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Agonist Inhibitors
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- Structure:

- Chemical Name:KDU691
- CAS:1513879-19-0
- MF:C22H18ClN5O2
- Structure:

- Chemical Name:4-PHENYLAMINO-6,7-DIMETHOXYQUINAZOLINE
- CAS:21561-09-1
- MF:C16H15N3O2
- Structure:

- Chemical Name:5,5-Dimethyloxazolidine-2,4-dione
- CAS:695-53-4
- MF:C5H7NO3
- Structure:

- Chemical Name:SU5402
- CAS:215543-92-3
- MF:C17H16N2O3
- Structure:

- Chemical Name:5BETA-PREGNANE-3ALPHA,20ALPHA-DIOL
- CAS:80-92-2
- MF:C21H36O2
- Chemical Name:PP2
- CAS:
- MF:
- Structure:

- Chemical Name:TONABERSAT
- CAS:175013-84-0
- MF:C20H19ClFNO4
- Structure:

- Chemical Name:BAPTA-AM
- CAS:139890-68-9
- MF:C25H28N2O12
- Structure:

- Chemical Name:R-121,919
- CAS:195055-03-9
- MF:C22H32N6
- Structure:

- Chemical Name:Menbutone
- CAS:3562-99-0
- MF:C15H14O4
- Structure:

- Chemical Name:SB 269970 HYDROCHLORIDE
- CAS:201038-74-6
- MF:C18H28N2O3S
- Structure:

- Chemical Name:4-KETO 13-CIS-RETINOIC ACID METHYL ESTER
- CAS:71748-57-7
- MF:C21H28O3
- Structure:

- Chemical Name:1H-Indole, 4-[4-[(2-chlorophenyl)methyl]-1-piperazinyl]-
- CAS:334974-31-1
- MF:C19H20ClN3
- Structure:

- Chemical Name:JAK INHIBITOR I
- CAS:457081-03-7
- MF:C18H16FN3O
- Structure:

- Chemical Name:PIROMIDIC ACID
- CAS:19562-30-2
- MF:C14H16N4O3
- Structure:

- Chemical Name:CALPAIN INHIBITOR III
- CAS:88191-84-8
- MF:C22H26N2O4
- Structure:

- Chemical Name:6-(4-FLUOROPHENYL)-2,3-DIHYDRO-5-(4-PYRIDINYL)IMIDAZO[2,1-B]THIAZOLE DIHYDROCHLORIDE
- CAS:72873-74-6
- MF:C16H12FN3S
- Structure:

- Chemical Name:Fenoldopam mesylate
- CAS:67227-57-0
- MF:C17H20ClNO6S
- Structure:

- Chemical Name:4'-HYDROXYPHENYL CARVEDILOL-D5
- CAS:1261395-96-3
- MF:C24H26N2O5
- Structure:

- Chemical Name:H-SER-LEU-ILE-GLY-LYS-VAL-OH
- CAS:202933-49-1
- MF:C28H53N7O8
- Structure:

- Chemical Name:ibopamine
- CAS:66195-31-1
- MF:C17H25NO4
- Structure:

- Chemical Name:TRIPROLIDINE HYDROCHLORIDE
- CAS:550-70-9
- MF:C19H23ClN2
- Structure:

- Chemical Name:2(3H)-BENZOXAZOLONE, 7-(4-METHYL-1-PIPERAZINYL)-, MONOHYDROCHLORIDE
- CAS:269718-83-4
- MF:C12H16ClN3O2
- Structure:

- Chemical Name:FARAMPATOR
- CAS:211735-76-1
- MF:C12H13N3O2
- Structure:

- Chemical Name:Cevimelinehydrochloride
- CAS:153504-70-2
- MF:C10H20ClNO2S
- Structure:

- Chemical Name:Apricitabine
- CAS:160707-69-7
- MF:C8H11N3O3S
- Structure:

- Chemical Name:Dimethylenastron
- CAS:863774-58-7
- MF:C16H18N2O2S
- Structure:

