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Agonist Inhibitors

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  • Structure:1415559-43-1
  • Chemical Name:CDK9 inhibitor
  • CAS:1415559-43-1
  • MF:C26H21N5O4S

  • Structure:1065559-56-9
  • Chemical Name:SMND-309
  • CAS:1065559-56-9
  • MF:C18H14O8


  • Structure:473719-41-4
  • Chemical Name:AMG 487
  • CAS:473719-41-4
  • MF:C32H28F3N5O4

  • Structure:943962-47-8
  • Chemical Name:BMS 303141
  • CAS:943962-47-8
  • MF:C19H15Cl2NO4S

  • Structure:308242-62-8
  • Chemical Name:CNS 7056
  • CAS:308242-62-8
  • MF:C21H19BrN4O2

  • Structure:229476-53-3
  • Chemical Name:EBE-A 22
  • CAS:229476-53-3
  • MF:C17H16BrN3O2

  • Structure:1233948-61-2
  • Chemical Name:EL-102
  • CAS:1233948-61-2
  • MF:C19H16N2O3S2

  • Structure:577778-58-6
  • Chemical Name:Topiroxostat
  • CAS:577778-58-6
  • MF:C13H8N6

  • Structure:361444-66-8
  • Chemical Name:JDTic
  • CAS:361444-66-8
  • MF:C28H39N3O3

  • Structure:1094873-14-9
  • Chemical Name:JNJ 31020028
  • CAS:1094873-14-9
  • MF:C34H36FN5O2

  • Structure:928134-65-0
  • Chemical Name:LCI699
  • CAS:928134-65-0
  • MF:C13H10FN3

  • Structure:1123231-07-1
  • Chemical Name:MAY-262611
  • CAS:1123231-07-1
  • MF:C20H22N4

  • Structure:328232-95-7
  • Chemical Name:MK 0557
  • CAS:328232-95-7
  • MF:C22H19FN4O3

  • Structure:168828-58-8
  • Chemical Name:PNU 100480
  • CAS:168828-58-8
  • MF:C16H20FN3O3S

  • Structure:415713-60-9
  • Chemical Name:RI-1
  • CAS:415713-60-9
  • MF:C14H11Cl3N2O3

  • Structure:618385-01-6
  • Chemical Name:Vorapaxar
  • CAS:618385-01-6
  • MF:C29H33FN2O4



  • Structure:1092539-44-0
  • Chemical Name:SAR131675
  • CAS:1092539-44-0
  • MF:C18H22N4O4

  • Structure:1019331-10-2
  • Chemical Name:S0859
  • CAS:1019331-10-2
  • MF:C29H24ClN3O3S


  • Structure:956590-23-1
  • Chemical Name:UNBS-5162
  • CAS:956590-23-1
  • MF:C17H18N4O3

  • Structure:185039-89-8
  • Chemical Name:PD0166285
  • CAS:185039-89-8
  • MF:C26H27Cl2N5O2

  • Structure:55726-47-1
  • Chemical Name:Enocitabine
  • CAS:55726-47-1
  • MF:C31H55N3O6

  • Structure:737763-37-0
  • Chemical Name:360 A iodide
  • CAS:737763-37-0
  • MF:C27H23IN5O2+

  • Structure:864953-29-7
  • Chemical Name:Fostemsavir
  • CAS:864953-29-7
  • MF:C25H26N7O8P

  • Structure:929007-72-7
  • Chemical Name:DB-07268
  • CAS:929007-72-7
  • MF:C17H15N5O2



  • Structure:1088991-73-4
  • Chemical Name:MK 6096
  • CAS:1088991-73-4
  • MF:C24H25FN4O2


  • Structure:160800-57-7
  • Chemical Name:Auristatin E
  • CAS:160800-57-7
  • MF:C40H69N5O7

  • Structure:1204416-97-6
  • Chemical Name:TMC-647055
  • CAS:1204416-97-6
  • MF:C32H38N4O6S

  • Structure:878141-96-9
  • Chemical Name:S1RA
  • CAS:878141-96-9
  • MF:C20H23N3O2


  • Structure:1327167-19-0
  • Chemical Name:BPR1J-097
  • CAS:1327167-19-0
  • MF:C27H28N6O3S

  • Structure:926037-48-1
  • Chemical Name:Radotinib
  • CAS:926037-48-1
  • MF:C27H21F3N8O

  • Structure:436133-68-5
  • Chemical Name:Kobe-0065
  • CAS:436133-68-5
  • MF:C15H11ClF3N5O4S



  • Structure:1270138-40-3
  • Chemical Name:NSI-189
  • CAS:1270138-40-3
  • MF:C22H30N4O


  • Structure:1456858-58-4
  • Chemical Name:HG-9-91-01
  • CAS:1456858-58-4
  • MF:C32H37N7O3

  • Structure:1426944-49-1
  • Chemical Name:HBX 19818
  • CAS:1426944-49-1
  • MF:C25H28ClN3O


  • Structure:1401033-86-0
  • Chemical Name:AMG 925
  • CAS:1401033-86-0
  • MF:C26H29N7O2





  • Structure:1380672-07-0
  • Chemical Name:G007-LK
  • CAS:1380672-07-0
  • MF:C25H16ClN7O3S



  • Structure:1220699-06-8
  • Chemical Name:PF-04979064
  • CAS:1220699-06-8
  • MF:C24H26N6O3

