Items	Specifications
Chemical Formula	C25H25N5O4
Molecular Weight	459.5 g/mol
CAS Number	503612-47-3
IUPAC Name	1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide
Appearance	White to off-white powder
Melting Point	235-238°C
Solubility	Soluble in organic solvents, slightly soluble in water
Stability	Stable under recommended storage conditions
Storage	Store in a tightly closed container, in a dry place, at room temperature
Usage	Anticoagulant
Pharmacological Class	Factor Xa inhibitor
Mechanism of Action	Selectively inhibits factor Xa, thereby inhibiting thrombin generation and preventing blood clot formation
Half-Life	Approximately 12 hours in healthy individuals
Route of Administration	Oral
Bioavailability	Approximately 50%
Protein Binding	Approximately 87%
Metabolism	Primarily hepatic metabolism via CYP3A4 and CYP3A5
Excretion	Renal (27%) and fecal (66%)
Dosage Forms	Tablets (2.5 mg, 5 mg)
Onset of Action	Within 3 hours after oral administration
Duration of Action	Approximately 12-24 hours

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