- Chemical Name:Forodesine
- CAS:209799-67-7
- MF:C11H14N4O4
- Structure:

- Chemical Name:Ametantrone
- CAS:64862-96-0
- MF:C22H28N4O4
- Structure:

- Chemical Name:Fexinidazole
- CAS:59729-37-2
- MF:C12H13N3O3S
- Structure:

- Chemical Name:ZM 241385
- CAS:139180-30-6
- MF:C16H15N7O2
- Structure:

- Chemical Name:ACPA
- CAS:229021-64-1
- MF:C23H37NO
- Structure:

- Chemical Name:Etimizol
- CAS:64-99-3
- MF:C9H14N4O2
- Structure:

- Chemical Name:laxogenin
- CAS:1177-71-5
- MF:C27H42O4
- Structure:

- Chemical Name:Pretomanid
- CAS:187235-37-6
- MF:C14H12F3N3O5
- Structure:

- Chemical Name:YS 49
- CAS:132836-42-1
- MF:C20H20BrNO2
- Structure:

- Chemical Name:Aurothioglucose
- CAS:12192-57-3
- MF:C6H11AuO5S
- Structure:

- Chemical Name:H-D-Phe-Pip-Arg-pNA acetate
- CAS:115388-96-0
- MF:C29H40N8O7
- Structure:

- Chemical Name:avosentan
- CAS:290815-26-8
- MF:C23H21N5O5S
- Structure:

- Chemical Name:Terutroban
- CAS:165538-40-9
- MF:C20H22ClNO4S
- Structure:

- Chemical Name:IMISOPASEM MANGANESE
- CAS:218791-21-0
- MF:C21H35N5.Cl2Mn
- Structure:

- Chemical Name:Levomilnacipran
- CAS:96847-55-1
- MF:C15H22N2O
- Structure:

- Chemical Name:Tasimelteon
- CAS:609799-22-6
- MF:C15H19NO2
- Structure:

- Chemical Name:Methanone, [4-(2-chloro-4-nitrophenyl)-1-piperazinyl](5-methyl-3-phenyl-4-isoxazolyl)-
- CAS:341001-38-5
- MF:C21H19ClN4O4
- Structure:

- Chemical Name:BIX 01294, 2-(Hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6,7-dimethoxy-N-[1-(phenylmethyl)-4-piperidinyl]-4-quinazolinamine hydrate trihydrochloride
- CAS:935693-62-2
- MF:C28H38N6O2
- Structure:

- Chemical Name:(+)-4-[2-HYDROXY-3-[(1-METHYLETHYL)-AMINO]PROPOXY]BENZENEACETAMIDE
- CAS:56715-13-0
- MF:C14H22N2O3
- Structure:

- Chemical Name:4-Hydroxyisophthalic acid
- CAS:636-46-4
- MF:C8H6O5
- Structure:

- Chemical Name:(5Z,7E,22E)-9,10-Seco-26,27-cyclo-1α,3β-dihydroxycholesta-5,7,10(19),22-tetren-24-one
- CAS:126860-83-1
- MF:C27H38O3
- Structure:

- Chemical Name:ENIPORIDE
- CAS:176644-21-6
- MF:C14H16N4O3S
- Structure:

- Chemical Name:Tavaborole
- CAS:174671-46-6
- MF:C7H6BFO2
- Structure:

- Chemical Name:N-(4-CHLOROBENZYL)-S-[3-(4(5)-IMIDAZOLYL)PROPYL]ISOTHIOUREA
- CAS:145231-35-2
- MF:C14H17ClN4S.2BrH
- Structure:

- Chemical Name:SNS-032
- CAS:345627-92-1
- MF:2C17H24N4O2S2.C4H6O6
- Structure:

- Chemical Name:N-[4-[(6,7-Dimethoxy-4-quinolinyl)oxy]-2-methoxyphenyl]-N'-[1-(2-thiazolyl)ethyl]urea
- CAS:623142-96-1
- MF:C24H24N4O5S
- Structure:

