CAS:6964-62-1
- MF:C23H20N2O
- Structure:

- Chemical Name:VCH-916
- CAS:1200133-34-1
- MF:C26H36KNO4S
- Structure:

- Chemical Name:GW791343 (HCl)
- CAS:1019779-04-4
- MF:C20H24F2N4O
- Structure:

- Chemical Name:Vaniprevir
- CAS:923590-37-8
- MF:C38H55N5O9S
- Structure:

- Chemical Name:1-(4-Methoxyphenyl)-2-methyl-3-nitro-1H-indol-6-ol
- CAS:147591-46-6
- MF:C16H14N2O4
- Structure:

- Chemical Name:Losartan-d4 Carboxylic Acid
- CAS:1246820-62-1
- MF:C22H21ClN6O2
- Structure:

- Chemical Name:Delamanid
- CAS:681492-22-8
- MF:C25H25F3N4O6
- Structure:

- Chemical Name:MK-8998
- CAS:953778-58-0
- MF:C20H23F3N2O2
- Structure:

- Chemical Name:Amg 517
- CAS:659730-32-2
- MF:C20H13F3N4O2S
- Structure:

- Chemical Name:AC-55541
- CAS:916170-19-9
- MF:C25H20BrN5O3
- Structure:

- Chemical Name:Unii-950o97nupo
- CAS:377727-87-2
- MF:C25H29N9O3
- Structure:

- Chemical Name:N-[trans-4-[2-(6-Cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide
- CAS:215803-78-4
- MF:C28H30N4O
- Structure:

- Chemical Name:BML-210
- CAS:537034-17-6
- MF:C20H25N3O2
- Structure:

- Chemical Name:FIPI
- CAS:939055-18-2
- MF:C23H24FN5O2
- Structure:

- Chemical Name:2-Amino-6-[2-(cyclopropylmethoxy)-6-hydroxyphenyl]-4-(4-piperidinyl)-3-pyridinecarbonitrile hydrochloride
- CAS:406209-26-5
- MF:C21H25ClN4O2
- Structure:

- Chemical Name:SCH-900776
- CAS:891494-64-7
- MF:C15H18BrN7
- Structure:

- Chemical Name:AnaMorelin hydrochloride
- CAS:861998-00-7
- MF:C31H43ClN6O3
- Structure:

- Chemical Name:BN-2629
- CAS:232931-57-6
- MF:C31H32N4O6
- Structure:

- Chemical Name:ARRY-520
- CAS:885060-09-3
- MF:C20H22F2N4O2S
- Structure:

- Chemical Name:KN-92 (hydrochloride)
- CAS:1431698-47-3
- MF:C24H26Cl2N2O3S
- Structure:

- Chemical Name:PSN632408
- CAS:857652-30-3
- MF:C18H24N4O4
- Structure:

- Chemical Name:CEP-32496
- CAS:1227678-26-3
- MF:C24H23ClF3N5O5
- Structure:

- Chemical Name:A 804598
- CAS:1125758-85-1
- MF:C19H17N5
- Structure:

- Chemical Name:NDT 9513727
- CAS:439571-48-9
- MF:C36H35N3O4
- Structure:

- Chemical Name:(E)-1-(3-chloro-4-fluorophenyl)-4-((5-nitrofuran-2-yl)Methylene)pyrazolidine-3,5-dione
- CAS:423148-78-1
- MF:C14H7ClFN3O5
- Structure:

- Chemical Name:GAP 27
- CAS:198284-64-9
- MF:C60H101N15O17
- Structure:

- Chemical Name:AST-1306
- CAS:897383-62-9
- MF:C24H18ClFN4O2
- Structure:

- Chemical Name:GSK-25
- CAS:874119-56-9
- MF:C24H16Cl2F2N6O
- Structure:

- Chemical Name:1alpha, 24, 25-Trihydroxy VD2
- CAS:457048-34-9
- MF:C28H44O4
- Structure:

- Chemical Name:BAY 61-3606 (dihydrochloride)
- CAS:648903-57-5
- MF:C20H20Cl2N6O3
- Structure:

- Chemical Name:BIX02189
- CAS:1265916-41-3
- MF:C27H28N4O2
- Structure:

- Chemical Name:PDK1 inhibitor
- CAS:1001409-50-2
- MF:C28H22F2N4O4
- Structure:

- Chemical Name:Belumosudil
- CAS:911417-87-3
- MF:C26H24N6O2
- Structure:

- Chemical Name:5-PyriMidinecarboxaMide, 2-[[2-(3-chloro-4-hydroxyphenyl)ethyl]aMino]-4-[(phenylMethyl)aMino]-
- CAS:919486-40-1
- MF:C20H20ClN5O2
- Structure:

- Chemical Name:BAY-57-1293
- CAS:348086-71-5
- MF:C18H18N4O3S2
- Structure:

- Chemical Name:BenzenesulfonaMide, 5-(phenylsulfonyl)-N-4-piperidinyl-2-(trifluoroMethyl)-
- CAS:915759-45-4
- MF:C18H19F3N2O4S2
- Structure:

- Chemical Name:ELN 441958
- CAS:913064-47-8
- MF:C29H29ClN4O2
- Structure:

- Chemical Name:GeMigliptin
- CAS:911637-19-9
- MF:C18H19F8N5O2
- Structure:

- Chemical Name:GLI1-Mediated transcription inhibitor
- CAS:496794-70-8
- MF:C24H23ClN4O3
- Structure:

- Chemical Name:LOR 253
- CAS:916151-99-0
- MF:C22H14FN5
- Structure:

- Chemical Name:MibaMpator
- CAS:375345-95-2
- MF:C21H30N2O4S2
- Structure:

- Chemical Name:N3PT
- CAS:13860-66-7
- MF:C13H19Cl2N3OS
- Structure:

- Chemical Name:Opicapone
- CAS:923287-50-7
- MF:C15H10Cl2N4O6
- Structure:

- Chemical Name:PPQ-102
- CAS:931706-15-9
- MF:C26H22N4O3
- Structure:

- Chemical Name:Repertaxin
- CAS:266359-83-5
- MF:C14H21NO3S
- Structure:

- Chemical Name:XL-647
- CAS:781613-23-8
- MF:C24H25Cl2FN4O2
- Structure:

- Chemical Name:PF 04447943
- CAS:1082744-20-4
- MF:C20H25N7O2
- Structure:

- Chemical Name:Hederagenin 3-O-α-L-rhaMnopyranosyl(1→2)-(β-D-glucopyranosyl(1→4))-α-L-arabinopyranoside
- CAS:68027-15-6
- MF:C47H76O17
- Structure:

- Chemical Name:L 2-401
- CAS:883050-24-6
- MF:C16H13FN2O2S
- Structure:

- Chemical Name:Roniciclib
- CAS:1223498-69-8
- MF:C18H21F3N4O3S
- Structure:

- Chemical Name:(2S)-Methyl 2-(2-chlorophenyl)-2-(2-oxo-7,7a-dihydrothieno[3,2-c]pyridin-5(2H,4H,6H)-yl)acetate
- CAS:1147350-75-1
- MF:C16H16ClNO3S
- Structure:

- Chemical Name:AT 7867 dihydrochloride
- CAS:1431697-86-7
- MF:C20H21Cl2N3
- Structure:

- Chemical Name:CC401 HCl
- CAS:1438391-30-0
- MF:C22H25ClN6O
- Structure:

- Chemical Name:c-Met inhibitor 1
- CAS:1357072-61-7
- MF:C17H14N8S
- Structure:

- Chemical Name:XR9576
- CAS:625375-83-9
- MF:C39H42N4O9S
- Structure:

- Chemical Name:QNZ-46
- CAS:1237744-13-6
- MF:C24H17N3O6
- Structure:

- Chemical Name:LH-846
- CAS:639052-78-1
- MF:C16H13ClN2OS
- Structure:

- Chemical Name:PF 4618433
- CAS:1166393-85-6
- MF:C24H27N7O2
- Structure:

- Chemical Name:Pyrido[2,3-d]pyriMidin-7(8H)-one, 6-(2,4-dichlorophenyl)-8-ethyl-2-[[3-fluoro-4-(1-piperazinyl)phenyl]aMino]-
- CAS:1232030-35-1
- MF:C25H23Cl2FN6O
- Structure:

- Chemical Name:LY 2606368
- CAS:1234015-52-1
- MF:C18H19N7O2
- Structure:

- Chemical Name:ADH 1
- CAS:229971-81-7
- MF:C22H34N8O6S2