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Agonist Inhibitors
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- Structure:

- Chemical Name:Afamelanotide acetate
- CAS:1566590-77-9
- MF:C80H115N21O21
- Structure:

- Chemical Name:Saroglitazar (Magnesium)
- CAS:1639792-20-3
- MF:C50H56MgN2O8S2
- Chemical Name:Eloralintide
- CAS:2883634-40-8
- MF:
- Structure:

- Chemical Name:(1R,3S)-5-[2-[(1R,3aR,7aS)-1-[(2R,5S)-5-hydroxy-6-methyl-heptan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-4-methylidene-cyclohexane-1,3-diol
- CAS:93129-94-3
- MF:C27H46O4
- Structure:

- Chemical Name:1 NM-PP1
- CAS:221244-14-0
- MF:C20H21N5
- Structure:

- Chemical Name:(E)-1-[(1S)-1-(4-Fluorophenyl)ethyl]-3-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzylidene]piperidin-2-one
- CAS:870843-42-8
- MF:C25H26FN3O2
- Structure:

- Chemical Name:LASOFOXIFENE HCL
- CAS:190791-29-8
- MF:C32H37NO8
- Structure:

- Chemical Name:SAG
- CAS:912545-86-9
- MF:C28H28ClN3OS
- Structure:

- Chemical Name:Coelenterazine
- CAS:55779-48-1
- MF:C26H21N3O3
- Structure:

- Chemical Name:5'-D(ATGAAAATCAGGGTTAGG)-3', SODIUM SALT
- CAS:1047953-91-2
- MF:C19H17Cl3N4O3
- Structure:

- Chemical Name:H-ALA-TYR-PRO-GLY-LYS-PHE-NH2
- CAS:352017-71-1
- MF:C34H48N8O7
- Structure:

- Chemical Name:ML-7 HYDROCHLORIDE
- CAS:110448-33-4
- MF:C15H18ClIN2O2S
- Structure:

- Chemical Name:Sapropterin Hydrochloride
- CAS:69056-38-8
- MF:C9H17Cl2N5O3
- Structure:

- Chemical Name:EFONIDIPINE
- CAS:111011-63-3
- MF:C34H38N3O7P
- Structure:

- Chemical Name:MONASTROL
- CAS:329689-23-8
- MF:C14H16N2O3S
- Structure:

- Chemical Name:3-[3-[N-(2-CHLORO-3-TRIFLUOROMETHYLBENZYL)-(2,2-DIPHENYLETHYL)AMINO]PROPYLOXY]PHENYLACETIC ACID HYDROCHLORIDE
- CAS:405911-09-3
- MF:C33H31ClF3NO3
- Structure:

- Chemical Name:ORITAVANCIN
- CAS:171099-57-3
- MF:C86H97Cl3N10O26
- Structure:

- Chemical Name:OTAVA-BB 7070707015
- CAS:934593-90-5
- MF:C26H29NO5
- Structure:

- Chemical Name:(2-METHOXY-5-[2-(2,4,6-TRIMETHOXY-PHENYL)-ETHENESULFONYLMETHYL]-PHENYLAMINO)-ACETIC ACID, SODIUM SALT
- CAS:592542-59-1
- MF:C21H25NO8S
- Structure:

- Chemical Name:BIBF-1120
- CAS:928326-83-4
- MF:C31H33N5O4
- Structure:

- Chemical Name:ONO-AE3-208
- CAS:402473-54-5
- MF:C24H21FN2O3
- Structure:

- Chemical Name:(R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Z)-2-butenedioate
- CAS:179386-44-8
- MF:C15H17N3O5
- Structure:

- Chemical Name:3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole
- CAS:851776-28-8
- MF:C7H8N6
- Structure:

- Chemical Name:LX-1606 Hippurate
- CAS:1033805-22-9
- MF:C27H26ClF3N6O3
- Structure:

- Chemical Name:Doravirine
- CAS:1338225-97-0
- MF:C17H11ClF3N5O3
- Structure:

- Chemical Name:AZ-23
- CAS:915720-21-7
- MF:C17H19ClFN7O
- Structure:

- Chemical Name:3--Phenyl-N-(2,2,2-trichloro-1-((((4-chlorophenyl)amino)carbonothioyl)amino)ethyl)acrylamide
- CAS:1164470-53-4
- MF:C18H15Cl4N3OS
- Structure:

- Chemical Name:2-[(1-Methylpropyl)dithio]-1H-imidazole
- CAS:141400-58-0
- MF:C7H12N2S2
- Structure:

- Chemical Name:4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2,4-dihydro-5-[(5-nitro-2-thiazolyl)thio]-3H-1,2,4-triazol-3-one
- CAS:883065-90-5
- MF:C13H9N5O5S2
- Structure:

- Chemical Name:BMS-599626
- CAS:873837-23-1
- MF:C27H28ClFN8O3
- Structure:

