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Agonist Inhibitors
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- Structure:

- Chemical Name:LY2334737
- CAS:892128-60-8
- MF:C17H25F2N3O5
- Structure:

- Chemical Name:ML281
- CAS:1404437-62-2
- MF:C22H19N3O2S
- Structure:

- Chemical Name:O-Propargyl-PuroMycin
- CAS:1416561-90-4
- MF:C24H29N7O5
- Structure:

- Chemical Name:20-O-Acetylingenol-3-angelate
- CAS:82425-35-2
- MF:C27H36O7
- Structure:

- Chemical Name:AICAR (phosphate)
- CAS:681006-28-0
- MF:C9H17N4O9P
- Structure:

- Chemical Name:LHW090-A7
- CAS:1308256-94-1
- MF:C20H22ClNO4
- Structure:

- Chemical Name:ZLN005
- CAS:49671-76-3
- MF:C17H18N2
- Structure:

- Chemical Name:ADIPORON
- CAS:924416-43-3
- MF:C27H28N2O3
- Structure:

- Chemical Name:LEE011 (hydrochloride)
- CAS:1211443-80-9
- MF:C23H31ClN8O
- Structure:

- Chemical Name:ML314
- CAS:1448895-09-7
- MF:C24H28N4O3
- Structure:

- Chemical Name:Emixustat hydrochloride
- CAS:1141934-97-5
- MF:C16H26ClNO2
- Structure:

- Chemical Name:1-tert-butyl-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyriMidin-4-aMine hydrochloride
- CAS:956025-47-1
- MF:C19H20ClN5
- Structure:

- Chemical Name:Atglistatin
- CAS:1469924-27-3
- MF:C17H21N3O
- Structure:

- Chemical Name:PCI-32765 (RaceMate)
- CAS:936563-87-0
- MF:C25H24N6O2
- Structure:

- Chemical Name:GNE-7915 (tosylate)
- CAS:2070015-00-6
- MF:C26H29F4N5O6S
- Structure:

- Chemical Name:4EGI-1
- CAS:315706-13-9
- MF:C18H12Cl2N4O4S
- Structure:

- Chemical Name:2-AMino-6-chloro-α-cyano-3-(ethoxycarbonyl)-4H-1-benzopyran-4-acetic Acid Ethyl Ester
- CAS:305834-79-1
- MF:C17H17ClN2O5
- Structure:

- Chemical Name:Thiazolidine-4-carboxylic acid
- CAS:444-27-9
- MF:C4H7NO2S
- Structure:

- Chemical Name:RO5126766(CH5126766)
- CAS:946128-88-7
- MF:C21H18FN5O5S
- Structure:

- Chemical Name:I-CBP112
- CAS:1640282-31-0
- MF:C27H36N2O5
- Structure:

- Chemical Name:IWP-3
- CAS:687561-60-0
- MF:C22H17FN4O2S3
- Structure:

- Chemical Name:Cerdulatinib
- CAS:1198300-79-6
- MF:C20H27N7O3S
- Structure:

- Chemical Name:HG-14-10-04
- CAS:1356962-34-9
- MF:C29H34ClN7O
- Structure:

- Chemical Name:kb-NB77-78
- CAS:1350622-33-1
- MF:C18H25NO3Si
- Structure:

- Chemical Name:NIBR189
- CAS:1599432-08-2
- MF:C21H21BrN2O3
- Structure:

- Chemical Name:VT-464
- CAS:1610537-15-9
- MF:C18H17F4N3O3
- Structure:

- Chemical Name:Gilteritinib
- CAS:1254053-43-4
- MF:C29H44N8O3
- Structure:

- Chemical Name:Chitinase-IN-1
- CAS:1579991-61-9
- MF:C18H16N4O2S
- Structure:

- Chemical Name:E-7449
- CAS:1140964-99-3
- MF:C18H15N5O
- Structure:

- Chemical Name:ZLN-024
- CAS:723249-01-2
- MF:C13H13BrN2OS
- Structure:

- Chemical Name:Mutant IDH1-IN-1
- CAS:1355326-21-4
- MF:C30H31FN4O2
- Structure:

- Chemical Name:LP533401 hcl
- CAS:1040526-12-2
- MF:C27H23ClF4N4O3
- Structure:

- Chemical Name:ML224
- CAS:1338824-21-7
- MF:C31H31N3O5
- Structure:

- Chemical Name:6-(octylaMino)pyriMidine-2,4(1H,3H)-dione
- CAS:83797-69-7
- MF:C12H21N3O2
- Structure:

- Chemical Name:BLU9931
- CAS:1538604-68-0
- MF:C26H22Cl2N4O3
- Structure:

