Basic information Safety Related Supplier

ChemicalBook Product Catalog Biochemical Engineering Biochemical Reagents Agonist Inhibitors Rostafuroxin

1/1

Rostafuroxin NEW

$38.00 2mg

$60.00 5mg

$108.00 10mg

Min. Order
Purity99.08%
Cas No156722-18-8
Supply Ability10g
Update time2026-04-14

TargetMol Chemicals Inc.

TargetMol Chemicals Inc.

VIP6Y

United States

United States

show more

Enterprise Verified

Business Bank account Basic Contact Infomation Business Address Trade Company

Chemical Properties

Product Name	Rostafuroxin
CAS No	156722-18-8
EC-No
Min. Order
Purity	99.08%
Supply Ability	10g
Release date	2026/04/14

Product Introduction

Bioactivity

Name	Rostafuroxin
Description	Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.
Kinase Assay	Kinase assay: Activity assays are conducted using Lance Ultra time-resolved fluorescence resonance energy transfer (TR-FRET) technology from Perkin-Elmer. Briefly, 10 ng/mL FLT3 enzyme, a serial diluted G-749, 80 nM substrate of ULight-poly-GT peptide and variable amounts of ATP (8.5 μM to 1088 μM) are mixed in kinase assay buffer (50 mM HEPES pH 7.5, 10 mM MgCl2, 1 mM EGTA, 2 mM DTT and 0.01% Tween-20) and are added to a 384-well OptiPlate-384 in a volume of 10 μL. Kinase reactions are incubated at room temperature for up to 1 h and then stopped by the addition of 5 μL of 10 mM EDTA. A volume of 5 μL of the specific Eu-labeled-anti-phosphopeptide antibody diluted in LANCE Detection Buffer is then added to a final concentration of 2 nM. After 30-minute incubation, assay plates are incubated at 23°C and the LANCE signal is measured on an EnVision Multilabel Reader. Excitation wavelength is set at 320 nm and emission monitored at 615 nm (donor) and 665 nm (acceptor). The IC50 is calculated using nonlinear regression analysis analysis by GradPad Prism 5.
Storage	Shipping with blue ice/Shipping at ambient temperature.
Solubility Information	DMSO : 50 mg/mL (133.51 mM), Sonication is recommended. 10% DMSO+40% PEG300+5% Tween 80+45% Saline : 2 mg/mL (5.34 mM), Sonication is recommended.
Keywords	Tyr845 \| Sodium potassium pump \| RSV-GFP \| RSV \| Rostafuroxin \| Respiratory syncytial virus \| PST-2238 \| PST2238 \| phosphorylation \| Ouabain \| Na+/K+-ATPase \| Na+/K+ ATPase \| Inhibitor \| inhibit \| EGFR \| digitoxigenin \| ATP1A1 \| antihypertensive
Inhibitors Related	Sodium oleate \| Ribavirin \| Permethrin \| Tolbutamide \| Roflumilast \| trans-Aconitic acid \| Phlorizin \| Chlorpropamide \| Perflubron \| 2,3-Butanedione 2-Monoxime \| Revaprazan hydrochloride \| Oleic acid
Related Compound Libraries	Bioactive Compound Library \| Membrane Protein-targeted Compound Library \| Anti-Cancer Clinical Compound Library \| Anti-Viral Compound Library \| Drug Repurposing Compound Library \| Inhibitor Library \| NO PAINS Compound Library \| Orally Active Compound Library \| Clinical Compound Library \| Bioactive Compounds Library Max \| Bioactive Lipid Compound Library \| Anti-Cancer Drug Library

show more

Company Profile Introduction

You may like

Recommended supplier

Send Inquriy