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Agonist Inhibitors

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  • Structure:1542135-76-1
  • Chemical Name:LML-134
  • CAS:1542135-76-1
  • MF:C19H29N5O3


  • Structure:118414-82-7
  • Chemical Name:MK-886
  • CAS:118414-82-7
  • MF:C27H34ClNO2S






  • Structure:79455-30-4
  • Chemical Name:Nicaraven
  • CAS:79455-30-4
  • MF:C15H16N4O2

  • Structure:406205-74-1
  • Chemical Name:BAY 59-3074
  • CAS:406205-74-1
  • MF:C18H13F6NO4S

  • Structure:186544-26-3
  • Chemical Name:LY 344864
  • CAS:186544-26-3
  • MF:C21H22FN3O



  • Structure:223652-90-2
  • Chemical Name:Garenoxacin
  • CAS:223652-90-2
  • MF:C23H20F2N2O4.CH4O3S.H2O

  • Structure:848354-66-5
  • Chemical Name:PTACH
  • CAS:848354-66-5
  • MF:C20H26N2O2S2

  • Structure:171335-80-1
  • Chemical Name:Exatecan
  • CAS:171335-80-1
  • MF:C24H22FN3O4



  • Structure:2410957-04-7
  • Chemical Name:TRV120055
  • CAS:2410957-04-7
  • MF:C34H54N12O7


  • Structure:26171-23-3
  • Chemical Name:Tolmetin
  • CAS:26171-23-3
  • MF:C15H15NO3



  • Structure:7759-35-5
  • Chemical Name:Nestoron
  • CAS:7759-35-5
  • MF:C23H30O4

  • Structure:125602-71-3
  • Chemical Name:BEPOTASTINE
  • CAS:125602-71-3
  • MF:C21H25ClN2O3


  • Structure:574013-66-4
  • Chemical Name:Fexaramine
  • CAS:574013-66-4
  • MF:C32H36N2O3

  • Structure:52128-35-5
  • Chemical Name:Trimetrexate
  • CAS:52128-35-5
  • MF:C19H23N5O3

  • Structure:173997-05-2
  • Chemical Name:Nepicastat
  • CAS:173997-05-2
  • MF:C14H15F2N3S

  • Structure:138071-82-6
  • Chemical Name:Gadobutrol
  • CAS:138071-82-6
  • MF:C18H31N4O9.Gd


  • Structure:509088-69-1
  • Chemical Name:KRP-203
  • CAS:509088-69-1
  • MF:C24H27Cl2NO3S

  • Structure:1146-98-1
  • Chemical Name:Bromindione
  • CAS:1146-98-1
  • MF:C15H9BrO2

  • Structure:69123-90-6
  • Chemical Name:Fiacitabine
  • CAS:69123-90-6
  • MF:C9H11FIN3O4

  • Structure:159634-47-6
  • Chemical Name:MK-677
  • CAS:159634-47-6
  • MF:C27H36N4O5S

  • Structure:88578-07-8
  • Chemical Name:Imoxiterol
  • CAS:88578-07-8
  • MF:C20H25N3O3



  • Structure:289656-45-7
  • Chemical Name:Senicapoc
  • CAS:289656-45-7
  • MF:C20H15F2NO



  • Structure:204697-65-4
  • Chemical Name:BIBN 4096BS
  • CAS:204697-65-4
  • MF:C38H47Br2N9O5

  • Structure:248282-07-7
  • Chemical Name:Laquinimod
  • CAS:248282-07-7
  • MF:C19H18ClN2NaO3



  • Structure:130641-38-2
  • Chemical Name:Bindarit
  • CAS:130641-38-2
  • MF:C19H20N2O3

  • Structure:116686-15-8
  • Chemical Name:FK-3311
  • CAS:116686-15-8
  • MF:C15H13F2NO4S


  • Structure:151823-14-2
  • Chemical Name:Sapacitabine
  • CAS:151823-14-2
  • MF:C26H42N4O5

  • Structure:173937-91-2
  • Chemical Name:atrasentan
  • CAS:173937-91-2
  • MF:C29H38N2O6

  • Structure:53185-12-9
  • Chemical Name:fagomine
  • CAS:53185-12-9
  • MF:C6H13NO3

  • Structure:136164-66-4
  • Chemical Name:E 3330
  • CAS:136164-66-4
  • MF:C21H30O6

  • Structure:131179-95-8
  • Chemical Name:Efaproxiral
  • CAS:131179-95-8
  • MF:C20H22NO4.Na


  • Structure:147366-41-4
  • Chemical Name:MKT 077
  • CAS:147366-41-4
  • MF:C21H22ClN3OS2

  • Structure:476-34-6
  • Chemical Name:isoindigotin
  • CAS:476-34-6
  • MF:C16H10N2O2

  • Structure:181630-15-9
  • Chemical Name:Picoplatin
  • CAS:181630-15-9
  • MF:C6H9Cl2N2Pt


  • Structure:199113-98-9
  • Chemical Name:Balaglitazone
  • CAS:199113-98-9
  • MF:C20H17N3O4S



  • Structure:857402-23-4
  • Chemical Name:Retaspimycin
  • CAS:857402-23-4
  • MF:C31H45N3O8

  • Structure:141136-84-7
  • Chemical Name:FLLRN
  • CAS:141136-84-7
  • MF:C31H51N9O7

  • Structure:112093-28-4
  • Chemical Name:Avacopan
  • CAS:112093-28-4
  • MF:C25H27NO2

  • Structure:134381-21-8
  • Chemical Name:EPOXOMICIN
  • CAS:134381-21-8
  • MF:C28H50N4O7


  • Structure:492-38-6
  • Chemical Name:Atropic acid
  • CAS:492-38-6
  • MF:C9H8O2

  • Structure:226954-04-7
  • Chemical Name:AC-5216
  • CAS:226954-04-7
  • MF:C23H23N5O2

  • Structure:224452-66-8
  • Chemical Name:RETAPAMULIN
  • CAS:224452-66-8
  • MF:C30H47NO4S

  • Structure:1082743-70-1
  • Chemical Name:PDE-9
  • CAS:1082743-70-1
  • MF:C22H27N5O2



  • Structure:182167-02-8
  • Chemical Name:Sch 57068
  • CAS:182167-02-8
  • MF:C29H31NO4


  • Structure:402567-16-2
  • Chemical Name:Firategrast
  • CAS:402567-16-2
  • MF:C27H27F2NO6

  • Structure:241479-67-4
  • Chemical Name:Isavuconazole
  • CAS:241479-67-4
  • MF:C22H17F2N5OS



  • Structure:19608-29-8
  • Chemical Name:Clascoterone
  • CAS:19608-29-8
  • MF:C24H34O5











  • Structure:1210004-12-8
  • Chemical Name:JZL 195
  • CAS:1210004-12-8
  • MF:C24H23N3O5

  • Structure:283159-90-0
  • Chemical Name:valiphenal
  • CAS:283159-90-0
  • MF:C19H27ClN2O5

  • Structure:1096708-71-2
  • Chemical Name:MLN 2480
  • CAS:1096708-71-2
  • MF:C17H12Cl2F3N7O2S






  • Structure:854601-70-0
  • Chemical Name:Naloxegol
  • CAS:854601-70-0
  • MF:C34H53NO11

  • Structure:1124381-69-6
  • Chemical Name:S-99
  • CAS:1124381-69-6
  • MF:C16H15F3N6O

  • Structure:761436-81-1
  • Chemical Name:ALK inhibitor 1
  • CAS:761436-81-1
  • MF:C23H28BrN7O3S