- Chemical Name:(E)-4-(5-(2-(3-methylbenzylidene)hydrazinyl)-2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)morpholine
- CAS:1232221-74-7
- MF:C23H23N7O
- Structure:

- Chemical Name:6-amino-1,3-dimethyl-4-(4-(trifluoromethyl)phenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
- CAS:1637739-82-2
- MF:C16H13F3N4O
- Structure:

- Chemical Name:AF38469
- CAS:1531634-31-7
- MF:C15H11F3N2O3
- Structure:

- Chemical Name:IWP 4
- CAS:686772-17-8
- MF:C23H20N4O3S3
- Structure:

- Chemical Name:TH287
- CAS:1609960-30-6
- MF:C11H10Cl2N4
- Structure:

- Chemical Name:N′-[3,5-Bis(trifluoromethyl)phenyl]-N-[4-bromo-2-(2H-tetrazol-5-yl)phenyl]-thiourea
- CAS:956014-19-0
- MF:C16H9BrF6N6S
- Structure:

- Chemical Name:3-(Phenylmethyl)-2-[(1E)-2-(3-pyridinyl)ethenyl]-4(3H)-quinazolinone
- CAS:1290541-46-6
- MF:C22H17N3O
- Structure:

- Chemical Name:3,3',5-TRIIODOTHYROACETIC ACID
- CAS:51-24-1
- MF:C14H9I3O4
- Structure:

- Chemical Name:Cyclosporin H
- CAS:83602-39-5
- MF:C62H111N11O12
- Structure:

- Chemical Name:NIPRADILOL
- CAS:81486-22-8
- MF:C15H22N2O6
- Structure:

- Chemical Name:YHO-13177
- CAS:912287-56-0
- MF:C20H22N2O3S
- Structure:

- Chemical Name:SBI-0206965
- CAS:1884220-36-3
- MF:C21H21BrN4O5
- Structure:

- Chemical Name:AR-13324 (mesylate)
- CAS:1422144-42-0
- MF:C28H27N3O3.2CH4O3S
- Structure:

- Chemical Name:DC_05
- CAS:890643-16-0
- MF:C25H25N3O
- Structure:

- Chemical Name:S1P1 Agonist III
- CAS:1324003-64-6
- MF:C21H16F3N3O3
- Structure:

- Chemical Name:RO8994
- CAS:1309684-94-3
- MF:C31H31Cl2FN4O4
- Structure:

- Chemical Name:1-(1-(3-methoxyphenyl)-7-propoxyindolizin-3-yl)ethanone
- CAS:1693766-04-9
- MF:C20H21NO3
- Structure:

- Chemical Name:RPT-835(alofanib)
- CAS:1612888-66-0
- MF:C19H15N3O6S
- Structure:

- Chemical Name:GSK-2256098
- CAS:1224887-10-8
- MF:C20H23ClN6O2
- Structure:

- Chemical Name:Olmutinib
- CAS:1353550-13-6
- MF:C26H26N6O2S
- Structure:

- Chemical Name:(S)-N-(2-(2-cyano-4,4-difluoropyrrolidin-1-yl)-2-oxoethyl)quinoline-4-carboxamide
- CAS:1448440-52-5
- MF:C17H14F2N4O2
- Structure:

- Chemical Name:Lorediplon
- CAS:917393-39-6
- MF:C20H15FN4O2S
- Structure:

- Chemical Name:PLX8394
- CAS:1393466-87-9
- MF:C25H21F3N6O3S
- Structure:

- Chemical Name:NS-018
- CAS:1239358-86-1
- MF:C21H20FN7
- Structure:

- Chemical Name:A-1331852
- CAS:1430844-80-6
- MF:C38H38N6O3S
- Structure:

- Chemical Name:MI-136
- CAS:1628316-74-4
- MF:C23H21F3N6S
- Structure:

- Chemical Name:PF-04929113 (Mesylate)
- CAS:1173111-67-5
- MF:C26H34F3N5O7S
- Structure:

- Chemical Name:PD-126055 free acid
- CAS:1316755-16-4
- MF:C32H29NO5
- Structure:

- Chemical Name:CP21R7(CP21)
- CAS:125314-13-8
- MF:C19H15N3O2
- Structure:

- Chemical Name:EAI-045
- CAS:1942114-09-1
- MF:C19H14FN3O3S
- Structure:

- Chemical Name:I-BRD9
- CAS:1714146-59-4
- MF:C22H22F3N3O3S2
- Structure:

- Chemical Name:TA-02
- CAS:1784751-19-4
- MF:C20H13F2N3
- Structure:

