PF-04781340 is a potent, selective, and CNS penetrant 5-HT2C receptor agonist.
Uses
PF-04781340 is a potent and selective 5-HT2C receptor agonist. PF-04781340 is orally available and have central nervous system penetrant profile[1].
References
[1] Rouquet G, et al. Design, Synthesis, and Evaluation of Tetrasubstituted Pyridines as Potent 5-HT2C Receptor Agonists. ACS Med Chem Lett. 2015 Jan 20;6(3):329-33. DOI:10.1021/ml500507v