  • Structure:891025-25-5
  • Chemical Name:BAMB-4
  • CAS:891025-25-5
  • MF:C15H12N2O2

  • Structure:1047634-63-8
  • Chemical Name:GSK2110183
  • CAS:1047634-63-8
  • MF:C18H16Cl2F2N4OS

  • Structure:1401242-74-7
  • Chemical Name:ML277
  • CAS:1401242-74-7
  • MF:C23H25N3O4S2


  • Structure:944118-01-8
  • Chemical Name:Peficitinib
  • CAS:944118-01-8
  • MF:C18H22N4O2


  • Structure:191089-59-5
  • Chemical Name:K-7174
  • CAS:191089-59-5
  • MF:C33H48N2O6

  • Structure:1000023-04-0
  • Chemical Name:Voruciclib
  • CAS:1000023-04-0
  • MF:C22H19ClF3NO5

  • Structure:1627494-13-6
  • Chemical Name:AZD8186
  • CAS:1627494-13-6
  • MF:C24H25F2N3O4

  • Structure:1616113-45-1
  • Chemical Name:VRT-1353385
  • CAS:1616113-45-1
  • MF:C35H39NO11

  • Structure:1608125-21-8
  • Chemical Name:AMG319
  • CAS:1608125-21-8
  • MF:C21H16FN7

  • Structure:23146-22-7
  • Chemical Name:IQ-1 sodium
  • CAS:23146-22-7
  • MF:C15H9N3O

  • Structure:31083-55-3
  • Chemical Name:NSC 600157
  • CAS:31083-55-3
  • MF:C15H9NO2



  • Structure:1508250-71-2
  • Chemical Name:EGF816
  • CAS:1508250-71-2
  • MF:C26H31ClN6O2

  • Structure:956274-94-5
  • Chemical Name:mavatrep
  • CAS:956274-94-5
  • MF:C25H21F3N2O

  • Structure:56632-39-4
  • Chemical Name:BHPI
  • CAS:56632-39-4
  • MF:C21H17NO3

  • Structure:1228013-30-6
  • Chemical Name:CC-223
  • CAS:1228013-30-6
  • MF:C21H27N5O3

  • Structure:1443763-60-7
  • Chemical Name:Mps1-IN-5
  • CAS:1443763-60-7
  • MF:C29H26FN5O4S

  • Structure:1415716-58-3
  • Chemical Name:TG6-10-1
  • CAS:1415716-58-3
  • MF:C23H23F3N2O4

  • Structure:115088-06-7
  • Chemical Name:SPDB
  • CAS:115088-06-7
  • MF:C13H14N2O4S2

  • Structure:181223-80-3
  • Chemical Name:DEL-22379
  • CAS:181223-80-3
  • MF:C26H28N4O3

  • Structure:1821496-27-8
  • Chemical Name:BDA-366
  • CAS:1821496-27-8
  • MF:C25H29N3O4

  • Structure:1174161-86-4
  • Chemical Name:SCR-1481B1
  • CAS:1174161-86-4
  • MF:C28H29ClF2N5O10P


  • Structure:1297537-33-7
  • Chemical Name:ORM-15341
  • CAS:1297537-33-7
  • MF:C19H17ClN6O2


  • Structure:1627709-94-7
  • Chemical Name:LJI308
  • CAS:1627709-94-7
  • MF:C21H18F2N2O2

  • Structure:1661839-45-7
  • Chemical Name:CCT251545
  • CAS:1661839-45-7
  • MF:C23H24ClN5O

  • Structure:878978-76-8
  • Chemical Name:ML-098
  • CAS:878978-76-8
  • MF:C19H19NO3

  • Structure:1243245-18-2
  • Chemical Name:GNF-6231
  • CAS:1243245-18-2
  • MF:C24H25FN6O2

  • Structure:1616391-87-7
  • Chemical Name:GSK591
  • CAS:1616391-87-7
  • MF:C22H28N4O2

  • Structure:374913-63-0
  • Chemical Name:Madrasin
  • CAS:374913-63-0
  • MF:C16H17N5O2

  • Structure:1434048-34-6
  • Chemical Name:GDC-0853
  • CAS:1434048-34-6
  • MF:C37H44N8O4

  • Structure:1621862-70-1
  • Chemical Name:CPI-1205
  • CAS:1621862-70-1
  • MF:C27H33F3N4O3

  • Structure:342639-96-7
  • Chemical Name:KRIBB11
  • CAS:342639-96-7
  • MF:C13H12N6O2



  • Structure:1632118-69-4
  • Chemical Name:BAR 501
  • CAS:1632118-69-4
  • MF:C26H46O3

  • Structure:1250963-36-0
  • Chemical Name:CLR1501
  • CAS:1250963-36-0
  • MF:C38H59BF2N3O3P

  • Structure:924473-59-6
  • Chemical Name:T5601640
  • CAS:924473-59-6
  • MF:C19H14F3N3O3

  • Structure:1021497-97-1
  • Chemical Name:KR-33494
  • CAS:1021497-97-1
  • MF:C20H18BrN3O3S

  • Structure:1610759-22-2
  • Chemical Name:CFI-402257
  • CAS:1610759-22-2
  • MF:C28H30N6O3

  • Structure:1304630-27-0
  • Chemical Name:NGP 555
  • CAS:1304630-27-0
  • MF:C23H23FN4S