- Chemical Name:N-[2-Fluoro-5-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]amino]phenyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
- CAS:319460-94-1
- MF:C26H22FN7O
- Structure:

- Chemical Name:Saxagliptin hydrate
- CAS:945667-22-1
- MF:C18H27N3O3
- Structure:

- Chemical Name:KX2-391
- CAS:1038395-65-1
- MF:C20H21ClN4O
- Structure:

- Chemical Name:5-Phenyl-1,2,5-thiadiazolidin-3-one 1,1-dioxide
- CAS:612530-44-6
- MF:C8H8N2O3S
- Structure:

- Chemical Name:VU 0357017 hydrochloride
- CAS:1135242-13-5
- MF:C18H28ClN3O3
- Structure:

- Chemical Name:N-[2-[[(2,3-Difluorophenyl)methyl]thio]-6-[[(1S,2R)-2,3-dihydroxy-1-methylpropyl]amino]-4-pyrimidinyl]-1-azetidinesulfonamide
- CAS:1204707-73-2
- MF:C18H23F2N5O4S2
- Structure:

- Chemical Name:Azilsartan kaMedoxoMil
- CAS:863031-24-7
- MF:C30H25KN4O8
- Structure:

- Chemical Name:Nortadalafil
- CAS:171596-36-4
- MF:C21H17N3O4
- Structure:

- Chemical Name:(R)-XL518
- CAS:934660-94-3
- MF:C21H21F3IN3O2
- Structure:

- Chemical Name:AM-679
- CAS:1206880-66-1
- MF:C40H44N4O5S
- Structure:

- Chemical Name:SMER 28
- CAS:307538-42-7
- MF:C11H10BrN3
- Structure:

- Chemical Name:(RS)-4-(3-MethylaMino-1-thiophen-2-yl-propyl)-naphthalen-1-ol
- CAS:949095-98-1
- MF:C18H19NOS
- Structure:

- Chemical Name:NSC-348884
- CAS:81624-55-7
- MF:C38H40N10
- Structure:

- Chemical Name:N-2-Biphenylyl-7-nitro-2,1,3-benzoxadiazol-4-aMine
- CAS:413611-93-5
- MF:C18H12N4O3
- Structure:

- Chemical Name:(1,3-Benzothiazol-2-yl)[2-[[4-[(morpholin-4-yl)methyl]benzyl]oxy]pyrimidin-4-yl]acetonitrile
- CAS:848344-36-5
- MF:C25H23N5O2S
- Structure:

- Chemical Name:2-Methyl-5-(1-methylethyl)-2,5-cyclohexadiene-1,4-dione 1-[O-(2-methylbenzoyl)oxime]
- CAS:321688-88-4
- MF:C18H19NO3
- Structure:

- Chemical Name:GAP 26
- CAS:197250-15-0
- MF:C70H107N19O19S
- Structure:

- Chemical Name:GNE-490
- CAS:1033739-92-2
- MF:C18H22N6O2S
- Structure:

- Chemical Name:BEZ235 (Tosylate)
- CAS:1028385-32-1
- MF:C37H31N5O4S
- Structure:

- Chemical Name:Daun02
- CAS:290304-24-4
- MF:C41H44N2O20
- Structure:

- Chemical Name:I2906
- CAS:331963-29-2
- MF:C25H37N3O4
- Structure:

- Chemical Name:NBD-556
- CAS:333353-44-9
- MF:C17H24ClN3O2
- Structure:

- Chemical Name:D3263 HCl salt
- CAS:1008763-54-9
- MF:C21H32ClN3O3
- Structure:

- Chemical Name:Umeclidinium bromide
- CAS:869113-09-7
- MF:C29H34BrNO2
- Structure:

- Chemical Name:4-IsoxazolecarboxaMide, 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-diMethyl-
- CAS:1197300-24-5
- MF:C18H14Cl2N2O2
- Structure:

- Chemical Name:A-443654
- CAS:552325-16-3
- MF:C24H23N5O
- Structure:

- Chemical Name:LeterMovir
- CAS:917389-32-3
- MF:C29H28F4N4O4
- Structure:

- Chemical Name:AP1903
- CAS:195514-63-7
- MF:C78H98N4O20
- Structure:

- Chemical Name:Bavisant
- CAS:929622-08-2
- MF:C19H27N3O2
- Structure:

- Chemical Name:CHR-6494
- CAS:1333377-65-3
- MF:C16H16N6
- Structure:

- Chemical Name:DG 051 (HCl salt)
- CAS:929915-58-2
- MF:C21H25Cl2NO4
- Structure:

- Chemical Name:Elagolix Sodium
- CAS:832720-36-2
- MF:C32H29F5N3NaO5
- Structure:

- Chemical Name:EMD638683
- CAS:1181770-72-8
- MF:C18H18F2N2O4
- Structure:

- Chemical Name:N6022
- CAS:1208315-24-5
- MF:C24H22N4O3
- Structure:

- Chemical Name:SB-674042
- CAS:483313-22-0
- MF:C24H21FN4O2S
- Structure:

- Chemical Name:SQ 109
- CAS:502487-67-4
- MF:C22H38N2
- Structure:

- Chemical Name:UNC0321
- CAS:1238673-32-9
- MF:C27H45N7O3
- Structure:

- Chemical Name:tiraseMtiv (CK-2017357)
- CAS:1005491-05-3
- MF:C12H14N4O
- Structure:

- Chemical Name:ARRY-520 (R enantioMer)
- CAS:885060-08-2
- MF:C20H22F2N4O2S
- Structure:

- Chemical Name:MK8245 Trifluoroacetate
- CAS:1415559-41-9
- MF:C19H17BrF4N6O6
- Structure:

- Chemical Name:VUF11207
- CAS:1378524-41-4
- MF:C27H35FN2O4
- Structure:

- Chemical Name:Bexagliflozin
- CAS:1118567-05-7
- MF:C24H29ClO7
- Structure:

- Chemical Name:LY2801653
- CAS:1206799-15-6
- MF:C30H22F2N6O3
- Structure:

- Chemical Name:LGD-4033
- CAS:1165910-22-4
- MF:C14H12F6N2O
- Structure:

- Chemical Name:1-(4-AMino-phenyl)-3-(4-tert-butyl-benzoyl)-thiourea
- CAS:1011301-27-1
- MF:C18H21N3OS
- Structure:

- Chemical Name:RRX-001
- CAS:925206-65-1
- MF:C5H6BrN3O5
- Structure:

- Chemical Name:PST2286
- CAS:26629-41-4
- MF:C23H34O5
- Structure:

- Chemical Name:A 438079 (hydrochloride)
- CAS:899431-18-6
- MF:C13H10Cl3N5
- Structure:

- Chemical Name:Bavisant (dihydrochloride)
- CAS:929622-09-3
- MF:C19H28ClN3O2
- Structure:

- Chemical Name:(S)-2-(1-((2-aMino-9H-purin-6-yl)aMino)ethyl)-5-Methyl-3-(o-tolyl)quinazolin-4(3H)-one hydrochloride
- CAS:1431697-78-7
- MF:C23H23ClN8O
- Structure:

- Chemical Name:Delafloxacin meglumine
- CAS:352458-37-8
- MF:C18H12ClF3N4O4.C7H17NO5
- Structure:

- Chemical Name:GS9620
- CAS:1228585-88-3
- MF:C22H30N6O2
- Structure:

- Chemical Name:Kalydeco hydrate
- CAS:1134822-07-3
- MF:C24H30N2O4
- Structure:

- Chemical Name:MethylproaMine
- CAS:188247-01-0
- MF:C28H31N7
- Structure:

- Chemical Name:MLN-120B
- CAS:783348-36-7
- MF:C19H15ClN4O2
- Structure:

- Chemical Name:RAS-2410 hydrochloride
- CAS:1187075-34-8
- MF:C16H20ClN3O4S
- Structure:

- Chemical Name:VcMMAD
- CAS:1401963-17-4
- MF:C70H104N12O14S
- Structure:

- Chemical Name:ARN-2966
- CAS:102212-26-0
- MF:C12H12N2O
- Structure:

- Chemical Name:Auristatin F
- CAS:163768-50-1
- MF:C40H67N5O8
- Structure:

- Chemical Name:PF-4989216
- CAS:1276553-09-3
- MF:C18H13FN6OS
- Structure:

- Chemical Name:PDK1 Inhibitor
- CAS:850717-64-5
- MF:C15H14N4O2
- Structure:

- Chemical Name:2-Naphthalenecarboxylic acid, 3-hydroxy-, 2-[(2,4,5-trihydroxyphenyl)Methylene]hydrazide
- CAS:1256493-34-1
- MF:C18H14N2O5
- Structure:

- Chemical Name:CCT 244747
- CAS:1404095-34-6
- MF:C20H24N8O2
- Structure:

- Chemical Name:Cort-108297
- CAS:1018679-79-2
- MF:C26H25F4N3O3S
- Structure:

- Chemical Name:(S)-2-[4-(4-Chloro-phenyl)-2,3,9-triMethyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulen-6-yl]-acetaMide
- CAS:202591-23-9
- MF:C19H18ClN5OS
- Structure:

- Chemical Name:NISOXETINE HYDROCHLORIDE
- CAS:57754-86-6
- MF:C17H22ClNO2
- Structure:

- Chemical Name:N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide
- CAS:942206-85-1
- MF:C28H32Cl2N4O6S2
- Structure:

- Chemical Name:K145
- CAS:1309444-75-4
- MF:C18H24N2O3S
- Structure:

- Chemical Name:AP20187
- CAS:195514-80-8
- MF:C82H107N5O20
- Structure:

- Chemical Name:2 - (4 - Methylphenyl) - 1,2 - benzisothiazol - 3(2H)-one
- CAS:2514-30-9
- MF:C14H11NOS