- Chemical Name:Z-Vad-fmk, non-methylated
- CAS:161401-82-7
- MF:C21H28FN3O7
- Structure:

- Chemical Name:BMS-690514
- CAS:859853-30-8
- MF:C19H24N6O2
- Structure:

- Chemical Name:CHIR 98014
- CAS:556813-39-9
- MF:C20H17Cl2N9O2
- Structure:

- Chemical Name:(3aR,4S,7aR)-Octahydro-4-hydroxy-4-[2-(3-methylphenyl)ethynyl]-1H-indole-1-carboxylic acid methyl ester
- CAS:543906-09-8
- MF:C19H23NO3
- Structure:

- Chemical Name:4-Hydroxy-N-[4-methoxy-7-(4-morpholinyl)-2-benzothiazolyl]-4-methyl-1-piperidinecarboxamide
- CAS:870070-55-6
- MF:C19H26N4O4S
- Structure:

- Chemical Name:JNJ-40411813
- CAS:1127498-03-6
- MF:C20H25ClN2O
- Structure:

- Chemical Name:(2R)-3-Cyclopentyl-2-[4-(methanesulfonyl)phenyl]-N-(thiazol-2-yl)propionamide
- CAS:300353-13-3
- MF:C18H22N2O3S2
- Structure:

- Chemical Name:Crisaborole
- CAS:906673-24-3
- MF:C14H10BNO3
- Structure:

- Chemical Name:GLYX 13
- CAS:117928-94-6
- MF:C18H31N5O6
- Structure:

- Chemical Name:N-[2-(Benzoylamino)-6-benzothiazolyl]tricyclo[3.3.1.13,7]decane-1-carboxamide
- CAS:362003-83-6
- MF:C25H25N3O2S
- Structure:

- Chemical Name:(2R)-1-(Phenylmethyl)-N-[3-(spiro[isobenzofuran-1(3H),4'-piperidin]-1-yl)propyl-2-pyrrolidinecarboxamide
- CAS:475150-69-7
- MF:C27H35N3O2
- Structure:

- Chemical Name:Piperidine-3-carboxylic acid [5-chloro-4-(5-fluoro-2-methoxy-phenyl)-pyridin-2-yl]-amide
- CAS:1269815-17-9
- MF:C18H19ClFN3O2
- Structure:

- Chemical Name:Vicriviroc Malate
- CAS:541503-81-5
- MF:C32H44F3N5O7
- Structure:

- Chemical Name:(S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-carboxaMide
- CAS:1038915-64-8
- MF:C19H20N4O
- Structure:

- Chemical Name:KH CB19
- CAS:1354037-26-5
- MF:C15H13Cl2N3O2
- Structure:

- Chemical Name:BS-181 hydrochloride
- CAS:1092443-52-1
- MF:C22H32N6
- Structure:

- Chemical Name:SC 66
- CAS:871361-88-5
- MF:C18H16N2O
- Structure:

- Chemical Name:TTP 22
- CAS:329907-28-0
- MF:C16H14N2O2S2
- Structure:

- Chemical Name:EMD 534085
- CAS:858668-07-2
- MF:C25H31F3N4O2
- Structure:

- Chemical Name:3-Quinolinecarboxylic acid, 8-cyano-1-cyclopropyl-6-fluoro-7-[(4aS,7aS)-hexahydropyrrolo[3,4-b]-1,4-oxazin-6(2H)-yl]-1,4-dihydro-4-oxo-
- CAS:209342-40-5
- MF:C20H19FN4O4
- Structure:

- Chemical Name:(2E)-3-(4'-Hydroxy-3'-tricyclo[3.3.1.13,7]dec-1-yl[1,1'-biphenyl]-4-yl)-2-propenoic acid
- CAS:496868-77-0
- MF:C25H26O3
- Structure:

- Chemical Name:6-Chloro-2-methyl-4-phenyl-alpha-propyl-3-quinolineacetic acid
- CAS:957890-42-5
- MF:C21H20ClNO2
- Structure:

- Chemical Name:[2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl](propyl)(4,5,6,7-tetrahydrobenzothiazol-6-yl)amine
- CAS:1148156-63-1
- MF:C23H34N4OS
- Structure:

- Chemical Name:4-(3-(2H-1,2,3-Triazo-2-yl)phenylaMino)-2-((1R,2S)-2-aMinocyclohexylaMino) pyriMidine-5-carboxaMide
- CAS:1370261-96-3
- MF:C19H23N9O
- Structure:

- Chemical Name:BenzaMide, N-[3-[1,4-dihydro-1-Methyl-7-[(6-Methyl-3-pyridinyl)aMino]-2-oxopyriMido[4,5-d]pyriMidin-3(2H)-yl]-4-Methylphenyl]-3-(trifluoroMethyl)-
- CAS:839706-07-9
- MF:C28H24F3N7O2
- Structure:

- Chemical Name:BS194
- CAS:1092443-55-4
- MF:C20H27N5O3
- Structure:

- Chemical Name:Quinoxaline, 6-[3-(6-Methyl-2-pyridinyl)-1H-pyrazol-4-yl]-
- CAS:746667-48-1
- MF:C17H13N5
- Structure:

- Chemical Name:CarbaMiMidothioic acid, 3-cyanopropyl ester, hydrochloride (1:1)
- CAS:66592-89-0
- MF:C5H10ClN3S
- Structure:

- Chemical Name:ABC294640
- CAS:915385-81-8
- MF:C23H25ClN2O
- Structure:

- Chemical Name:Omadacycline
- CAS:389139-89-3
- MF:C29H40N4O7
- Structure:

- Chemical Name:AS601245
- CAS:345987-15-7
- MF:C20H16N6S
- Structure:

- Chemical Name:AZ-505
- CAS:1035227-44-1
- MF:C31H39Cl2F3N4O6
- Structure:

- Chemical Name:AZD7545
- CAS:252017-04-2
- MF:C19H18ClF3N2O5S
- Structure:

- Chemical Name:BIX-02565
- CAS:1311367-27-7
- MF:C26H30N6O2
- Structure:

- Chemical Name:BMS-538203
- CAS:543730-41-2
- MF:C12H12FNO5
- Structure:

- Chemical Name:CC0651
- CAS:1319207-44-7
- MF:C20H21Cl2NO6
- Structure:

- Chemical Name:CS 7017
- CAS:223132-38-5
- MF:C27H28Cl2N4O4S
- Structure:

- Chemical Name:Ketone Ester
- CAS:1208313-97-6
- MF:C8H16O4
- Structure:

- Chemical Name:NVP-QAV-572
- CAS:957209-68-6
- MF:C17H19F2N7O3S2
- Structure:

- Chemical Name:Nirogacestat
- CAS:1290543-63-3
- MF:C27H41F2N5O
- Structure:

- Chemical Name:ST 2825
- CAS:894787-30-5
- MF:C27H28Cl2N4O5S
- Structure:

- Chemical Name:TG 100572 (Hydrochloride)
- CAS:867331-64-4
- MF:C26H27Cl2N5O2
- Structure:

- Chemical Name:Saxagliptin hydrochloride
- CAS:709031-78-7
- MF:C18H25N3O2.HCl
- Structure:

- Chemical Name:N-(2-(4'-cyanobiphenyl-4-yl)propyl)propane-2-sulfonaMide
- CAS:211311-95-4
- MF:C19H22N2O2S
- Structure:

- Chemical Name:CID-2011756,5-(3-chlorophenyl)-N-(4-(MorpholinoMethyl)phenyl)furan-2-carboxaMide
- CAS:638156-11-3
- MF:C22H21ClN2O3
- Structure:

- Chemical Name:Rimegepant
- CAS:1289023-67-1
- MF:C28H28F2N6O3
- Structure:

- Chemical Name:EVP 6124
- CAS:550999-75-2
- MF:C16H17ClN2OS