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Agonist Inhibitors
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- Structure:

- Chemical Name:LML-134
- CAS:1542135-76-1
- MF:C19H29N5O3
- Structure:

- Chemical Name:4-(2-HYDROXYETHYLAMINO)-2-(4-METHOXYPHENYLAMINO)-PYRIMIDINE HYDROCHLORIDE
- CAS:1049741-55-0
- MF:C13H17ClN4O2
- Structure:

- Chemical Name:MK-886
- CAS:118414-82-7
- MF:C27H34ClNO2S
- Structure:

- Chemical Name:4-[4-(4-CHLOROPHENYL)-4-HYDROXY-1-PIPERIDINYL]-1-(4-FLUOROPHENYL)-1-BUTANONE HYDROCHLORIDE
- CAS:1511-16-6
- MF:C21H24Cl2FNO2
- Structure:

- Chemical Name:DL-ADRENALINE HYDROCHLORIDE
- CAS:329-63-5
- MF:C9H14ClNO3
- Structure:

- Chemical Name:Potassium canrenoate
- CAS:2181-04-6
- MF:C11H15KO2
- Structure:

- Chemical Name:6-[4-(2-PIPERIDIN-1-YLETHOXY)PHENYL]-3-PYRIDIN-4-YLPYRAZOLO[1,5-A]PYRIMIDINE
- CAS:866405-64-3
- MF:C24H25N5O
- Structure:

- Chemical Name:(2'Z,3'E)-6-BROMOINDIRUBIN-3'-ACETOXIME
- CAS:667463-85-6
- MF:C18H12BrN3O3
- Structure:

- Chemical Name:Nicaraven
- CAS:79455-30-4
- MF:C15H16N4O2
- Structure:

- Chemical Name:BAY 59-3074
- CAS:406205-74-1
- MF:C18H13F6NO4S
- Structure:

- Chemical Name:LY 344864
- CAS:186544-26-3
- MF:C21H22FN3O
- Structure:

- Chemical Name:GABOXADOL HYDROCHLORIDE
- CAS:85118-33-8
- MF:C6H9ClN2O2
- Structure:

- Chemical Name:1-(4-hydroxy-3-methoxyphenyl)decan-5-one
- CAS:27113-22-0
- MF:C17H26O3
- Structure:

- Chemical Name:Garenoxacin
- CAS:223652-90-2
- MF:C23H20F2N2O4.CH4O3S.H2O
- Structure:

- Chemical Name:PTACH
- CAS:848354-66-5
- MF:C20H26N2O2S2
- Structure:

- Chemical Name:Exatecan
- CAS:171335-80-1
- MF:C24H22FN3O4
- Structure:

- Chemical Name:SA-4503,1-(3,4-DIMETHOXYPHENETHYL)-4-(3-PHENYLPROPYL)PIPERAZINE DIHYDROCHLORIDE
- CAS:165377-44-6
- MF:C23H32N2O2.2ClH
- Chemical Name:Palmitoyl Pentapeptide
- CAS:
- MF:
- Structure:

- Chemical Name:TRV120055
- CAS:2410957-04-7
- MF:C34H54N12O7
- Structure:

- Chemical Name:4-(2,3-DIMETHYL-BENZYL)-1H-IMIDAZOLE
- CAS:76631-46-4
- MF:C12H14N2
- Structure:

- Chemical Name:Tolmetin
- CAS:26171-23-3
- MF:C15H15NO3
- Structure:

- Chemical Name:2,5-DiMethoxy-4-iodophenethylaMine Hydrochloride
- CAS:64584-32-3
- MF:C10H15ClINO2
- Structure:

- Chemical Name:1,3-Bis(4-aminophenyl)urea
- CAS:4550-72-5
- MF:C13H14N4O
- Structure:

- Chemical Name:Nestoron
- CAS:7759-35-5
- MF:C23H30O4
- Structure:

- Chemical Name:BEPOTASTINE
- CAS:125602-71-3
- MF:C21H25ClN2O3
- Structure:

- Chemical Name:TRIMIPRAMINE MALEATE SALT
- CAS:521-78-8
- MF:C24H30N2O4
- Structure:

- Chemical Name:Fexaramine
- CAS:574013-66-4
- MF:C32H36N2O3
- Structure:

- Chemical Name:Trimetrexate
- CAS:52128-35-5
- MF:C19H23N5O3
- Structure:

- Chemical Name:Nepicastat
- CAS:173997-05-2
- MF:C14H15F2N3S
- Structure:

- Chemical Name:Gadobutrol
- CAS:138071-82-6
- MF:C18H31N4O9.Gd
- Structure:

- Chemical Name:7-METHOXYISOFLAVONE
- CAS:1621-56-3
- MF:C16H12O3
- Structure:

- Chemical Name:KRP-203
- CAS:509088-69-1
- MF:C24H27Cl2NO3S
- Structure:

- Chemical Name:Bromindione
- CAS:1146-98-1
- MF:C15H9BrO2
- Structure:

- Chemical Name:Fiacitabine
- CAS:69123-90-6
- MF:C9H11FIN3O4
- Structure:

- Chemical Name:MK-677
- CAS:159634-47-6
- MF:C27H36N4O5S
- Structure:

- Chemical Name:Imoxiterol
- CAS:88578-07-8
- MF:C20H25N3O3
- Structure:

- Chemical Name:5-Aziridino-2,4-dinitrobenzamide
- CAS:21919-05-1
- MF:C9H8N4O5
- Structure:

- Chemical Name:(2S)-2-[[4-[(2-fluorophenyl)methoxy]phenyl]methylamino]propanamide
- CAS:133865-88-0
- MF:C17H19FN2O2
- Structure:

- Chemical Name:Senicapoc
- CAS:289656-45-7
- MF:C20H15F2NO
- Structure:

- Chemical Name:Pirmenol hydrochloride
- CAS:61477-94-9
- MF:C22H31ClN2O
- Structure:

- Chemical Name:1-naphthylacetylspermine
- CAS:122306-11-0
- MF:C22H34N4O
- Structure:

- Chemical Name:BIBN 4096BS
- CAS:204697-65-4
- MF:C38H47Br2N9O5
- Structure:

- Chemical Name:Laquinimod
- CAS:248282-07-7
- MF:C19H18ClN2NaO3
- Structure:

- Chemical Name:4,5,6,7-TETRABROMOBENZOTRIAZOLE
- CAS:17374-26-4
- MF:C6HBr4N3
- Structure:

- Chemical Name:PMPA(NAALADaseinhibitor)
- CAS:173039-10-6
- MF:C6H11O7P
- Structure:

- Chemical Name:Bindarit
- CAS:130641-38-2
- MF:C19H20N2O3
- Structure:

- Chemical Name:FK-3311
- CAS:116686-15-8
- MF:C15H13F2NO4S
- Structure:

- Chemical Name:4-(cyclohexylsulfamoyl)benzoic acid
- CAS:6314-70-1
- MF:C13H17NO4S
- Structure:

- Chemical Name:Sapacitabine
- CAS:151823-14-2
- MF:C26H42N4O5
- Structure:

- Chemical Name:atrasentan
- CAS:173937-91-2
- MF:C29H38N2O6
- Structure:

- Chemical Name:fagomine
- CAS:53185-12-9
- MF:C6H13NO3
- Structure:

- Chemical Name:E 3330
- CAS:136164-66-4
- MF:C21H30O6
- Structure:

- Chemical Name:Efaproxiral
- CAS:131179-95-8
- MF:C20H22NO4.Na
- Chemical Name:ODN 2006
- CAS:
- MF:
- Structure:

- Chemical Name:MKT 077
- CAS:147366-41-4
- MF:C21H22ClN3OS2
- Structure:

- Chemical Name:isoindigotin
- CAS:476-34-6
- MF:C16H10N2O2
- Structure:

- Chemical Name:Picoplatin
- CAS:181630-15-9
- MF:C6H9Cl2N2Pt
- Structure:

- Chemical Name:[2R-(2a,3b,11bb)]-1,3,4,6,7,11b-Hexahydro-9,10-dimethoxy-3-(2-methylpropyl)-2H-benzo[a]quinolizin-2-ol
- CAS:85081-18-1
- MF:C19H29NO3
- Structure:

- Chemical Name:Balaglitazone
- CAS:199113-98-9
- MF:C20H17N3O4S
- Structure:

- Chemical Name:BITHIONOL SULFOXIDE
- CAS:844-26-8
- MF:C12H6Cl4O3S
- Structure:

- Chemical Name:Ethyl 2-amino-8-(perfluoroethyl)-3H-benzo[b]azepine-4-carboxylate
- CAS:926927-42-6
- MF:C15H13F5N2O2
- Structure:

- Chemical Name:Retaspimycin
- CAS:857402-23-4
- MF:C31H45N3O8
- Structure:

- Chemical Name:FLLRN
- CAS:141136-84-7
- MF:C31H51N9O7
- Structure:

- Chemical Name:Avacopan
- CAS:112093-28-4
- MF:C25H27NO2
- Structure:

- Chemical Name:EPOXOMICIN
- CAS:134381-21-8
- MF:C28H50N4O7
- Structure:

- Chemical Name:Glycochenodeoxycholic Acid
- CAS:640-79-9
- MF:C26H43NO5
- Structure:

- Chemical Name:Atropic acid
- CAS:492-38-6
- MF:C9H8O2
- Structure:

- Chemical Name:AC-5216
- CAS:226954-04-7
- MF:C23H23N5O2
- Structure:

- Chemical Name:RETAPAMULIN
- CAS:224452-66-8
- MF:C30H47NO4S
- Structure:

- Chemical Name:PDE-9
- CAS:1082743-70-1
- MF:C22H27N5O2
- Structure:

- Chemical Name:N-(1,1-Dimethylethyl)-3-[[5-methyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]benzenesulfonamide
- CAS:936091-56-4
- MF:C26H34N6O3S
- Structure:

- Chemical Name:N-(2-Aminophenyl)-N'-phenylheptanediamide
- CAS:537034-15-4
- MF:C19H23N3O2
- Structure:

- Chemical Name:Sch 57068
- CAS:182167-02-8
- MF:C29H31NO4
- Structure:

- Chemical Name:Retaspimycin Hydrochloride
- CAS:857402-63-2
- MF:C31H47N3O8.ClH
- Structure:

- Chemical Name:Firategrast
- CAS:402567-16-2
- MF:C27H27F2NO6
- Structure:

- Chemical Name:Isavuconazole
- CAS:241479-67-4
- MF:C22H17F2N5OS
- Structure:

- Chemical Name:N-[5-(4-Cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-3-pyridinecarboxamide
- CAS:1093222-27-5
- MF:C20H13N5O
- Structure:

- Chemical Name:(+/-)-6-CHLORO-7,8-DIHYDROXY-3-ALLYL-1-PHENYL-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINE HYDROBROMIDE
- CAS:80751-65-1
- MF:C19H20ClNO2
- Structure:

- Chemical Name:Clascoterone
- CAS:19608-29-8
- MF:C24H34O5
- Structure:

- Chemical Name:N-(5-((5-(4-Acetylpiperazine-1-carbonyl)-4-methoxy-2-methylphenyl)thio)thiazol-2-yl)-4-(((3-methylbutan-2-yl)amino)methyl)benzamide
- CAS:439574-61-5
- MF:C31H39N5O4S2
- Structure:

- Chemical Name:(3R,4R)-3-(5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl)-4-(1H-indol-3-yl)pyrrolidine-2,5-dione
- CAS:1000873-98-2
- MF:C23H19N3O2
- Structure:

- Chemical Name:N-Hydroxy-4-[(1,2,3,4-tetrahydro-2-methyl-5H-pyrido[4,3-b]indol-5-yl)methyl]benzamide 2,2,2-Trifluoroacetate
- CAS:1239262-52-2
- MF:C22H22F3N3O4
- Structure:

- Chemical Name:2-(4-(5-(3,4-Diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)ethanolhydrochloride
- CAS:1094042-01-9
- MF:C23H27N3O4
- Structure:

- Chemical Name:3-(2-Chlorophenyl)-2-[2-[6-[(diethylamino)methyl]-2-pyridinyl]ethenyl]-6-fluoro-4(3H)-quinazolinonehydrochloride
- CAS:199655-36-2
- MF:C26H24ClFN4O
- Structure:

- Chemical Name:2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-[4-(1-methylpropyl)phenyl]acetamide
- CAS:332117-28-9
- MF:C19H23N5O3
- Structure:

- Chemical Name:4-[1-Cyclohexyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]-2-pyrimidinaminedihydrochloride
- CAS:950912-80-8
- MF:C19H20FN5.2HCl
- Chemical Name:ARRY-543
- CAS:
- MF:
- Structure:

- Chemical Name:(R)-4-(1-aMinoethyl)-N-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzaMide dihydrochloride
- CAS:173897-44-4
- MF:C16H18Cl2N4O
- Structure:

- Chemical Name:Glutaminase C-IN-1
- CAS:311795-38-7
- MF:C27H27BrN2O
- Structure:

- Chemical Name:JZL 195
- CAS:1210004-12-8
- MF:C24H23N3O5
- Structure:

- Chemical Name:valiphenal
- CAS:283159-90-0
- MF:C19H27ClN2O5
- Structure:

- Chemical Name:MLN 2480
- CAS:1096708-71-2
- MF:C17H12Cl2F3N7O2S
- Structure:

- Chemical Name:4-[6-[[(Furan-2-yl)methyl]amino]imidazo[1,2-b]pyridazin-3-yl]phenol
- CAS:928333-30-6
- MF:C17H14N4O2
- Structure:

- Chemical Name:4-[[[3-(3,4-Dimethoxyphenyl)imidazo[1,2-b]pyridazin-6-yl]amino]methyl]benzenesulfonamide
- CAS:1012343-93-9
- MF:C21H21N5O4S
- Structure:

- Chemical Name:N-[2-Methoxy-4-(4-morpholinyl)phenyl]-2-(3-pyridinyl)-4-thiazolecarboxamide
- CAS:1042672-97-8
- MF:C20H20N4O3S
- Structure:

- Chemical Name:5-[(Z)-(5-Fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-N-[(2S)-2-hydroxy-3-(4-morpholinyl)propyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide (2Z)-2-butenedioate
- CAS:849643-15-8
- MF:C23H27FN4O4.C4H4O4
- Structure:

- Chemical Name:2-[[6-[[[2-(3-Hydroxypropyl)-5-methylphenyl]amino]methyl]-2-[[3-(morpholin-4-yl)propyl]amino]benzimidazol-1-yl]methyl]-6-methylpyridin-3-ol
- CAS:857066-90-1
- MF:C32H42N6O3
- Structure:

- Chemical Name:Naloxegol
- CAS:854601-70-0
- MF:C34H53NO11
- Structure:

- Chemical Name:S-99
- CAS:1124381-69-6
- MF:C16H15F3N6O
- Structure:

- Chemical Name:ALK inhibitor 1
- CAS:761436-81-1
- MF:C23H28BrN7O3S