- Chemical Name:GAL-021
- CAS:1380341-99-0
- MF:C11H22N6O
- Structure:

- Chemical Name:CPI-455
- CAS:1628208-23-0
- MF:C16H14N4O
- Structure:

- Chemical Name:EFT-508
- CAS:1849590-01-7
- MF:C17H20N6O2
- Structure:

- Chemical Name:LTX-315
- CAS:1345407-05-7
- MF:C78H106N18O9
- Structure:

- Chemical Name:1-[(3,4-dichlorophenyl)methyl]-N-[4-(hydroxymethyl)phenyl]-5-methyl-1H-1,2,3-triazole-4-carboxamide
- CAS:1150701-66-8
- MF:C18H16Cl2N4O2
- Structure:

- Chemical Name:ON1231320
- CAS:1312471-39-8
- MF:C22H15F2N5O3S
- Structure:

- Chemical Name:XL-652
- CAS:918348-67-1
- MF:C28H29ClN2O3S
- Structure:

- Chemical Name:CZ415
- CAS:1429639-50-8
- MF:C22H29N5O4S
- Structure:

- Chemical Name:RN-1 (hydrochloride)
- CAS:1781835-13-9
- MF:C23H30ClN3O2
- Structure:

- Chemical Name:HT-2157
- CAS:303149-14-6
- MF:C21H13F3N2O
- Structure:

- Chemical Name:CeMMEC13
- CAS:1790895-25-8
- MF:C19H16N2O4
- Structure:

- Chemical Name:Org-26576
- CAS:1026791-61-6
- MF:C11H12N2O2
- Structure:

- Chemical Name:KYA1797K
- CAS:1956356-56-1
- MF:C17H11KN2O6S2
- Structure:

- Chemical Name:Saccharin 1-methylimidazole (SMI)
- CAS:482333-74-4
- MF:C11H11N3O3S
- Structure:

- Chemical Name:CDD3506
- CAS:197913-15-8
- MF:C22H19N3
- Structure:

- Chemical Name:Thiomyristoyl
- CAS:1429749-41-6
- MF:C34H51N3O3S
- Structure:

- Chemical Name:CeMMEC1
- CAS:440662-09-9
- MF:C19H16N2O4
- Structure:

- Chemical Name:(Z)-2-CARBOXY-4,6-DICHLOROINDOLE-3-(2'-PHENYL-2'-CARBOXY)-ENE
- CAS:161230-88-2
- MF:C18H11Cl2NO4
- Structure:

- Chemical Name:Repotrectinib
- CAS:1802220-02-5
- MF:C18H18FN5O2
- Structure:

- Chemical Name:WIN 55,212-2 MESYLATE
- CAS:131543-23-2
- MF:C28H30N2O6S
- Structure:

- Chemical Name:Takinib
- CAS:1111556-37-6
- MF:C18H18N4O2
- Structure:

- Chemical Name:Estra-4,9-diene-3,17-dione
- CAS:5173-46-6
- MF:C18H22O2
- Structure:

- Chemical Name:NS 1619
- CAS:153587-01-0
- MF:C15H8F6N2O2
- Structure:

- Chemical Name:1H-1,2,4-Triazole-3-carboxylic acid
- CAS:4928-87-4
- MF:C3H3N3O2
- Structure:

- Chemical Name:Doxercalciferol
- CAS:54573-75-0
- MF:C28H44O2
- Structure:

- Chemical Name:N-[2-[4-(2-METHOXYPHENYL)-1-PIPERAZINYL]ETHYL]-N-2-PYRIDINYL-CYCLOHEXANECARBOXAMIDE MALEATE
- CAS:634908-75-1
- MF:C29H38N4O6
- Structure:

- Chemical Name:3-(Methylamino)toluene
- CAS:696-44-6
- MF:C8H11N
- Structure:

- Chemical Name:TAUROURSODEOXYCHOLIC ACID SODIUM SALT
- CAS:35807-85-3
- MF:C26H46NNaO6S
- Structure:

- Chemical Name:2-(4-[(4-METHOXYBENZYL)OXY]PHENYL)ACETONITRILE
- CAS:175135-47-4
- MF:C16H15NO2
- Structure:

- Chemical Name:diABZI STING agonist-1 trihydrochloride
- CAS:2138299-34-8
- MF:C42H52ClN13O7
- Structure:

- Chemical Name:Telratolimod
- CAS:1359993-59-1
- MF:C36H59N5O2
- Structure:

- Chemical Name:NVP-AAM077
- CAS:459836-30-7
- MF:C17H17BrN3O5P
- Structure:

- Chemical Name:L-838417
- CAS:286456-42-6
- MF:C19H19F2N7O